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RU94027580A - Трициклические бензазепиновые антагонисты вазопрессина, способ получения, фармацевтичекая композиция, способ лечения - Google Patents

Трициклические бензазепиновые антагонисты вазопрессина, способ получения, фармацевтичекая композиция, способ лечения

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Publication number
RU94027580A
RU94027580A RU94027580/04A RU94027580A RU94027580A RU 94027580 A RU94027580 A RU 94027580A RU 94027580/04 A RU94027580/04 A RU 94027580/04A RU 94027580 A RU94027580 A RU 94027580A RU 94027580 A RU94027580 A RU 94027580A
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synthesis
vasopressin
treatment
compounds
antagonists
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RU94027580/04A
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English (en)
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RU2149160C1 (ru
Inventor
Д.Олбрайт Джей
Us]
Ф.Рейч Мэрвин
Сам Фук-Вах
Ду Ксюмей
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Американ Цианамид Компани (US)
Американ Цианамид Компани
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Publication of RU2149160C1 publication Critical patent/RU2149160C1/ru

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Abstract

Трициклические соединения общей формулыопределенные здесь, проявляющие антагонистическую активность на Vи/или Vрецепторах и проявляющие антагонистическую по отношению к вазопрессину активность in vivo, способ применения этих соединений при лечении болезней, характеризующихся избыточной реальной водной реабсорбцией, и способ получения таких соединений.

Claims (1)

  1. Трициклические соединения общей формулы
    Figure 00000001

    определенные здесь, проявляющие антагонистическую активность на V1 и/или V2 рецепторах и проявляющие антагонистическую по отношению к вазопрессину активность in vivo, способ применения этих соединений при лечении болезней, характеризующихся избыточной реальной водной реабсорбцией, и способ получения таких соединений.
RU94027580/04A 1993-07-29 1994-07-28 Трициклические производные, способ получения, фармацевтическая композиция, способ ингибирования вазопрессина RU2149160C1 (ru)

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US10000393A 1993-07-29 1993-07-29
US08/100,003 1993-07-29

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RU94027580A true RU94027580A (ru) 1997-05-27
RU2149160C1 RU2149160C1 (ru) 2000-05-20

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