SE0004244D0 - Novel compounds and their use - Google Patents
Novel compounds and their useInfo
- Publication number
- SE0004244D0 SE0004244D0 SE0004244A SE0004244A SE0004244D0 SE 0004244 D0 SE0004244 D0 SE 0004244D0 SE 0004244 A SE0004244 A SE 0004244A SE 0004244 A SE0004244 A SE 0004244A SE 0004244 D0 SE0004244 D0 SE 0004244D0
- Authority
- SE
- Sweden
- Prior art keywords
- novel compounds
- compounds
- serotonin
- ligands
- general formula
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- QZAYGJVTTNCVMB-UHFFFAOYSA-N serotonin Chemical compound C1=C(O)C=C2C(CCN)=CNC2=C1 QZAYGJVTTNCVMB-UHFFFAOYSA-N 0.000 abstract 2
- 102000006902 5-HT2C Serotonin Receptor Human genes 0.000 abstract 1
- 108010072553 5-HT2C Serotonin Receptor Proteins 0.000 abstract 1
- 239000003446 ligand Substances 0.000 abstract 1
- 229940076279 serotonin Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/20—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (25)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0004244A SE0004244D0 (sv) | 2000-11-20 | 2000-11-20 | Novel compounds and their use |
US09/988,966 US6756377B2 (en) | 2000-11-20 | 2001-11-19 | Compounds and their use |
YU39603A YU39603A (sh) | 2000-11-20 | 2001-11-20 | Jedinjenja piperazinilpirazina kao antagonisti serotonin 5-ht2 receptora |
AT01983901T ATE433962T1 (de) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazinverbindungen als antagonisten des serotonin-5-ht2-rezeptors |
MXPA03004391A MXPA03004391A (es) | 2000-11-20 | 2001-11-20 | Compuestos de piperazinilpirazinas como antagonistas del receptor 5-ht2 de serotonina. |
DK01983901T DK1337518T3 (da) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazinforbindelser som antagonister for serotonin-5-HT2-receptoren |
EA200300595A EA005975B1 (ru) | 2000-11-20 | 2001-11-20 | Соединения пиперазинилпиразинов в качестве антагонистов серотонин 5-ht2 рецептора |
PL36098201A PL360982A1 (en) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor |
CNB018192416A CN1227237C (zh) | 2000-11-20 | 2001-11-20 | 作为五羟色胺5-ht2受体拮抗剂的哌嗪基吡嗪化合物 |
AU1529402A AU1529402A (en) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor |
PCT/SE2001/002570 WO2002040457A1 (en) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor |
BR0115436-2A BR0115436A (pt) | 2000-11-20 | 2001-11-20 | Compostos de piperazinilpirazina atuando como antagonistas do receptor 5ht-2 de serotonina |
KR1020037006822A KR100831909B1 (ko) | 2000-11-20 | 2001-11-20 | 세로토닌 5-ht2 수용체의 안타고니스트로서의피페라지닐피라진 화합물 |
CA002428905A CA2428905A1 (en) | 2000-11-20 | 2001-11-20 | PIPERAZINYLPYRAZINE COMPOUNDS FOR USE AS ANTAGONISTS OF THE SEROTONIN 5-HT2 RECEPTOR |
CA2449899A CA2449899C (en) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor |
EP01983901A EP1337518B1 (en) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor |
NZ525699A NZ525699A (en) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazines compounds as antagonists of serotonin 5-HT2 receptor |
JP2002542785A JP4204315B2 (ja) | 2000-11-20 | 2001-11-20 | セロトニン5−ht2レセプターのアンタゴニストとしてのピペラジニルピラジン化合物 |
IL15587501A IL155875A0 (en) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor |
DE60139021T DE60139021D1 (de) | 2000-11-20 | 2001-11-20 | Piperazinylpyrazinverbindungen als antagonisten des serotonin-5-ht2-rezeptors |
ES01983901T ES2328671T3 (es) | 2000-11-20 | 2001-11-20 | Compuestos de piperazilpirazinas como antagonistas del receptor de serotonina 5-ht2. |
IL155875A IL155875A (en) | 2000-11-20 | 2003-05-12 | Piperazinylpirazine compounds as serotonin HT2 - 5 receptor agonists |
NO20032253A NO325321B1 (no) | 2000-11-20 | 2003-05-19 | Piperazinylpyrazinforbindelser, preparat, fremgangsmate for fremstilling samt anvendelse av slike |
ZA200303452A ZA200303452B (en) | 2000-11-20 | 2004-05-06 | Piperaznylpyrazines compounds as antagonists of serotonin 5-HT2 receptor. |
HK04109907A HK1066810A1 (en) | 2000-11-20 | 2004-12-14 | Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0004244A SE0004244D0 (sv) | 2000-11-20 | 2000-11-20 | Novel compounds and their use |
Publications (1)
Publication Number | Publication Date |
---|---|
SE0004244D0 true SE0004244D0 (sv) | 2000-11-20 |
Family
ID=20281885
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE0004244A SE0004244D0 (sv) | 2000-11-20 | 2000-11-20 | Novel compounds and their use |
Country Status (4)
Country | Link |
---|---|
US (1) | US6756377B2 (sv) |
SE (1) | SE0004244D0 (sv) |
YU (1) | YU39603A (sv) |
ZA (1) | ZA200303452B (sv) |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4081542A (en) | 1975-04-21 | 1978-03-28 | Merck & Co., Inc. | Piperazinylpyrazines |
GB9420999D0 (en) | 1994-10-18 | 1994-12-07 | Smithkline Beecham Plc | Novel compounds |
JPH11279159A (ja) | 1998-03-24 | 1999-10-12 | Nippon Soda Co Ltd | 光学活性なピペラジンカルボン酸エステルの製造方法 |
MXPA01011905A (es) | 1999-05-21 | 2004-03-19 | Biovitrum Ab | Compuestos novedosos, su uso y preparacion. |
US6465467B1 (en) * | 1999-05-21 | 2002-10-15 | Biovitrum Ab | Certain aryl-aliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases |
-
2000
- 2000-11-20 SE SE0004244A patent/SE0004244D0/sv unknown
-
2001
- 2001-11-19 US US09/988,966 patent/US6756377B2/en not_active Expired - Fee Related
- 2001-11-20 YU YU39603A patent/YU39603A/sh unknown
-
2004
- 2004-05-06 ZA ZA200303452A patent/ZA200303452B/en unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200303452B (en) | 2004-05-06 |
US20020103204A1 (en) | 2002-08-01 |
YU39603A (sh) | 2006-05-25 |
US6756377B2 (en) | 2004-06-29 |
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