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PA8815101A1 - Asoc. entre unasal de bis-tiazolio o uno de sus precursosres y artemisinina o uno de sus derivados para el trat....... - Google Patents

Asoc. entre unasal de bis-tiazolio o uno de sus precursosres y artemisinina o uno de sus derivados para el trat.......

Info

Publication number
PA8815101A1
PA8815101A1 PA20098815101A PA8815101A PA8815101A1 PA 8815101 A1 PA8815101 A1 PA 8815101A1 PA 20098815101 A PA20098815101 A PA 20098815101A PA 8815101 A PA8815101 A PA 8815101A PA 8815101 A1 PA8815101 A1 PA 8815101A1
Authority
PA
Panama
Prior art keywords
artemisinine
derivatives
tiazolio
bis
unasal
Prior art date
Application number
PA20098815101A
Other languages
English (en)
Inventor
Laurent Fraisse
Henri Vial
Sharon Aurore Wein
Original Assignee
Sanofi Aventis
Univ Montpellier Ii
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39705083&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PA8815101(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis, Univ Montpellier Ii filed Critical Sanofi Aventis
Publication of PA8815101A1 publication Critical patent/PA8815101A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • A61K31/366Lactones having six-membered rings, e.g. delta-lactones
    • A61K31/37Coumarins, e.g. psoralen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

LA INVENCIÓN TIENE POR OBJETO UNA ASOCIACIÓN, QUE COMPRENDE UNA SAL DE BISTIAZOLIO, COMPUESTO DE FÓRMULA (VI) O UNO DE SUS PRECURSORES, Y ARTEMISININA O UNO DE SUS DERIVADOS. LA INVENCIÓN TIENE IGUALMENTE POR OBJETO UNA COMPOSICIÓN FARMACÉUTICA QUE COMPRENDE AL MENOS UNA SAL DE BIS-TIAZOLIO, COMPUESTO DE FÓRMULA (VI) O UNO DE SUS PRECURSORES, Y ARTEMISININA O UNO DE SUS DERIVADOS. LA INVENCIÓN TIENE TAMBIÉN POR OBJETO LA UTILIZACIÓN DE DICHA ASOCIACIÓN PARA LA PREPARACIÓN DE UN MEDICAMENTO DESTINADO AL TRATAMIENTO O A LA PREVENCIÓN DEL PALUDISMO GRAVE. LA INVENCIÓN TIENE FINALMENTE POR OBJETO UN KIT PARA EL TRATAMIENTO O LA PREVENCIÓN DEL PALUDISMO GRAVE.
PA20098815101A 2008-02-06 2009-02-05 Asoc. entre unasal de bis-tiazolio o uno de sus precursosres y artemisinina o uno de sus derivados para el trat....... PA8815101A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0800618A FR2926993B1 (fr) 2008-02-06 2008-02-06 Association entre un sel de bis-thiazolium ou l'un de ses precurseurs et l'artemisinine ou l'un de ses derives pour le traitement du paludisme

Publications (1)

Publication Number Publication Date
PA8815101A1 true PA8815101A1 (es) 2009-09-17

Family

ID=39705083

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20098815101A PA8815101A1 (es) 2008-02-06 2009-02-05 Asoc. entre unasal de bis-tiazolio o uno de sus precursosres y artemisinina o uno de sus derivados para el trat.......

Country Status (39)

