RS62415B1 - Farmaceutski oblici i metode koji se odnose na piridinoilpiperidin 5-ht1f agoniste - Google Patents
Farmaceutski oblici i metode koji se odnose na piridinoilpiperidin 5-ht1f agonisteInfo
- Publication number
- RS62415B1 RS62415B1 RS20211233A RSP20211233A RS62415B1 RS 62415 B1 RS62415 B1 RS 62415B1 RS 20211233 A RS20211233 A RS 20211233A RS P20211233 A RSP20211233 A RS P20211233A RS 62415 B1 RS62415 B1 RS 62415B1
- Authority
- RS
- Serbia
- Prior art keywords
- pyridinoylpiperidine
- compositions
- methods related
- ht1f agonists
- ht1f
- Prior art date
Links
- 239000000556 agonist Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- YSWVIKAWHDUJFE-UHFFFAOYSA-N piperidin-1-yl(pyridin-2-yl)methanone Chemical compound C=1C=CC=NC=1C(=O)N1CCCCC1 YSWVIKAWHDUJFE-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201662430662P | 2016-12-06 | 2016-12-06 | |
EP17829372.6A EP3551617B1 (en) | 2016-12-06 | 2017-12-05 | Compositions and methods related to pyridinoylpiperidine 5-ht1f agonists |
PCT/US2017/064652 WO2018106657A1 (en) | 2016-12-06 | 2017-12-05 | Compositions and methods related to pyridinoylpiperidine 5-ht1f agonists |
Publications (1)
Publication Number | Publication Date |
---|---|
RS62415B1 true RS62415B1 (sr) | 2021-10-29 |
Family
ID=60972336
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RS20211233A RS62415B1 (sr) | 2016-12-06 | 2017-12-05 | Farmaceutski oblici i metode koji se odnose na piridinoilpiperidin 5-ht1f agoniste |
Country Status (38)
Country | Link |
---|---|
US (1) | US11053214B2 (sr) |
EP (1) | EP3551617B1 (sr) |
JP (4) | JP2020500936A (sr) |
KR (3) | KR20210102497A (sr) |
CN (3) | CN115385893A (sr) |
AU (1) | AU2017373784B2 (sr) |
BR (1) | BR112019010934A2 (sr) |
CA (1) | CA3043772C (sr) |
CL (1) | CL2019001426A1 (sr) |
CO (1) | CO2019005290A2 (sr) |
CR (1) | CR20190251A (sr) |
CY (1) | CY1124540T1 (sr) |
DK (1) | DK3551617T3 (sr) |
DO (1) | DOP2019000139A (sr) |
EA (1) | EA201991112A1 (sr) |
EC (1) | ECSP19040190A (sr) |
ES (1) | ES2889476T3 (sr) |
HR (1) | HRP20211557T1 (sr) |
HU (1) | HUE056820T2 (sr) |
IL (1) | IL266598B2 (sr) |
JO (1) | JOP20190129B1 (sr) |
LT (1) | LT3551617T (sr) |
MA (1) | MA52920B1 (sr) |
MD (1) | MD3551617T2 (sr) |
MX (2) | MX2019006520A (sr) |
MY (1) | MY196855A (sr) |
NZ (1) | NZ752906A (sr) |
PE (2) | PE20241297A1 (sr) |
PH (1) | PH12019501252B1 (sr) |
PL (1) | PL3551617T3 (sr) |
PT (1) | PT3551617T (sr) |
RS (1) | RS62415B1 (sr) |
SI (1) | SI3551617T1 (sr) |
TN (1) | TN2019000174A1 (sr) |
TW (1) | TWI671290B (sr) |
UA (1) | UA124433C2 (sr) |
WO (1) | WO2018106657A1 (sr) |
ZA (1) | ZA201903449B (sr) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI826514B (zh) | 2018-09-04 | 2023-12-21 | 美商美國禮來大藥廠 | 用於預防偏頭痛之拉米迪坦(lasmiditan)長期夜間投藥 |
TWI776175B (zh) | 2019-07-09 | 2022-09-01 | 美商美國禮來大藥廠 | 大規模製備2,4,6-三氟-n-[6-(1-甲基-哌啶-4-羰基)-吡啶-2-基]-苯甲醯胺半琥珀酸鹽的方法及中間體,以及2,4,6-三氟-n-[6-(1-甲基-哌啶-4-羰基)-吡啶-2-基]-苯甲醯胺醋酸鹽之製備 |
CN111004214B (zh) * | 2019-11-22 | 2021-06-08 | 广东东阳光药业有限公司 | 吡啶酰基哌啶衍生物及其用途 |
BR112023022680A2 (pt) | 2021-05-07 | 2024-01-23 | Lilly Co Eli | Composições com sabor mascarado de hemissuccinato de 2,4,6-trifluoro-n-[6-(1-metil-piperidin-4-carbonil)-piridin-2-il]-benzamida, comprimido desintegrante oralmente compreendendo o mesmo, seus usos, e processo para fabricação de comprimido |
CN116270505A (zh) * | 2021-12-20 | 2023-06-23 | 南京科默生物医药有限公司 | 含半琥珀酸拉司米地坦的口服固体制剂及其3d打印制备技术 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5023252A (en) | 1985-12-04 | 1991-06-11 | Conrex Pharmaceutical Corporation | Transdermal and trans-membrane delivery of drugs |
US5011472A (en) | 1988-09-06 | 1991-04-30 | Brown University Research Foundation | Implantable delivery system for biological factors |
TWI263497B (en) | 2002-03-29 | 2006-10-11 | Lilly Co Eli | Pyridinoylpiperidines as 5-HT1F agonists |
US20060178349A1 (en) | 2005-01-24 | 2006-08-10 | Pozen Inc. | Compositions and therapeutic methods utilizing a combination of a 5-HT1F inhibitor and an NSAID |
