[go: up one dir, main page]

NO971544D0 - Cykliske heksapeptider med antibiotisk aktivitet - Google Patents

Cykliske heksapeptider med antibiotisk aktivitet

Info

Publication number
NO971544D0
NO971544D0 NO971544A NO971544A NO971544D0 NO 971544 D0 NO971544 D0 NO 971544D0 NO 971544 A NO971544 A NO 971544A NO 971544 A NO971544 A NO 971544A NO 971544 D0 NO971544 D0 NO 971544D0
Authority
NO
Norway
Prior art keywords
antibiotic activity
cyclic hexapeptides
hexapeptides
cyclic
antibiotic
Prior art date
Application number
NO971544A
Other languages
English (en)
Other versions
NO971544L (no
NO328483B1 (no
Inventor
Hidenori Ohki
Masaki Tomishima
Akira Yamada
Hisashi Takasugi
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26305774&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO971544(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB9420425A external-priority patent/GB9420425D0/en
Priority claimed from GBGB9508745.8A external-priority patent/GB9508745D0/en
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Publication of NO971544D0 publication Critical patent/NO971544D0/no
Publication of NO971544L publication Critical patent/NO971544L/no
Publication of NO328483B1 publication Critical patent/NO328483B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
NO19971544A 1994-10-07 1997-04-04 Polypeptidforbindelser, farmasoytiske preparater inneholdende disse og fremgangsmate for a fremstille forbindelsene samt deres anvendelse. NO328483B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB9420425A GB9420425D0 (en) 1994-10-07 1994-10-07 New compound
GBGB9508745.8A GB9508745D0 (en) 1995-04-28 1995-04-28 New compound
PCT/JP1995/001983 WO1996011210A1 (en) 1994-10-07 1995-09-29 Cyclic hexapeptides having antibiotic activity

Publications (3)

Publication Number Publication Date
NO971544D0 true NO971544D0 (no) 1997-04-04
NO971544L NO971544L (no) 1997-06-04
NO328483B1 NO328483B1 (no) 2010-03-01

Family

ID=26305774

Family Applications (2)

Application Number Title Priority Date Filing Date
NO19971544A NO328483B1 (no) 1994-10-07 1997-04-04 Polypeptidforbindelser, farmasoytiske preparater inneholdende disse og fremgangsmate for a fremstille forbindelsene samt deres anvendelse.
NO2010016C NO2010016I2 (no) 1994-10-07 2010-08-09 Micafungin Sodium

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO2010016C NO2010016I2 (no) 1994-10-07 2010-08-09 Micafungin Sodium

Country Status (27)

Country Link
US (2) US6107458A (no)
EP (1) EP0788511B1 (no)
JP (2) JP2897427B2 (no)
KR (1) KR100353303B1 (no)
CN (1) CN1203089C (no)
AR (1) AR041770A1 (no)
AT (1) ATE229541T1 (no)
AU (1) AU696949B2 (no)
BR (2) BRPI9504791B8 (no)
CA (1) CA2202058C (no)
DE (2) DE122008000025I2 (no)
DK (1) DK0788511T3 (no)
ES (1) ES2187575T3 (no)
FI (1) FI119988B (no)
FR (1) FR08C0028I2 (no)
HK (1) HK1004136A1 (no)
HU (1) HU228151B1 (no)
IL (1) IL115484A (no)
LU (1) LU91452I2 (no)
MX (1) MX9702531A (no)
NL (1) NL300352I2 (no)
NO (2) NO328483B1 (no)
OA (1) OA10475A (no)
PT (1) PT788511E (no)
RU (1) RU2165423C2 (no)
TR (1) TR199501229A2 (no)
WO (1) WO1996011210A1 (no)