Country Link
US (1) US8304440B2 (es)
EP (1) EP2252286B1 (es)
JP (1) JP5469095B2 (es)
KR (1) KR20100137442A (es)
CN (1) CN101980706B (es)
AP (1) AP2613A (es)
AR (1) AR070581A1 (es)
AT (1) ATE521347T1 (es)
AU (1) AU2009227092B2 (es)
BR (1) BRPI0907484A2 (es)
CA (1) CA2714184A1 (es)
CL (1) CL2009000264A1 (es)
CO (1) CO6300843A2 (es)
CR (1) CR11613A (es)
CY (1) CY1112113T1 (es)
DK (1) DK2252286T3 (es)
EA (1) EA022711B1 (es)
EC (1) ECSP10010381A (es)
ES (1) ES2372148T3 (es)
FR (1) FR2926993B1 (es)
HR (1) HRP20110858T8 (es)
IL (1) IL207442A0 (es)
JO (1) JO2820B1 (es)
MA (1) MA32128B1 (es)
MX (1) MX2010008653A (es)
MY (1) MY150776A (es)
NI (1) NI201000135A (es)
NZ (1) NZ587232A (es)
PA (1) PA8815101A1 (es)
PE (1) PE20091410A1 (es)
PL (1) PL2252286T3 (es)
PT (1) PT2252286E (es)
RS (1) RS52046B (es)
SI (1) SI2252286T1 (es)
TW (1) TWI402071B (es)
UA (1) UA99510C2 (es)
UY (1) UY31640A1 (es)
WO (1) WO2009115666A2 (es)
ZA (1) ZA201005611B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2951945B1 (fr) * 2009-11-05 2013-08-09 Sanofi Aventis Composition pharmaceutique
AU2014346668C1 (en) 2013-11-08 2018-04-26 Exthera Medical Corporation Methods for diagnosing infectious diseases using adsorption media
US10714230B2 (en) * 2017-12-06 2020-07-14 C3Nano Inc. Thin and uniform silver nanowires, method of synthesis and transparent conductive films formed from the nanowires
CN110604733A (zh) * 2019-09-19 2019-12-24 同济大学 青蒿素类药物与其它药物联用在制备抗疟疾药物中的应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1058717A (zh) * 1990-08-08 1992-02-19 中国人民解放军军事医学科学院微生物流行病研究所 抗疟新药—复方蒿甲醚及其制备方法
FR2796642B1 (fr) * 1999-07-21 2001-10-19 Centre Nat Rech Scient Precurseurs de sels de bis-ammonium quaternaire et leurs applications comme prodrogues ayant une activite anti-parasitaire
JP2003050535A (ja) * 2001-08-07 2003-02-21 T-Zone Corp ネットワーク教育システム、ネットワーク教育方法、および、プログラム
FR2884715B1 (fr) * 2005-04-20 2007-06-15 Sanofi Aventis Sa Association entre la ferroquine et un derive d'artemisinine pour le traitement du paludisme

Also Published As

Publication number Publication date
PT2252286E (pt) 2011-12-07
EP2252286A2 (fr) 2010-11-24
NZ587232A (en) 2012-06-29
JP5469095B2 (ja) 2014-04-09
AU2009227092A1 (en) 2009-09-24
TW201000098A (en) 2010-01-01
CL2009000264A1 (es) 2010-04-09
CN101980706B (zh) 2013-11-27
RS52046B (en) 2012-04-30
CY1112113T1 (el) 2015-11-04
AP2613A (en) 2013-03-13
NI201000135A (es) 2011-04-27
EA022711B1 (ru) 2016-02-29
IL207442A0 (en) 2010-12-30
AU2009227092B2 (en) 2014-08-07
AR070581A1 (es) 2010-04-21
BRPI0907484A2 (pt) 2019-09-24
CA2714184A1 (fr) 2009-09-24
DK2252286T3 (da) 2011-12-19
US8304440B2 (en) 2012-11-06
HRP20110858T8 (hr) 2012-02-29
TWI402071B (zh) 2013-07-21
FR2926993A1 (fr) 2009-08-07
CR11613A (es) 2010-11-22
SI2252286T1 (sl) 2012-01-31
HK1152892A1 (en) 2012-03-16
JO2820B1 (en) 2014-09-15
KR20100137442A (ko) 2010-12-30
ZA201005611B (en) 2012-06-27
UY31640A1 (es) 2009-08-31
EA201070923A1 (ru) 2011-02-28
MY150776A (en) 2014-02-28
ECSP10010381A (es) 2010-11-30
CN101980706A (zh) 2011-02-23
UA99510C2 (ru) 2012-08-27
US20110160254A1 (en) 2011-06-30
PE20091410A1 (es) 2009-10-14
FR2926993B1 (fr) 2011-03-11
AP2010005353A0 (en) 2010-08-31
MA32128B1 (fr) 2011-03-01
WO2009115666A2 (fr) 2009-09-24
MX2010008653A (es) 2011-03-04
ES2372148T3 (es) 2012-01-16
HRP20110858T1 (hr) 2012-01-31
JP2011514319A (ja) 2011-05-06
WO2009115666A3 (fr) 2009-12-23
PL2252286T3 (pl) 2012-02-29
EP2252286B1 (fr) 2011-08-24
CO6300843A2 (es) 2011-07-21
ATE521347T1 (de) 2011-09-15

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