PT838469E - Derivados de 10,13,15-trioxatriciclo¬9.2.1.1.<9.6>|-pentadecanona processo para a sua preparacao e medicamentos que contem estes compostos - Google Patents
Derivados de 10,13,15-trioxatriciclo¬9.2.1.1.<9.6>|-pentadecanona processo para a sua preparacao e medicamentos que contem estes compostosInfo
- Publication number
- PT838469E PT838469E PT97118000T PT97118000T PT838469E PT 838469 E PT838469 E PT 838469E PT 97118000 T PT97118000 T PT 97118000T PT 97118000 T PT97118000 T PT 97118000T PT 838469 E PT838469 E PT 838469E
- Authority
- PT
- Portugal
- Prior art keywords
- trioxatriciclo
- pentadecanone
- derivatives
- compounds
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Genetics & Genomics (AREA)
- Public Health (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19644195A DE19644195A1 (de) | 1996-10-24 | 1996-10-24 | 10,13,15-Trioxatricyclo[9.2.1.1.·9·.·6·]-pentadecanon-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
PT838469E true PT838469E (pt) | 2002-05-31 |
Family
ID=7809858
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT97118000T PT838469E (pt) | 1996-10-24 | 1997-10-17 | Derivados de 10,13,15-trioxatriciclo¬9.2.1.1.<9.6>|-pentadecanona processo para a sua preparacao e medicamentos que contem estes compostos |
Country Status (27)
Country | Link |
---|---|
US (1) | US5912235A (pt) |
EP (1) | EP0838469B1 (pt) |
JP (1) | JP4175682B2 (pt) |
KR (1) | KR100466495B1 (pt) |
CN (1) | CN1093133C (pt) |
AR (1) | AR009809A1 (pt) |
AT (1) | ATE211745T1 (pt) |
AU (1) | AU726092B2 (pt) |
BR (2) | BR9705157A (pt) |
CA (1) | CA2219311C (pt) |
CZ (1) | CZ291768B6 (pt) |
DE (2) | DE19644195A1 (pt) |
DK (1) | DK0838469T3 (pt) |
DZ (1) | DZ2322A1 (pt) |
ES (1) | ES2170318T3 (pt) |
HK (1) | HK1010885A1 (pt) |
HU (1) | HU222540B1 (pt) |
IL (1) | IL121969A (pt) |
MX (1) | MX9707974A (pt) |
NO (1) | NO308362B1 (pt) |
NZ (1) | NZ328979A (pt) |
PL (1) | PL184693B1 (pt) |
PT (1) | PT838469E (pt) |
RU (1) | RU2181727C2 (pt) |
SK (1) | SK283114B6 (pt) |
UA (1) | UA44310C2 (pt) |
ZA (1) | ZA979059B (pt) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1998023629A1 (fr) * | 1996-11-26 | 1998-06-04 | Chugai Seiyaku Kabushiki Kaisha | Composes de macrolides comportant une chaine a 13 elements, medicament les contenant et leur procede de preparation |
CA2386828C (en) * | 2000-08-17 | 2006-01-24 | The Kitasato Institute | Novel pseudoerythromycin derivatives |
JP2003007917A (ja) * | 2001-06-19 | 2003-01-10 | Sanyo Electric Co Ltd | 回路装置の製造方法 |
US6986882B2 (en) * | 2002-01-17 | 2006-01-17 | Astrazeneca Ab | Therapy for functional dyspepsia |
JP4928261B2 (ja) | 2003-06-18 | 2012-05-09 | トランザイム・ファーマ・インコーポレイテッド | モチリン受容体の大環状拮抗薬 |
GB0611907D0 (en) | 2006-06-15 | 2006-07-26 | Glaxo Group Ltd | Compounds |
US20080312209A1 (en) | 2005-07-12 | 2008-12-18 | Glaxo Group Limited | Piperazine Heteroaryl Derivatives as Gpr38 Agonists |
AU2006274212B2 (en) * | 2005-07-26 | 2011-06-09 | Glaxo Group Limited | Benzylpiperazine derivates and their medical use |
CA2632779A1 (en) * | 2005-12-08 | 2007-06-14 | Pfizer Inc. | Method for demethylating the 3'-dimethylamino group of erythromycin compounds |
ES2344484T3 (es) | 2006-06-28 | 2010-08-27 | Glaxo Group Limited | Derivados de piperazinilo utiles en el tratamiento de enfermedades mediadas por el receptor gpr38. |