Families Citing this family (59)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5696084A (en) * 1996-08-16 1997-12-09 Abbott Laboratories Amino-lipopetide antifungal agents
AUPO371596A0 (en) * 1996-11-19 1996-12-12 Fujisawa Pharmaceutical Co., Ltd. New compound
AUPO381496A0 (en) * 1996-11-25 1996-12-19 Fujisawa Pharmaceutical Co., Ltd. New compound
EP0994101A4 (en) * 1997-06-18 2002-05-02 Fujisawa Pharmaceutical Co NEW PREPARATION PROCESS
AU756792B2 (en) * 1998-02-09 2003-01-23 Fujisawa Pharmaceutical Co., Ltd. New compound
KR100396737B1 (ko) * 1998-02-09 2003-09-13 후지사와 야꾸힝 고교 가부시키가이샤 신규 화합물
US7084279B1 (en) * 1999-02-11 2006-08-01 Emisphere Technologies Inc. Oxadiazole compounds and compositions for delivering active agents
WO2000047188A1 (en) * 1999-02-11 2000-08-17 Emisphere Technologies, Inc. Oxadiazole compounds and compositions for delivering active agents
AUPP999799A0 (en) * 1999-04-27 1999-05-20 Fujisawa Pharmaceutical Co., Ltd. New compound
AUPQ066399A0 (en) * 1999-05-31 1999-06-24 Fujisawa Pharmaceutical Co., Ltd. Antifungal combination use
TWI233805B (en) * 1999-07-01 2005-06-11 Fujisawa Pharmaceutical Co Stabilized pharmaceutical composition in lyophilized form as antifungal agent
JP2003505468A (ja) 1999-07-27 2003-02-12 アヴェンティス ファルマ ドイチェラント ゲーエムベーハー 新規なシクロヘキサペプチド化合物、それらの製造方法及びそれらの医薬品としての使用
AUPQ462399A0 (en) * 1999-12-13 2000-01-13 Fujisawa Pharmaceutical Co., Ltd. New use
TWI250992B (en) * 2000-02-21 2006-03-11 Astellas Pharma Inc Polypeptide compounds for the prophylactic and/or therapeutic treatment of infectious diseases caused by pathogenic microorganisms
ES2191516B1 (es) * 2000-07-28 2005-01-01 Consejo Superior De Investigaciones Cientificas Antibioticos antifungicos de naturaleza peptidica inhibidores de la germinacion y el crecimiento de hongos fitopatogenos.
AUPQ938700A0 (en) * 2000-08-14 2000-09-07 Fujisawa Pharmaceutical Co., Ltd. Antifungal combination use
WO2003079972A2 (en) 2002-02-22 2003-10-02 New River Parmaceuticals Inc. Active agent delivery systems and methods for protecting and administering active agents
ATE452637T1 (de) 2001-01-29 2010-01-15 Shionogi & Co Arzneipräparat, das als wirkstoff 5-methyl-1- phenyl-2-(1h)-pyridon enthält
JP2005053782A (ja) * 2001-08-31 2005-03-03 Fujisawa Pharmaceut Co Ltd 環状リポペプチド化合物の新規結晶
WO2004014879A1 (en) * 2002-08-08 2004-02-19 Fujisawa Pharmaceutical Co., Ltd. New process
AU2003903205A0 (en) * 2003-06-23 2003-07-10 Fujisawa Pharmaceutical Co., Ltd. New compound
US7452861B2 (en) 2003-07-22 2008-11-18 Theravance, Inc. Use of an echinocandin antifungal agent in combination with a glycopeptide antibacterial agent
WO2005026323A2 (en) * 2003-09-05 2005-03-24 Merck & Co., Inc. Stationary phases and a purification process using the stationary phases
ATE547404T1 (de) * 2003-09-22 2012-03-15 Msd Kk Piperidinderivate
US7476673B2 (en) * 2003-12-30 2009-01-13 Allergan, Inc. Disubstituted chalcone oximes as selective agonists of RARγ retinoid receptors
US20050261365A1 (en) * 2004-05-20 2005-11-24 The Scripps Research Institute Transthyretin stabilization
AR051093A1 (es) 2004-09-20 2006-12-20 Xenon Pharmaceuticals Inc Derivados heterociclicos y su uso como inhibidores de estearoil-coa desaturasa
CN101083992A (zh) 2004-09-20 2007-12-05 泽农医药公司 抑制人硬脂酰CoA去饱和酶的哒嗪衍生物
CN101083994A (zh) 2004-09-20 2007-12-05 泽农医药公司 杂环衍生物及其用作硬脂酰CoA去饱和酶抑制剂的用途
BRPI0515483A (pt) 2004-09-20 2008-07-22 Xenon Pharmaceuticals Inc derivados heterocìclicos para o tratamento de doenças mediadas por enzimas estearoil-coa desaturase
