OA11423A - Combination effective for the treatment of impotence - Google Patents

Combination effective for the treatment of impotence Download PDF

Info

Publication number: OA11423A
Authority: OA; OAPI
Prior art keywords: composition; daim; compound; cgmp; pharmaceutically acceptable
Prior art date: 1997-12-16

Application number

OA1200000169A

Other languages

English (en)

Inventor

Michael Grant Wiyllie

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-12-16

Filing date

2000-06-15

Publication date

2004-04-21

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22090927&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA11423(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2000-06-15 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2004-04-21 Publication of OA11423A publication Critical patent/OA11423A/en

Links

201000001881 impotence Diseases 0.000 title claims abstract description 36
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239000000203 mixture Substances 0.000 claims abstract description 71
239000000674 adrenergic antagonist Substances 0.000 claims abstract description 58
150000003839 salts Chemical class 0.000 claims abstract description 35
BNRNXUUZRGQAQC-UHFFFAOYSA-N sildenafil Chemical compound CCCC1=NN(C)C(C(N2)=O)=C1N=C2C(C(=CC=1)OCC)=CC=1S(=O)(=O)N1CCN(C)CC1 BNRNXUUZRGQAQC-UHFFFAOYSA-N 0.000 claims abstract description 30
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RUZYUOTYCVRMRZ-UHFFFAOYSA-N doxazosin Chemical compound C1OC2=CC=CC=C2OC1C(=O)N(CC1)CCN1C1=NC(N)=C(C=C(C(OC)=C2)OC)C2=N1 RUZYUOTYCVRMRZ-UHFFFAOYSA-N 0.000 claims description 34
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VCKUSRYTPJJLNI-UHFFFAOYSA-N terazosin Chemical compound N=1C(N)=C2C=C(OC)C(OC)=CC2=NC=1N(CC1)CCN1C(=O)C1CCCO1 VCKUSRYTPJJLNI-UHFFFAOYSA-N 0.000 claims description 21
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
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Medicinal Chemistry (AREA)
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Chemical Kinetics & Catalysis (AREA)
Reproductive Health (AREA)
Endocrinology (AREA)
Gynecology & Obstetrics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medicines Containing Plant Substances (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

OA1200000169A 1997-12-16 2000-06-15 Combination effective for the treatment of impotence OA11423A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US6974197P	1997-12-16	1997-12-16

Publications (1)

Publication Number	Publication Date
OA11423A true OA11423A (en)	2004-04-21

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ID=22090927

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OA1200000169A OA11423A (en)	1997-12-16	2000-06-15	Combination effective for the treatment of impotence

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WO (1)	WO1999030697A2 (es)
YU (1)	YU33700A (es)
ZA (1)	ZA9811507B (es)