WO2008033328A2 (en) | 2006-09-11 | 2008-03-20 | Tranzyme Pharma, Inc. | Macrocyclic antagonists of the motilin receptor for treatment of gastrointestinal dysmotility disorders |
JP5663743B2 (ja) | 2009-02-27 | 2015-02-04 | ラクオリア創薬株式会社 | モチリン受容体作動活性を有するオキシインドール誘導体 |
JP6295247B2 (ja) * | 2013-03-25 | 2018-03-14 | ゼリア新薬工業株式会社 | 食後期の胃運動亢進剤 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3725385A (en) * | 1970-11-02 | 1973-04-03 | Abbott Lab | Process for the demethylation of 3-amino macrolides |
US5106961A (en) * | 1987-05-26 | 1992-04-21 | Eli Lilly And Company | Erythromycin ring-contracted derivatives |
US4920102A (en) * | 1988-04-18 | 1990-04-24 | Eli Lilly And Company | Method for treating gastrointestinal disorders |
DE4200145A1 (de) * | 1992-01-07 | 1993-07-08 | Kali Chemie Pharma Gmbh | 7,10-epoxy-oxacyclododecan-derivate, verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
-
1996
- 1996-10-24 DE DE19644195A patent/DE19644195A1/de not_active Withdrawn
-
1997
- 1997-09-23 AR ARP970104375A patent/AR009809A1/es active IP Right Grant
- 1997-09-29 DZ DZ970172A patent/DZ2322A1/xx active
- 1997-10-01 CZ CZ19973106A patent/CZ291768B6/cs not_active IP Right Cessation
- 1997-10-07 KR KR1019970051470A patent/KR100466495B1/ko not_active IP Right Cessation
- 1997-10-09 ZA ZA9709059A patent/ZA979059B/xx unknown
- 1997-10-14 IL IL12196997A patent/IL121969A/xx not_active IP Right Cessation
- 1997-10-16 MX MX9707974A patent/MX9707974A/es not_active IP Right Cessation
- 1997-10-17 ES ES97118000T patent/ES2170318T3/es not_active Expired - Lifetime
- 1997-10-17 DK DK97118000T patent/DK0838469T3/da active
- 1997-10-17 NZ NZ328979A patent/NZ328979A/xx unknown
- 1997-10-17 DE DE59705964T patent/DE59705964D1/de not_active Expired - Fee Related
- 1997-10-17 HU HU9701660A patent/HU222540B1/hu not_active IP Right Cessation
- 1997-10-17 SK SK1419-97A patent/SK283114B6/sk not_active IP Right Cessation
- 1997-10-17 PT PT97118000T patent/PT838469E/pt unknown
- 1997-10-17 AT AT97118000T patent/ATE211745T1/de not_active IP Right Cessation
- 1997-10-17 EP EP97118000A patent/EP0838469B1/de not_active Expired - Lifetime
- 1997-10-21 US US08/954,891 patent/US5912235A/en not_active Expired - Lifetime
- 1997-10-22 AU AU42788/97A patent/AU726092B2/en not_active Ceased
- 1997-10-22 JP JP28986197A patent/JP4175682B2/ja not_active Expired - Fee Related
- 1997-10-22 CN CN97121157A patent/CN1093133C/zh not_active Expired - Fee Related
- 1997-10-23 PL PL97322802A patent/PL184693B1/pl not_active IP Right Cessation
- 1997-10-23 RU RU97117347/04A patent/RU2181727C2/ru not_active IP Right Cessation
- 1997-10-23 UA UA97105178A patent/UA44310C2/uk unknown
- 1997-10-24 BR BR9705157-8A patent/BR9705157A/pt not_active Application Discontinuation
- 1997-10-24 NO NO974934A patent/NO308362B1/no not_active IP Right Cessation
- 1997-10-24 BR BR9705143-8A patent/BR9705143A/pt active Search and Examination
- 1997-10-24 CA CA002219311A patent/CA2219311C/en not_active Expired - Fee Related
-
1998
- 1998-11-10 HK HK98111873A patent/HK1010885A1/xx not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PT885204E (pt) | Novos derivados de arilglicinamida, processo para a sua preparacao e composicoes farmaceuticas que contem estes compostos | |