AR051091A1 (es) 2004-09-20 2006-12-20 Xenon Pharmaceuticals Inc Derivados heterociclicos y su uso como inhibidores de la estearoil-coa desaturasa
JP2008513515A (ja) 2004-09-20 2008-05-01 ゼノン・ファーマシューティカルズ・インコーポレイテッド 複素環誘導体および治療薬としてのそれらの使用
CA2580762A1 (en) 2004-09-20 2006-03-30 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as therapeutic agents
MX2007004484A (es) * 2004-10-13 2007-06-25 Ptc Therapeutics Inc Compuestos de pirazol o triazol y su uso para la fabricacion de un medicamento para tratar las enfermedades relacionadas con la mutacion somatica.
MX2007015216A (es) 2005-06-03 2008-02-22 Xenon Pharmaceuticals Inc Derivados de aminotiazol y sus usos como agentes terapeuticos.
JP5222561B2 (ja) * 2005-10-07 2013-06-26 キッセイ薬品工業株式会社 含窒素芳香族複素環化合物およびそれを含有する医薬組成物
CN101516387B (zh) * 2006-07-26 2014-06-04 桑多斯股份公司 卡泊芬净制剂
US8853392B2 (en) 2007-06-03 2014-10-07 Vanderbilt University Benzamide mGluR5 positive allosteric modulators and methods of making and using same
CA2699980C (en) 2007-08-13 2015-06-02 Divergence, Inc. Methods for the control of plant parasitic nematodes comprising application of oxadiazole compounds to plants, seeds or soil
CA2704562A1 (en) * 2007-10-29 2009-05-07 Astellas Pharma Inc. Polypeptide compound
US8034806B2 (en) 2007-11-02 2011-10-11 Vanderbilt University Bicyclic mGluR5 positive allosteric modulators and methods of making and using same
EP2300442A2 (en) * 2008-06-24 2011-03-30 Irm Llc Compounds and methods for modulating g protein-coupled receptors
US9394340B2 (en) 2009-03-24 2016-07-19 Cadila Healthcare Limited Purification process for lipopeptides
BR112013023531A2 (pt) * 2011-04-04 2016-12-06 Xellia Pharmaceuticals Aps processo de um único vaso para a fabricação de micafungina ou de um sal desta
RS54240B1 (en) 2011-04-20 2015-12-31 Xellia Pharmaceuticals Aps PROCEDURE FOR PURIFICATION OF MIKAFUNGIN
CN102775476B (zh) 2011-05-12 2015-01-07 上海天伟生物制药有限公司 一种米卡芬净钠盐的制备方法
EP2709609B1 (en) 2011-05-17 2017-10-04 Shionogi & Co., Ltd. Heterocyclic compounds
HUE029720T2 (en) * 2011-09-09 2017-03-28 Sandoz Ag Preparation of micafungin intermediates
CN102627689B (zh) 2012-03-30 2014-08-06 上海天伟生物制药有限公司 一种环肽类化合物的水合物及其制备方法和用途
CN102627688B (zh) 2012-03-30 2014-12-31 上海天伟生物制药有限公司 一种高纯度环肽化合物及其制备方法和用途
CN102659930B (zh) 2012-03-30 2014-04-23 上海天伟生物制药有限公司 一种高纯度环肽类物质的晶体及其制备方法和用途
US10183973B2 (en) * 2014-05-29 2019-01-22 Shanghai Techwell Biopharmaceutical Co., Ltd. Solvate of cyclic peptide compound, preparation method for same, and uses thereof
JP7109189B2 (ja) * 2014-05-29 2022-07-29 シャンハイ テックウェル バイオファーマシューティカル カンパニー リミテッド シクロペプチド系化合物の組成物およびその製造方法と使用
EP3226885A4 (en) * 2014-10-07 2018-07-18 Alaparthi, Lakshmi Prasad Intermediates and processes to prepare micafungin
CA2937365C (en) 2016-03-29 2018-09-18 F. Hoffmann-La Roche Ag Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same
EP3485873A1 (en) 2017-11-17 2019-05-22 Cadila Healthcare Limited Stable pharmaceutical injectable compositions of micafungin
CN113087775B (zh) * 2018-05-31 2022-07-08 杭州中美华东制药有限公司 米卡芬净钠新晶型ii及其制备方法
WO2020013116A1 (ja) * 2018-07-10 2020-01-16 京都薬品工業株式会社 Ｐｔｐ－１ｂ阻害剤およびその用途
CN110734408A (zh) * 2019-10-22 2020-01-31 重庆康乐制药有限公司 一种米卡芬净类衍生物侧链中间体的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE912046A1 (en) * 1990-06-18 1991-12-18 Fujisawa Pharmaceutical Co New polypeptide compound and a process for preparation¹thereof
MY136593A (en) * 1992-03-19 2008-10-31 Lilly Co Eli Cyclic peptide antifungal agents and process for preparation thereof

