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NO994071D0 - Epotilones med en modifisert sidekjede - Google Patents

Epotilones med en modifisert sidekjede

Info

Publication number
NO994071D0
NO994071D0 NO994071A NO994071A NO994071D0 NO 994071 D0 NO994071 D0 NO 994071D0 NO 994071 A NO994071 A NO 994071A NO 994071 A NO994071 A NO 994071A NO 994071 D0 NO994071 D0 NO 994071D0
Authority
NO
Norway
Prior art keywords
epotilones
side chain
modified side
modified
chain
Prior art date
Application number
NO994071A
Other languages
English (en)
Other versions
NO994071L (no
NO327211B1 (no
Inventor
Gerhard Hoefle
Michael Sefkow
Original Assignee
Biotechnolog Forschung Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biotechnolog Forschung Gmbh filed Critical Biotechnolog Forschung Gmbh
Publication of NO994071D0 publication Critical patent/NO994071D0/no
Publication of NO994071L publication Critical patent/NO994071L/no
Publication of NO327211B1 publication Critical patent/NO327211B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Epoxy Compounds (AREA)
  • Silicon Polymers (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other Resins Obtained By Reactions Not Involving Carbon-To-Carbon Unsaturated Bonds (AREA)
NO19994071A 1997-02-25 1999-08-24 Epotiloner med en modifisert sidekjede, samt fremgangsmate for fremstilling derav NO327211B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19707505 1997-02-25
PCT/EP1998/001060 WO1998038192A1 (de) 1997-02-25 1998-02-25 Seitenkettenmodifizierte epothilone

Publications (3)

Publication Number Publication Date
NO994071D0 true NO994071D0 (no) 1999-08-24
NO994071L NO994071L (no) 1999-10-21
NO327211B1 NO327211B1 (no) 2009-05-11

Family

ID=7821415

Family Applications (1)

Application Number Title Priority Date Filing Date
NO19994071A NO327211B1 (no) 1997-02-25 1999-08-24 Epotiloner med en modifisert sidekjede, samt fremgangsmate for fremstilling derav

Country Status (25)

Country Link
US (1) US6359140B1 (no)
EP (2) EP1201666A3 (no)
JP (1) JP2001513098A (no)
KR (1) KR100494179B1 (no)
CN (2) CN1128803C (no)
AR (1) AR011878A1 (no)
AT (1) ATE221888T1 (no)
AU (1) AU736062B2 (no)
BR (1) BR9807742B1 (no)
CA (1) CA2281105A1 (no)
CZ (1) CZ298027B6 (no)
DE (2) DE59805110D1 (no)
DK (1) DK0975638T3 (no)
ES (1) ES2183338T3 (no)
HK (1) HK1023774A1 (no)
HU (1) HU228851B1 (no)
IL (1) IL131343A (no)
NO (1) NO327211B1 (no)
NZ (1) NZ337195A (no)
PL (1) PL190422B1 (no)
PT (1) PT975638E (no)
RU (1) RU2201932C2 (no)
TW (1) TW480263B (no)
WO (1) WO1998038192A1 (no)
ZA (1) ZA981575B (no)

Families Citing this family (94)

* Cited by examiner, † Cited by third party
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US20050043376A1 (en) * 1996-12-03 2005-02-24 Danishefsky Samuel J. Synthesis of epothilones, intermediates thereto, analogues and uses thereof
US6204388B1 (en) 1996-12-03 2001-03-20 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
US6867305B2 (en) 1996-12-03 2005-03-15 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto and analogues thereof
AU756699B2 (en) 1996-12-03 2003-01-23 Sloan-Kettering Institute For Cancer Research Synthesis of epothilones, intermediates thereto, analogues and uses thereof
US6380394B1 (en) 1996-12-13 2002-04-30 The Scripps Research Institute Epothilone analogs
US6441186B1 (en) * 1996-12-13 2002-08-27 The Scripps Research Institute Epothilone analogs
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US6518421B1 (en) 2000-03-20 2003-02-11 Bristol-Myers Squibb Company Process for the preparation of epothilone analogs
US6593115B2 (en) 2000-03-24 2003-07-15 Bristol-Myers Squibb Co. Preparation of epothilone intermediates
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US7820702B2 (en) 2004-02-04 2010-10-26 Bristol-Myers Squibb Company Sulfonylpyrrolidine modulators of androgen receptor function and method
US7378426B2 (en) 2004-03-01 2008-05-27 Bristol-Myers Squibb Company Fused heterotricyclic compounds as inhibitors of 17β-hydroxysteroid dehydrogenase 3
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US7625923B2 (en) 2004-03-04 2009-12-01 Bristol-Myers Squibb Company Bicyclic modulators of androgen receptor function
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US20060134214A1 (en) * 2004-11-18 2006-06-22 Ismat Ullah Enteric coated bead comprising epothilone or epothilone analog, and preparation and administration thereof
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Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4138042C2 (de) * 1991-11-19 1993-10-14 Biotechnolog Forschung Gmbh Epothilone, deren Herstellungsverfahren sowie diese Verbindungen enthaltende Mittel
DK1186606T4 (da) * 1995-11-17 2011-12-05 Biotechnolog Forschung Gmbh Epothilonderivater, deres fremstilling og anvendelse
US6441186B1 (en) * 1996-12-13 2002-08-27 The Scripps Research Institute Epothilone analogs
EP1201666A3 (de) * 1997-02-25 2003-03-05 Gesellschaft für biotechnologische Forschung mbH (GBF) Seitenkettenmodifizierte Epothilone

Also Published As

Publication number Publication date
CZ298027B6 (cs) 2007-05-30
PL335329A1 (en) 2000-04-25
EP1201666A2 (de) 2002-05-02
BR9807742A (pt) 2000-02-22
HUP0002189A3 (en) 2001-12-28
CZ286599A3 (cs) 2000-03-15
IL131343A0 (en) 2001-01-28
BR9807742B1 (pt) 2010-12-14
AR011878A1 (es) 2000-09-13
AU6724998A (en) 1998-09-18
IL131343A (en) 2004-03-28
HU228851B1 (en) 2013-06-28
EP0975638B1 (de) 2002-08-07
CN1544436A (zh) 2004-11-10
ATE221888T1 (de) 2002-08-15
DE19880193D2 (de) 2000-08-24
NO994071L (no) 1999-10-21
NZ337195A (en) 2001-05-25
HK1023774A1 (en) 2000-09-22
NO327211B1 (no) 2009-05-11
EP1201666A3 (de) 2003-03-05
JP2001513098A (ja) 2001-08-28
CN1128803C (zh) 2003-11-26
AU736062B2 (en) 2001-07-26
CN1248974A (zh) 2000-03-29
PT975638E (pt) 2002-12-31
ZA981575B (en) 1998-09-08
US6359140B1 (en) 2002-03-19
ES2183338T3 (es) 2003-03-16
TW480263B (en) 2002-03-21
HUP0002189A2 (hu) 2001-10-28
RU2201932C2 (ru) 2003-04-10
DK0975638T3 (da) 2002-11-18
DE59805110D1 (de) 2002-09-12
KR100494179B1 (ko) 2005-06-10
EP0975638A1 (de) 2000-02-02
KR20000075705A (ko) 2000-12-26
WO1998038192A1 (de) 1998-09-03
PL190422B1 (pl) 2005-12-30
CA2281105A1 (en) 1998-09-03

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