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CA2362918A1 (en) *	1999-03-08	2000-09-14	Elizabeth Stoner	Methods and compositions for treating erectile dysfunction
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WO2002022127A1 (en) *	2000-09-13	2002-03-21	Isis Innovation Limited	Use of phosphodiesterase inhibitors for the treatment of anorectal disorders
AU2002223802A1 (en) *	2000-11-17	2002-05-27	Warner-Lambert Company Llc	Treatment of sexual dysfunction with non peptide bombesin receptor antagonists
US20030114469A1 (en) *	2001-09-27	2003-06-19	Cohen David Saul	Combinations
GB0219961D0 (en)	2002-08-28	2002-10-02	Pfizer Ltd	Oxytocin inhibitors
GB0225908D0 (en) *	2002-11-06	2002-12-11	Pfizer Ltd	Treatment of female sexual dysfunction
US7323462B2 (en)	2002-12-10	2008-01-29	Pfizer Inc.	Morpholine dopamine agonists
CA2451267A1 (en)	2002-12-13	2004-06-13	Warner-Lambert Company Llc	Pharmaceutical uses for alpha2delta ligands
US7291640B2 (en)	2003-09-22	2007-11-06	Pfizer Inc.	Substituted triazole derivatives as oxytocin antagonists
AP2007004047A0 (en)	2005-01-20	2007-06-30	Pfizer Ltd	Substituted triazole derivatives as oxtocin antagonists
US8506934B2 (en)	2005-04-29	2013-08-13	Robert I. Henkin	Methods for detection of biological substances
US20070225217A1 (en)	2005-11-09	2007-09-27	Combinatorx, Incorporated	Methods, compositions, and kits for the treatment of medical conditions
US8293489B2 (en)	2007-01-31	2012-10-23	Henkin Robert I	Methods for detection of biological substances
US8580801B2 (en)	2008-07-23	2013-11-12	Robert I. Henkin	Phosphodiesterase inhibitor treatment
CN101781302B (zh) *	2009-05-31	2013-07-10	段波	一种磷酸二酯酶抑制剂和异黄酮形成的加成物及其应用
US20150119399A1 (en)	2012-01-10	2015-04-30	President And Fellows Of Harvard College	Beta-cell replication promoting compounds and methods of their use
EP2903619B1 (en)	2012-10-05	2019-06-05	Robert I. Henkin	Phosphodiesterase inhibitors for treating taste and smell disorders
WO2015126944A1 (en)	2014-02-18	2015-08-27	Henkin Robert I	Methods and compositions for diagnosing and treating loss and/or distortion of taste or smell
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ZA878182B (en) *	1986-11-05	1988-05-02	Merrell Dow Pharmaceuticals Inc.	Enhancement of prazosin
FR2649613B1 (fr) *	1989-07-11	1991-09-27	Virag Ronald	Medicament vaso-actif
US5242391A (en) *	1990-04-25	1993-09-07	Alza Corporation	Urethral insert for treatment of erectile dysfunction
EP0459666B1 (en) *	1990-05-31	1994-11-09	Pfizer Inc.	Medicaments against impotence
GB9311920D0 (en) *	1993-06-09	1993-07-28	Pfizer Ltd	Therapeutic agents
GB9523752D0 (en) *	1995-11-21	1996-01-24	Pfizer Ltd	Pharmaceutical formulations