US20100256187A1 (en) | 2009-04-02 | 2010-10-07 | Colucid Pharmaceuticals, Inc. | Composition of 2,4,6- trifluoro-n-[6-(1-methyl-piperidin-4-carbonyl)-pyridin-2-yl]-benzamide |
US8697876B2 (en) | 2010-04-02 | 2014-04-15 | Colucid Pharmaceuticals, Inc. | Compositions and methods of synthesis of pyridinolypiperidine 5-HT1F agonists |
WO2012163365A1 (en) | 2011-06-01 | 2012-12-06 | Concit Pharma Aps | Combinations of serotonin receptor agonists for treatment of movement disorders |
WO2018010345A1 (zh) | 2016-07-15 | 2018-01-18 | 杭州领业医药科技有限公司 | 一种受体激动剂的晶型及其制备方法和药物组合物 |
TWI754772B (zh) | 2017-09-06 | 2022-02-11 | 美商美國禮來大藥廠 | 用於治療偏頭痛之拉米迪坦(lasmiditan)與cgrp拮抗劑之組合療法 |
-
2017
- 2017-12-05 US US16/467,208 patent/US11053214B2/en active Active
- 2017-12-05 PT PT17829372T patent/PT3551617T/pt unknown
- 2017-12-05 JO JOP/2019/0129A patent/JOP20190129B1/ar active
- 2017-12-05 CR CR20190251A patent/CR20190251A/es unknown
- 2017-12-05 IL IL266598A patent/IL266598B2/en unknown
- 2017-12-05 KR KR1020217025499A patent/KR20210102497A/ko not_active Ceased
- 2017-12-05 MY MYPI2019003189A patent/MY196855A/en unknown
- 2017-12-05 MX MX2019006520A patent/MX2019006520A/es unknown
- 2017-12-05 PE PE2023002466A patent/PE20241297A1/es unknown
- 2017-12-05 SI SI201730881T patent/SI3551617T1/sl unknown
- 2017-12-05 NZ NZ752906A patent/NZ752906A/en unknown
- 2017-12-05 PL PL17829372T patent/PL3551617T3/pl unknown
- 2017-12-05 AU AU2017373784A patent/AU2017373784B2/en active Active
- 2017-12-05 WO PCT/US2017/064652 patent/WO2018106657A1/en active Application Filing
- 2017-12-05 BR BR112019010934A patent/BR112019010934A2/pt not_active Application Discontinuation
- 2017-12-05 UA UAA201905483A patent/UA124433C2/uk unknown
- 2017-12-05 MA MA52920A patent/MA52920B1/fr unknown
- 2017-12-05 JP JP2019551251A patent/JP2020500936A/ja active Pending
- 2017-12-05 MD MDE20191169T patent/MD3551617T2/ro unknown
- 2017-12-05 CA CA3043772A patent/CA3043772C/en active Active
- 2017-12-05 CN CN202210944298.6A patent/CN115385893A/zh active Pending
- 2017-12-05 RS RS20211233A patent/RS62415B1/sr unknown
- 2017-12-05 PE PE2019001167A patent/PE20191134A1/es unknown
- 2017-12-05 PH PH1/2019/501252A patent/PH12019501252B1/en unknown
- 2017-12-05 ES ES17829372T patent/ES2889476T3/es active Active
- 2017-12-05 LT LTEPPCT/US2017/064652T patent/LT3551617T/lt unknown
- 2017-12-05 DK DK17829372.6T patent/DK3551617T3/da active
- 2017-12-05 EA EA201991112A patent/EA201991112A1/ru unknown
- 2017-12-05 KR KR1020227046438A patent/KR20230008257A/ko not_active Ceased
- 2017-12-05 CN CN202210944373.9A patent/CN115385894A/zh active Pending
- 2017-12-05 TW TW106142535A patent/TWI671290B/zh active
- 2017-12-05 MX MX2021014139A patent/MX2021014139A/es unknown
- 2017-12-05 EP EP17829372.6A patent/EP3551617B1/en active Active
- 2017-12-05 CN CN201780075750.7A patent/CN110291079A/zh active Pending
- 2017-12-05 TN TNP/2019/000174A patent/TN2019000174A1/en unknown
- 2017-12-05 HU HUE17829372A patent/HUE056820T2/hu unknown
- 2017-12-05 KR KR1020197016255A patent/KR20190075130A/ko active Application Filing
- 2017-12-05 HR HRP20211557TT patent/HRP20211557T1/hr unknown
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2019
- 2019-05-23 CO CONC2019/0005290A patent/CO2019005290A2/es unknown
- 2019-05-27 CL CL2019001426A patent/CL2019001426A1/es unknown
- 2019-05-30 ZA ZA2019/03449A patent/ZA201903449B/en unknown
- 2019-05-30 DO DO2019000139A patent/DOP2019000139A/es unknown
- 2019-06-06 EC ECSENADI201940190A patent/ECSP19040190A/es unknown
-
2021
- 2021-09-22 JP JP2021153729A patent/JP2022000451A/ja active Pending
- 2021-10-05 CY CY20211100864T patent/CY1124540T1/el unknown
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2023
- 2023-06-26 JP JP2023104019A patent/JP7561240B2/ja active Active
-
2024
- 2024-09-20 JP JP2024163884A patent/JP2024178323A/ja active Pending
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