PT1334106E - Derivados de imidazole, seu metodo de producao e sua utilizacao - Google Patents

Derivados de imidazole, seu metodo de producao e sua utilizacao

Info

Publication number: PT1334106E
Authority: PT; Portugal
Prior art keywords: production method; imidazole derivatives; imidazole; derivatives; production
Prior art date: 2000-11-17

Application number

PT01982800T

Other languages

English (en)

Inventor

Akihiro Tasaka

Hitaka Takenori

Matsunaga Nobuyuki

Masami Kusaka

Adachi Mari

Aoki Isao

Ojida Akio

Original Assignee

Takeda Pharmaceutical

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-17

Filing date

2001-11-16

Publication date

2006-08-31

2001-11-16 Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical

2006-08-31 Publication of PT1334106E publication Critical patent/PT1334106E/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/28—Antiandrogens
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Urology & Nephrology (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Medicinal Preparation (AREA)

PT01982800T 2000-11-17 2001-11-16 Derivados de imidazole, seu metodo de producao e sua utilizacao PT1334106E (pt)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP2000351780		2000-11-17
JP2001247618		2001-08-17
JP2001336880		2001-11-01

Publications (1)

Publication Number	Publication Date
PT1334106E true PT1334106E (pt)	2006-08-31

Family

ID=27345219

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT01982800T PT1334106E (pt)	2000-11-17	2001-11-16	Derivados de imidazole, seu metodo de producao e sua utilizacao

Country Status (27)

Country	Link
US (1)	US7141598B2 (pt)
EP (2)	EP1681290B9 (pt)
JP (2)	JP3753971B2 (pt)
KR (3)	KR20080002929A (pt)
CN (3)	CN100572363C (pt)
AR (1)	AR034854A1 (pt)
AT (2)	ATE327237T1 (pt)
AU (3)	AU1429602A (pt)
BR (1)	BR0115306B1 (pt)
CA (1)	CA2429133C (pt)
CY (1)	CY1105423T1 (pt)
DE (1)	DE60119963T2 (pt)
DK (1)	DK1334106T3 (pt)
ES (1)	ES2260303T3 (pt)
HK (1)	HK1056168A1 (pt)
HU (1)	HU229408B1 (pt)
IL (2)	IL155624A0 (pt)
MX (1)	MXPA03004347A (pt)
MY (1)	MY134929A (pt)
NO (1)	NO326366B1 (pt)
NZ (1)	NZ526387A (pt)
PE (1)	PE20020596A1 (pt)
PL (1)	PL204934B1 (pt)
PT (1)	PT1334106E (pt)
SI (1)	SI1334106T1 (pt)
TW (1)	TWI306099B (pt)
WO (1)	WO2002040484A2 (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA2472821C (en) *	2002-01-10	2011-05-24	Takeda Chemical Industries, Ltd.	Process for producing fused imidazole compound, and reformatsky reagent in stable form and process for producing the same
WO2004075890A1 (ja) *	2003-02-26	2004-09-10	Takeda Pharmaceutical Company	安定化されたイミダゾール誘導体含有医薬組成物、イミダゾ－ル誘導体の安定化方法
JP4745616B2 (ja) *	2003-02-26	2011-08-10	武田薬品工業株式会社	安定化されたイミダゾール誘導体含有医薬組成物、イミダゾール誘導体の安定化方法
CA2519211A1 (en) *	2003-03-17	2004-09-30	Takeda Pharmaceutical Company Limited	Release control compositions
JP4837895B2 (ja) *	2003-03-17	2011-12-14	武田薬品工業株式会社	放出制御組成物
EP1753749B1 (en) *	2004-05-03	2014-07-30	Janssen Pharmaceutica NV	Novel indole derivatives as selective androgen receptor modulators (sarms)
EP1765777A2 (en) *	2004-05-28	2007-03-28	Speedel Experimenta AG	Bicyclic, nitrogen-containing heterocycles as aromatase inhibitors
WO2006093353A1 (ja)	2005-03-03	2006-09-08	Takeda Pharmaceutical Company Limited	放出制御組成物
GT200600381A (es)	2005-08-25	2007-03-28		Compuestos organicos
TW200804378A (en) *	2005-12-09	2008-01-16	Speedel Experimenta Ag	Organic compounds
ATE473741T1 (de) *	2006-02-10	2010-07-15	Janssen Pharmaceutica Nv	Neue imidazolopyrazolderivate als selektive androgen-rezeptor-modulatoren
TW200804284A (en) *	2006-03-31	2008-01-16	Speedel Experimenta Ag	Process for preparing 6,7-dihydro-5H-imidazo[1,5-a]pyridin-8-one
RU2481107C2 (ru) *	2007-10-29	2013-05-10	Такеда Фармасьютикал Компани Лимитед	Средство для профилактики или лечения рака
JOP20190231A1 (ar) *	2009-01-15	2017-06-16	Incyte Corp	طرق لاصلاح مثبطات انزيم jak و المركبات الوسيطة المتعلقة به
UY33740A (es) *	2010-11-18	2012-05-31	Takeda Pharmaceutical	Método para tratar el cáncer de mama y cáncer de ovarios
MX2013010661A (es)	2011-04-01	2013-10-28	Takeda Pharmaceutical	Preparacion solida.
SG195036A1 (en) *	2011-06-15	2013-12-30	Takeda Pharmaceutical	Production method of imidazole derivatives