1998
- 1998-10-29 AT AT98947741T patent/ATE318602T1/de not_active IP Right Cessation
- 1998-10-29 CA CA002314993A patent/CA2314993A1/en not_active Abandoned
- 1998-10-29 TR TR2000/01733T patent/TR200001733T2/xx unknown
- 1998-10-29 PL PL98341575A patent/PL341575A1/xx unknown
- 1998-10-29 SK SK878-2000A patent/SK8782000A3/sk unknown
- 1998-10-29 DE DE69833671T patent/DE69833671T2/de not_active Expired - Fee Related
- 1998-10-29 CZ CZ20002199A patent/CZ20002199A3/cs unknown
- 1998-10-29 JP JP2000538680A patent/JP2002508315A/ja active Pending
- 1998-10-29 CN CN98812331A patent/CN1282248A/zh active Pending
- 1998-10-29 BR BR9813699-2A patent/BR9813699A/pt not_active Application Discontinuation
- 1998-10-29 YU YU33700A patent/YU33700A/sh unknown
- 1998-10-29 EP EP98947741A patent/EP1037616B1/en not_active Revoked
- 1998-10-29 ES ES98947741T patent/ES2258300T3/es not_active Expired - Lifetime
- 1998-10-29 HU HU0100705A patent/HUP0100705A3/hu unknown
- 1998-10-29 KR KR1020007006455A patent/KR20010033092A/ko not_active Application Discontinuation
- 1998-10-29 NZ NZ504487A patent/NZ504487A/xx unknown
- 1998-10-29 IL IL13651598A patent/IL136515A0/xx unknown
- 1998-10-29 EA EA200000526A patent/EA200000526A1/ru unknown
- 1998-10-29 AU AU94558/98A patent/AU759825B2/en not_active Ceased
- 1998-10-29 WO PCT/IB1998/001723 patent/WO1999030697A2/en active IP Right Grant
- 1998-11-09 GT GT199800177A patent/GT199800177A/es unknown
- 1998-11-10 PA PA19988462801A patent/PA8462801A1/es unknown
- 1998-11-11 HN HN1998000174A patent/HN1998000174A/es unknown
- 1998-11-30 CO CO98070722A patent/CO4810381A1/es unknown
- 1998-12-10 AP APAP/P/1998/001414A patent/AP915A/en active
- 1998-12-11 PE PE1998001206A patent/PE20000011A1/es not_active Application Discontinuation
- 1998-12-14 UY UY25300A patent/UY25300A1/es not_active Application Discontinuation
- 1998-12-15 MA MA25396A patent/MA26586A1/fr unknown
- 1998-12-15 ZA ZA9811507A patent/ZA9811507B/xx unknown
- 1998-12-15 DZ DZ980285A patent/DZ2675A1/xx active
- 1998-12-15 AR ARP980106360A patent/AR016433A1/es unknown
- 1998-12-15 TN TNTNSN98227A patent/TNSN98227A1/fr unknown
2000
- 2000-05-19 IS IS5504A patent/IS5504A/is unknown
- 2000-06-13 BG BG104528A patent/BG104528A/xx unknown
- 2000-06-15 NO NO20003065A patent/NO20003065L/no not_active Application Discontinuation
- 2000-06-15 OA OA1200000169A patent/OA11423A/en unknown
- 2000-06-16 HR HR20000407A patent/HRP20000407A2/hr not_active Application Discontinuation
2007
- 2007-08-20 JP JP2007213745A patent/JP2007332156A/ja not_active Withdrawn

Also Published As

Publication number	Publication date
PL341575A1 (en)	2001-04-23
SK8782000A3 (en)	2002-03-05
CA2314993A1 (en)	1999-06-24
HUP0100705A2 (hu)	2001-08-28
CN1282248A (zh)	2001-01-31
TNSN98227A1 (fr)	2005-03-15
HN1998000174A (es)	1999-01-08
AP915A (en)	2000-12-18
NO20003065L (no)	2000-08-15
HUP0100705A3 (en)	2001-12-28
IL136515A0 (en)	2001-06-14
EP1037616B1 (en)	2006-03-01
KR20010033092A (ko)	2001-04-25
DE69833671D1 (de)	2006-04-27
ES2258300T3 (es)	2006-08-16
CZ20002199A3 (cs)	2001-10-17
ATE318602T1 (de)	2006-03-15
JP2007332156A (ja)	2007-12-27
MA26586A1 (fr)	2004-12-20
DE69833671T2 (de)	2006-11-30
PA8462801A1 (es)	2000-05-24
WO1999030697A2 (en)	1999-06-24
CO4810381A1 (es)	1999-06-30
HRP20000407A2 (en)	2000-10-31
ZA9811507B (en)	2000-06-19
WO1999030697A3 (en)	1999-08-26
DZ2675A1 (fr)	2003-03-29
NO20003065D0 (no)	2000-06-15
AU759825B2 (en)	2003-05-01
EA200000526A1 (ru)	2000-12-25
IS5504A (is)	2000-05-19
UY25300A1 (es)	2000-12-29
AP9801414A0 (en)	1998-12-31
JP2002508315A (ja)	2002-03-19
BG104528A (en)	2001-02-28
YU33700A (sh)	2004-05-12
AU9455898A (en)	1999-07-05
AR016433A1 (es)	2001-07-04
NZ504487A (en)	2002-11-26
BR9813699A (pt)	2000-10-10
TR200001733T2 (tr)	2000-11-21
EP1037616A2 (en)	2000-09-27
GT199800177A (es)	2000-05-02
PE20000011A1 (es)	2000-01-18

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