PE20050722A1 - 3-NITRO-PIRAZOLO [1,5,a]PIRIMIDINAS 7-SUSTITUIDAS Y COMPOSICIONES Y METODOS RELACIONADOS - Google Patents
3-NITRO-PIRAZOLO [1,5,a]PIRIMIDINAS 7-SUSTITUIDAS Y COMPOSICIONES Y METODOS RELACIONADOSInfo
- Publication number
- PE20050722A1 PE20050722A1 PE2004000711A PE2004000711A PE20050722A1 PE 20050722 A1 PE20050722 A1 PE 20050722A1 PE 2004000711 A PE2004000711 A PE 2004000711A PE 2004000711 A PE2004000711 A PE 2004000711A PE 20050722 A1 PE20050722 A1 PE 20050722A1
- Authority
- PE
- Peru
- Prior art keywords
- phenyl
- nitro
- pyrazolo
- pyrimidin
- ethyl
- Prior art date
Links
- 150000003230 pyrimidines Chemical class 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title 1
- -1 PYRIMIDINYL Chemical class 0.000 abstract 8
- 150000001875 compounds Chemical class 0.000 abstract 3
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical group [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 2
- QUPDWYMUPZLYJZ-UHFFFAOYSA-N ethyl Chemical group C[CH2] QUPDWYMUPZLYJZ-UHFFFAOYSA-N 0.000 abstract 2
- JFSPBVWPKOEZCB-UHFFFAOYSA-N fenfuram Chemical compound O1C=CC(C(=O)NC=2C=CC=CC=2)=C1C JFSPBVWPKOEZCB-UHFFFAOYSA-N 0.000 abstract 2
- WCYWZMWISLQXQU-UHFFFAOYSA-N methyl Chemical group [CH3] WCYWZMWISLQXQU-UHFFFAOYSA-N 0.000 abstract 2
- MZRUFMBFIKGOAL-UHFFFAOYSA-N 5-nitro-1h-pyrazole Chemical compound [O-][N+](=O)C1=CC=NN1 MZRUFMBFIKGOAL-UHFFFAOYSA-N 0.000 abstract 1
- 208000019901 Anxiety disease Diseases 0.000 abstract 1
- 102000004300 GABA-A Receptors Human genes 0.000 abstract 1
- 108090000839 GABA-A Receptors Proteins 0.000 abstract 1
- 101100134922 Gallus gallus COR5 gene Proteins 0.000 abstract 1
- CZPWVGJYEJSRLH-UHFFFAOYSA-N Pyrimidine Chemical compound C1=CN=CN=C1 CZPWVGJYEJSRLH-UHFFFAOYSA-N 0.000 abstract 1
- 208000013738 Sleep Initiation and Maintenance disease Diseases 0.000 abstract 1
- 230000036506 anxiety Effects 0.000 abstract 1
- 206010015037 epilepsy Diseases 0.000 abstract 1
- 206010022437 insomnia Diseases 0.000 abstract 1
- 208000019116 sleep disease Diseases 0.000 abstract 1
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES200301747A ES2222814B1 (es) | 2003-07-24 | 2003-07-24 | 3-nitro-pirazolo(1,5-a)pirimidinas 7-sustituidas y composiciones y metodos relacionados. |
| ES200401696A ES2245893B1 (es) | 2003-07-24 | 2004-07-12 | Mejoras en el objeto de la patente de invencion n.p200301747 que se refiere a "3-nitro-pirazolo(1,5-a)pirimidinas 7-sustituidas y composiciones y metodos relacionados". |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20050722A1 true PE20050722A1 (es) | 2005-09-14 |
Family
ID=34354826
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2004000711A PE20050722A1 (es) | 2003-07-24 | 2004-07-23 | 3-NITRO-PIRAZOLO [1,5,a]PIRIMIDINAS 7-SUSTITUIDAS Y COMPOSICIONES Y METODOS RELACIONADOS |
Country Status (11)
| Country | Link |
|---|---|
| CN (1) | CN1829720A (ru) |
| AR (1) | AR045088A1 (ru) |
| CL (1) | CL2004001813A1 (ru) |
| EA (1) | EA200600318A1 (ru) |
| ES (2) | ES2222814B1 (ru) |
| IL (1) | IL173347A0 (ru) |
| MA (1) | MA27945A1 (ru) |
| PA (1) | PA8607401A1 (ru) |
| PE (1) | PE20050722A1 (ru) |
| TN (1) | TNSN05324A1 (ru) |
| ZA (1) | ZA200600471B (ru) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006084835A1 (en) * | 2005-02-10 | 2006-08-17 | Ferrer Internacional, S. A. | N-(3-(imidazo [1,5-a]pyrimidin-4-yl)phenyl]-sulfonamides and n-[3-(imidazo[1,5-a]pyrimidin-4-yl)-phenyl]-carboxamides and their use as gabaa receptor modulators |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4626538A (en) * | 1983-06-23 | 1986-12-02 | American Cyanamid Company | [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines |
| NZ208554A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions |
-
2003
- 2003-07-24 ES ES200301747A patent/ES2222814B1/es not_active Expired - Fee Related
-
2004
- 2004-07-12 ES ES200401696A patent/ES2245893B1/es not_active Expired - Fee Related
- 2004-07-20 PA PA8607401A patent/PA8607401A1/es unknown
- 2004-07-20 CL CL200401813A patent/CL2004001813A1/es unknown
- 2004-07-22 CN CN 200480021467 patent/CN1829720A/zh active Pending
- 2004-07-22 EA EA200600318A patent/EA200600318A1/ru unknown
- 2004-07-22 ZA ZA200600471A patent/ZA200600471B/xx unknown
- 2004-07-23 PE PE2004000711A patent/PE20050722A1/es not_active Application Discontinuation
- 2004-07-23 AR ARP040102618 patent/AR045088A1/es unknown
-
2005
- 2005-12-22 TN TNP2005000324A patent/TNSN05324A1/en unknown
-
2006
- 2006-01-24 IL IL173347A patent/IL173347A0/en unknown
- 2006-02-13 MA MA28798A patent/MA27945A1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EA200600318A1 (ru) | 2006-06-30 |
| AR045088A1 (es) | 2005-10-12 |
| MA27945A1 (fr) | 2006-06-01 |
| TNSN05324A1 (en) | 2007-07-10 |
| CN1829720A (zh) | 2006-09-06 |
| ES2245893B1 (es) | 2006-12-01 |
| ES2222814B1 (es) | 2005-12-01 |
| PA8607401A1 (es) | 2006-08-03 |
| ZA200600471B (en) | 2007-04-25 |
| CL2004001813A1 (es) | 2005-06-03 |
| ES2245893A1 (es) | 2006-01-16 |
| ES2222814A1 (es) | 2005-02-01 |
| IL173347A0 (en) | 2006-06-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application declared void or lapsed |