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4728645A (en) *	1982-12-21	1988-03-01	Ciba-Geigy Corporation	Substituted imidazo[1,5-A]pyridine derivatives and other substituted bicyclic derivatives, useful as aromatase inhibitors
NZ221729A (en)	1986-09-15	1989-07-27	Janssen Pharmaceutica Nv	Imidazolyl methyl-substituted benzimidazole derivatives and pharmaceutical compositions
NZ224288A (en)	1987-04-22	1989-12-21	Merrell Dow Pharma	17b-(cyclopropylamino)androst-5-en-3b-ol and related compounds and methods using these for treatment of non-humans
US5057521A (en) *	1988-10-26	1991-10-15	Ciba-Geigy Corporation	Use of bicyclic imidazole compounds for the treatment of hyperaldosteronism
US4966898A (en)	1989-08-15	1990-10-30	Merrell Dow Pharmaceuticals Inc.	4-substituted 17β-(cyclopropylamino)androst-5-en-3β-ol and related compounds useful as C17-20 lyase inhibitors
AU659632B2 (en)	1991-03-01	1995-05-25	Electrostatic Technology, Inc.	Powder coating method for producing circuit board laminae and the like
US5457102A (en)	1994-07-07	1995-10-10	Janssen Pharmaceutica, N.V.	Pyrroloimidazolyl and imidazopyridinyl substituted 1H-benzimidazole derivatives
ATE203992T1 (de)	1992-01-27	2001-08-15	Janssen Pharmaceutica Nv	Pyrroloimidazolyl und imidazopyridinyl substituierte 1h-benzimidazolderivate als aromatase inhibitoren
KR100235135B1 (ko)	1992-03-31	2000-01-15	말콤 카터	암치료에 유용한 17-치환된 스테로이드
GB9310635D0 (en)	1993-05-21	1993-07-07	Glaxo Group Ltd	Chemical compounds
CA2170874A1 (en)	1993-09-30	1995-04-06	Minoru Okada	Azole derivative and pharmaceutical composition thereof
AU3846395A (en)	1994-11-07	1996-05-31	Janssen Pharmaceutica N.V.	Compositions comprising carbazoles and cyclodextrins
AU6015796A (en)	1995-06-14	1997-01-15	Yamanouchi Pharmaceutical Co., Ltd.	Fused imidazole derivatives and medicinal composition thereof
US6420375B1 (en)	1997-02-21	2002-07-16	Takeda Chemical Industries, Ltd.	Fused ring compounds, process for producing the same and use thereof
ES2218853T3 (es)	1997-10-02	2004-11-16	Daiichi Pharmaceutical Co., Ltd.	Nuevos compuestos de dihidronaftaleno y procesos para la obtencion de los mismos.
CA2328973A1 (en)	1998-04-23	1999-10-28	Akio Ojida	Naphthalene derivatives, their production and use
PE20010781A1 (es) *	1999-10-22	2001-08-08	Takeda Chemical Industries Ltd	Compuestos 1-(1h-imidazol-4-il)-1-(naftil-2-sustituido)etanol, su produccion y utilizacion