BR9707839A (pt) | Primido-Ú5,4-D¾-primidas medicamentos contendo esses compostos sua aplicação e processo para a sua preparação | |
PT101732A (pt) | Novas di-hidrodibenzo<b,f>azepinas substituidas processo para a sua preparacao composicoes farmaceuticas que as contem e utilizacao dos novos compostos na preparacao de composicoes farmaceuticas empregues em doencas do sistema nervoso | |
PT927192E (pt) | Aminoacidos modificados medicamentos contendo estes compostos e processo para a sua preparacao | |
PT99671A (pt) | Processo para a preparacao de heparosanos-n,o-sulfatados e de composicoes farmaceuticas que os contem | |
PT92497A (pt) | Processo para a preparacao de derivados de ureia de dipeptideos inibidores de enzimas, e de composicoes farmaceuticas que os contem | |
BR9801606B1 (pt) | composto, processo para sua preparação, substáncia farmacêutica, uso do composto e processo para a produção de uma substáncia farmacêutica. | |
BR1100850A (pt) | Composto, processo para a preparação de um composto, e, composição farmacêutica | |
PT93094A (pt) | Processo para a preparacao de 1,3-oxatiolanos substituidos e de composicoes farmaceuticas que os contem | |
BR9711328A (pt) | 7Alfa-(epsilon-aminoalquil)-estratrienos processos para a sua prepara-Æo preparados farmaceuticos que contem estes 7 alfa-(epsilon-aminoalquil)- estratrienos bem como seu emprego para a prepara-Æo de medicamentos | |
BR9600821A (pt) | Composto formulação farmacêutica e processo para a preparação de um composto | |
BR9601093A (pt) | Pirido(3,2-E)pirazinoas processo para sua preparação medicamentos processo para sua preparação e utilização | |
BR9602802A (pt) | Derivados de naftaleno processo para a preparação dos mesmos e compostos | |
PT838469E (pt) | Derivados de 10,13,15-trioxatriciclo¬9.2.1.1.<9.6>|-pentadecanona processo para a sua preparacao e medicamentos que contem estes compostos | |
PT88381A (pt) | Processo para a preparacao de novos compostos 3,7-diazabiciclo{3,3,1} nonano, e de composicoes farmaceuticas que contem estes compostos | |
BR9609327A (pt) | Novos derivados de oxazolidinona processos para sua preparação e agentes farmacêuticos que contêm estes compostos | |
BR9202325A (pt) | Composto,processo para a sua preparacao,preparado farmaceutico e processo para a sua preparacao | |
PT909270E (pt) | Processo para a preparacao de 2,4-dihidroxipiridina e de 2,4-dihidroxi-3-nitropiridina | |
BR9711340A (pt) | Composto composi-Æo farmac-utica e processo para preparar um composto | |
BR9303456A (pt) | Compostos,processo para sua preparacao,medicamentos,processo para sua preparacao e emprego | |
PT84828B (pt) | Processo para a preparacao de compostos heterociclicos triciclicos fundidos e de composicoes farmaceuticas que os contem | |
PT864579E (pt) | Sais de bismuto de antibioticos do grupo da moenomicina processo para a sua preparacao sua utilizacao e medicamentos que contem esses sais | |
PT93138A (pt) | Processo para a preparacao de novos compostos derivados da acetamina e de composicoes farmaceuticas que os contem | |
BR9602025A (pt) | Composto composição farmacêutica uso e processo para a preparação de um composto | |
PT842927E (pt) | 3-AMIDO-CROMANILSULFONIL(TIO)-UREIAS PROCESSOS PARA A SUA PREPARACAO SUA UTILIZACAO E COMPOSICOES FARMACêUTICAS QUE AS CONTEM |