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RS58024B1 - Biciklični heterociklični derivati kao irak4 inhibitori - Google Patents

Biciklični heterociklični derivati kao irak4 inhibitori

Info

Publication number
RS58024B1
RS58024B1 RS20181355A RSP20181355A RS58024B1 RS 58024 B1 RS58024 B1 RS 58024B1 RS 20181355 A RS20181355 A RS 20181355A RS P20181355 A RSP20181355 A RS P20181355A RS 58024 B1 RS58024 B1 RS 58024B1
Authority
RS
Serbia
Prior art keywords
bicyclic heterocyclyl
irak4 inhibitors
heterocyclyl derivatives
derivatives
irak4
Prior art date
Application number
RS20181355A
Other languages
English (en)
Inventor
Venkateshwar Rao Gummadi
Susanta Samajdar
Original Assignee
Aurigene Discovery Tech Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aurigene Discovery Tech Ltd filed Critical Aurigene Discovery Tech Ltd
Publication of RS58024B1 publication Critical patent/RS58024B1/sr

Links

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
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  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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RS20181355A 2014-01-13 2015-01-12 Biciklični heterociklični derivati kao irak4 inhibitori RS58024B1 (sr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
IN158CH2014 2014-01-13
IN3000CH2014 2014-06-20
EP15735499.4A EP3094329B1 (en) 2014-01-13 2015-01-12 Bicyclic heterocyclyl derivatives as irak4 inhibitors
PCT/IB2015/050217 WO2015104688A1 (en) 2014-01-13 2015-01-12 Bicyclic heterocyclyl derivatives as irak4 inhibitors

Publications (1)

Publication Number Publication Date
RS58024B1 true RS58024B1 (sr) 2019-02-28

Family

ID=53523587

Family Applications (3)

Application Number Title Priority Date Filing Date
RS20181355A RS58024B1 (sr) 2014-01-13 2015-01-12 Biciklični heterociklični derivati kao irak4 inhibitori
RS20240415A RS65437B1 (sr) 2014-01-13 2015-01-12 (r) i (s) enantiomeri n-(5-(3-hidroksipirolidin-1-il)-2-morfolinooksazolo[4,5-b]piridin-6-il)-2-(2-metilpiridin-4-il)oksazol-karboksamida kao inhibitori irak4 za lečenje kancera
RS20210039A RS61448B1 (sr) 2014-01-13 2015-01-12 Način pripreme derivata oksazolo [4,5-b] piridina i tiazolo [4,5-b] piridina kao irak4 inhibitora za lečenje raka

Family Applications After (2)

Application Number Title Priority Date Filing Date
RS20240415A RS65437B1 (sr) 2014-01-13 2015-01-12 (r) i (s) enantiomeri n-(5-(3-hidroksipirolidin-1-il)-2-morfolinooksazolo[4,5-b]piridin-6-il)-2-(2-metilpiridin-4-il)oksazol-karboksamida kao inhibitori irak4 za lečenje kancera
RS20210039A RS61448B1 (sr) 2014-01-13 2015-01-12 Način pripreme derivata oksazolo [4,5-b] piridina i tiazolo [4,5-b] piridina kao irak4 inhibitora za lečenje raka

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US (7) US9732095B2 (sr)
EP (4) EP3466955B1 (sr)
JP (5) JP6479850B2 (sr)
KR (3) KR102574390B1 (sr)
CN (2) CN111362966B (sr)
AU (5) AU2015205374B2 (sr)
BR (1) BR112016016158B1 (sr)
CA (1) CA2935887A1 (sr)
CU (1) CU24389B1 (sr)
CY (2) CY1121433T1 (sr)
DK (3) DK3805233T3 (sr)
EA (2) EA038748B1 (sr)
ES (3) ES2975436T3 (sr)
FI (1) FI3805233T3 (sr)
HK (1) HK1231410A1 (sr)
HR (3) HRP20240489T1 (sr)
HU (3) HUE041926T2 (sr)
IL (7) IL294895B2 (sr)
LT (3) LT3466955T (sr)
MX (1) MX359909B (sr)
MY (1) MY197116A (sr)
NZ (2) NZ760657A (sr)
PH (2) PH12016501344A1 (sr)
PL (3) PL3805233T3 (sr)
PT (3) PT3466955T (sr)
RS (3) RS58024B1 (sr)
SG (2) SG10201811204RA (sr)
SI (3) SI3094329T1 (sr)
SM (3) SMT202400142T1 (sr)
TR (1) TR201815683T4 (sr)
WO (1) WO2015104688A1 (sr)
ZA (2) ZA202007274B (sr)

Families Citing this family (49)

* Cited by examiner, † Cited by third party
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