2001
- 2001-11-16 EP EP05077705.1A patent/EP1681290B9/en not_active Expired - Lifetime
- 2001-11-16 ES ES01982800T patent/ES2260303T3/es not_active Expired - Lifetime
- 2001-11-16 CN CNB2005100640723A patent/CN100572363C/zh not_active Expired - Fee Related
- 2001-11-16 US US10/416,986 patent/US7141598B2/en not_active Expired - Lifetime
- 2001-11-16 SI SI200130590T patent/SI1334106T1/sl unknown
- 2001-11-16 AT AT01982800T patent/ATE327237T1/de active
- 2001-11-16 WO PCT/JP2001/010002 patent/WO2002040484A2/en active IP Right Grant
- 2001-11-16 KR KR1020077025704A patent/KR20080002929A/ko not_active Application Discontinuation
- 2001-11-16 MY MYPI20015279A patent/MY134929A/en unknown
- 2001-11-16 IL IL15562401A patent/IL155624A0/xx active IP Right Grant
- 2001-11-16 PE PE2001001147A patent/PE20020596A1/es active IP Right Grant
- 2001-11-16 PL PL362766A patent/PL204934B1/pl unknown
- 2001-11-16 JP JP2001351035A patent/JP3753971B2/ja not_active Expired - Fee Related
- 2001-11-16 DE DE60119963T patent/DE60119963T2/de not_active Expired - Lifetime
- 2001-11-16 NZ NZ526387A patent/NZ526387A/en not_active IP Right Cessation
- 2001-11-16 CA CA002429133A patent/CA2429133C/en not_active Expired - Fee Related
- 2001-11-16 EP EP01982800A patent/EP1334106B1/en not_active Expired - Lifetime
- 2001-11-16 CN CNB018190251A patent/CN1329394C/zh not_active Expired - Fee Related
- 2001-11-16 AR ARP010105365A patent/AR034854A1/es active IP Right Grant
- 2001-11-16 AT AT05077705T patent/ATE533768T1/de active
- 2001-11-16 KR KR1020037006727A patent/KR100725442B1/ko active IP Right Grant
- 2001-11-16 AU AU1429602A patent/AU1429602A/xx active Pending
- 2001-11-16 PT PT01982800T patent/PT1334106E/pt unknown
- 2001-11-16 KR KR1020057018247A patent/KR100809899B1/ko active IP Right Grant
- 2001-11-16 CN CNA200610100666XA patent/CN1900079A/zh active Pending
- 2001-11-16 HU HU0400549A patent/HU229408B1/hu not_active IP Right Cessation
- 2001-11-16 TW TW090128440A patent/TWI306099B/zh not_active IP Right Cessation
- 2001-11-16 BR BRPI0115306-4B1A patent/BR0115306B1/pt not_active IP Right Cessation
- 2001-11-16 DK DK01982800T patent/DK1334106T3/da active
- 2001-11-16 AU AU2002214296A patent/AU2002214296C1/en not_active Ceased
- 2001-11-16 MX MXPA03004347A patent/MXPA03004347A/es active IP Right Grant
2003
- 2003-04-28 IL IL155624A patent/IL155624A/en not_active IP Right Cessation
- 2003-05-16 NO NO20032234A patent/NO326366B1/no not_active IP Right Cessation
- 2003-11-17 HK HK03108376A patent/HK1056168A1/xx not_active IP Right Cessation
2005
- 2005-08-31 JP JP2005252651A patent/JP4427496B2/ja not_active Expired - Fee Related
- 2005-10-18 AU AU2005225035A patent/AU2005225035B2/en not_active Ceased
2006
- 2006-06-26 CY CY20061100867T patent/CY1105423T1/el unknown

Also Published As

Publication number	Publication date
EP1681290A2 (en)	2006-07-19
HU229408B1 (hu)	2013-12-30
EP1681290B9 (en)	2013-06-19
BR0115306B1 (pt)	2013-12-24
IL155624A (en)	2006-12-31
ATE533768T1 (de)	2011-12-15
CN1329394C (zh)	2007-08-01
CN1474819A (zh)	2004-02-11
KR20030048156A (ko)	2003-06-18
ES2260303T3 (es)	2006-11-01
ATE327237T1 (de)	2006-06-15
DE60119963D1 (de)	2006-06-29
NO326366B1 (no)	2008-11-17
WO2002040484A2 (en)	2002-05-23
NO20032234L (no)	2003-07-16
AU2002214296C1 (en)	2006-04-13
EP1334106A2 (en)	2003-08-13
KR20050105287A (ko)	2005-11-03
JP4427496B2 (ja)	2010-03-10
KR20080002929A (ko)	2008-01-04
CA2429133C (en)	2009-08-18
EP1681290B1 (en)	2011-11-16
CN1900079A (zh)	2007-01-24
US20040033935A1 (en)	2004-02-19
AU2005225035A1 (en)	2005-11-10
CA2429133A1 (en)	2002-05-23
AU2002214296B2 (en)	2005-09-29
KR100809899B1 (ko)	2008-03-10
JP2003201282A (ja)	2003-07-18
HUP0400549A3 (en)	2004-09-28
MXPA03004347A (es)	2004-05-04
PL362766A1 (en)	2004-11-02
BR0115306A (pt)	2004-02-10
NO20032234D0 (no)	2003-05-16
AU2005225035B2 (en)	2007-02-22
AR034854A1 (es)	2004-03-24
JP2006045239A (ja)	2006-02-16
AU1429602A (en)	2002-05-27
HUP0400549A2 (hu)	2004-06-28
JP3753971B2 (ja)	2006-03-08
KR100725442B1 (ko)	2007-06-07
CY1105423T1 (el)	2010-04-28
MY134929A (en)	2008-01-31
EP1681290A3 (en)	2006-07-26
TWI306099B (en)	2009-02-11
US7141598B2 (en)	2006-11-28
CN1680336A (zh)	2005-10-12
DE60119963T2 (de)	2006-10-05
PL204934B1 (pl)	2010-02-26
EP1334106B1 (en)	2006-05-24
DK1334106T3 (da)	2006-09-18
SI1334106T1 (sl)	2006-10-31
WO2002040484A3 (en)	2002-09-26
CN100572363C (zh)	2009-12-23
NZ526387A (en)	2004-02-27
HK1056168A1 (en)	2004-02-06
PE20020596A1 (es)	2002-08-13
IL155624A0 (en)	2003-11-23

Publication	Publication Date	Title
ITRM20000228A0 (it)	2000-04-28	Scidula multistrato e procedimento per la sua produzione.
IS6662A (is)	2002-12-19	Imídasól afleiður
ATE360620T1 (de)	2007-05-15	Imidazolderivate
NO20024170D0 (no)	2002-09-02	Forminsket, nållös injektor
DK1292604T3 (da)	2009-06-15	2-Aminocarbonyl-9H-purinderivater
NO20021449D0 (no)	2002-03-22	Substituerte 2-tio-3,5-dicyano-4-aryl-6-aminopyridiner og anvendelse derav
PT1334106E (pt)	2006-08-31	Derivados de imidazole, seu metodo de producao e sua utilizacao
PT1303521E (pt)	2005-05-31	Derivados de tetra-hidro-heterocicloazepinil-pirimidina
FR2806720B1 (fr)	2006-12-08	Derives de 2,2,6,6-diethyl-dimethyl-1-alcoxypiperidines et 1-oxydes correspondants
ATE298332T1 (de)	2005-07-15	Decahydro-isochinolinderivate
DK1280809T3 (da)	2005-11-07	Antitumorecteinascidinderivater
DK1480983T3 (da)	2006-03-27	Heteroarylsubstituerede 2-pyridinyl- og 2-pyrimidinyl- 6,7,8,9-tetrahydropyrimido[1,2a]pyrimidin-4-onderivater
IT1321015B1 (it)	2003-12-18	Pacchetto di sigarette e metodo per la sua realizzazione.
PT1043307E (pt)	2003-10-31	Derivados de 3-amino-3-arilpropan-1-ol sua producao e utilizacao
IS2174B (is)	2006-11-15	Setnar fenýl-píperasín afleiður, framleiðsla þeirra og notkun
AR028602A1 (es)	2003-05-14	Derivados de pirrol
AR028282A1 (es)	2003-04-30	Derivados de aminofenil pirimidona
DK1322593T3 (da)	2004-10-11	O-substituerede-6-methyl-tramadol-derivater
FI20000194A0 (fi)	2000-01-31	Menetelmä kaupankäynnissä
DK1246791T3 (da)	2005-02-14	Aminomethyl-phenyl-cyklohexanonderivater
NO20023298L (no)	2002-09-06	Nye imidazolderivater
DE60117096D1 (de)	2006-04-20	Dihydroindol- und tetrahydrochinolinderivate
PT1043306E (pt)	2004-08-31	Derivados de 3-amino-3-arilpropan-1-ol sua producao e utilizacao
IS6403A (is)	2002-05-31	Nýjar heteróarýl afleiður, framleiðsla þeirra og notkun
ITBO20000398A0 (it)	2000-07-06	Tozzetto e metodo per la sua realizzazione .