Also Published As

Publication number Publication date
CA2202058C (en) 2007-11-06
JPH10324695A (ja) 1998-12-08
ATE229541T1 (de) 2002-12-15
AU696949B2 (en) 1998-09-24
BR9504791B1 (pt) 2010-10-05
ES2187575T3 (es) 2003-06-16
NO971544L (no) 1997-06-04
JPH10507174A (ja) 1998-07-14
FR08C0028I1 (no) 2008-08-15
HU228151B1 (en) 2012-12-28
RU2165423C2 (ru) 2001-04-20
MX9702531A (es) 1997-06-28
JP2897427B2 (ja) 1999-05-31
CN1203089C (zh) 2005-05-25
NO2010016I1 (no) 2010-08-16
NL300352I2 (nl) 2008-11-03
NO2010016I2 (no) 2011-10-17
FI971397A0 (fi) 1997-04-04
OA10475A (en) 2002-04-08
FI119988B (fi) 2009-05-29
JP3518665B2 (ja) 2004-04-12
IL115484A0 (en) 1996-01-19
EP0788511A1 (en) 1997-08-13
US6265536B1 (en) 2001-07-24
AR041770A1 (es) 2005-06-01
FI971397L (fi) 1997-05-27
FR08C0028I2 (no) 2009-11-20
LU91452I2 (fr) 2008-08-04
DE122008000025I2 (de) 2011-02-17
BRPI9504791B8 (pt) 2019-12-31
EP0788511B1 (en) 2002-12-11
WO1996011210A1 (en) 1996-04-18
HK1004136A1 (en) 1998-11-20
KR100353303B1 (ko) 2003-01-15
DE122008000025I1 (de) 2008-08-21
DE69529172T2 (de) 2003-04-17
IL115484A (en) 2000-07-16
CA2202058A1 (en) 1996-04-18
CN1168675A (zh) 1997-12-24
US6107458A (en) 2000-08-22
TR199501229A2 (tr) 1996-07-21
DK0788511T3 (da) 2003-03-31
KR970707150A (ko) 1997-12-01
HUT77736A (hu) 1998-07-28
BR9504791A (pt) 1996-10-22
DE69529172D1 (de) 2003-01-23
NL300352I1 (nl) 2008-08-01
AU3578095A (en) 1996-05-02
PT788511E (pt) 2003-04-30
NO328483B1 (no) 2010-03-01

Similar Documents

Publication Publication Date Title
DK0788511T3 (da) Cykliske hexapeptider med antibiotisk aktivitet
LV11547A (lv) Makrolidi ar imunodepresantu aktivitati
BR9708149A (pt) Imidazois substituídos com cicloalquila
FI931888L (fi) Kramploesande cykliska fruktopyranossulfiter -och sulfater
DE69517873D1 (de) Polsterungsstruktur
ATE228535T1 (de) Zyklische hexapeptide mit fungizider aktivität
NO952039D0 (no) Proteiner med glykosyltransferase-aktivitet
EE9700087A (et) Uued immunomodulatoorse toimega peptiidid
FI955182A0 (fi) Korirakenne
EE9600208A (et) Uued immuunomodulatoorse toimega peptiidid
DK0797579T3 (da) Erythromycin A-9-O-oxim-derivater udstyret med antibiotisk aktivitet
DE69533337D1 (de) Bakterielles protein mit xylanase aktivität
FI945227L (fi) Sykliset heksapeptidit, niiden valmistus ja käyttö
EP0500170A3 (en) Cyclic hexapeptides having antibiotic activity
DE69516958D1 (de) Zeitschaltungsanordnung
DK0731078T3 (da) Terpenquinon med antitumoraktivitet
NO934805D0 (no) Manifoldanordning
DE69414092D1 (de) Elastisches Doppelgestrick
EP0859007A4 (en) CYCLIC HEXAPEPTIDE
NO981939D0 (no) Tiomorfinaner med neurobeskyttende aktivitet
KR950018692U (ko) 배기 기능을 갖는 깔때기
KR970053563U (ko) 자석이 부착된 치솔
FI940841A0 (fi) Lockoeppnare foer konservburk med undertryck
KR970051287U (ko) 덕트 캡 체결구조
KR960012685U (ko) 씨모오스 구조

Legal Events

Date Code Title Description
CREP Change of representative

Representative=s name: PLOUGMANN 6 VINGTOFT POSTBOKS 1003 SENTRUM OSLO, 0

SPCF Filing of supplementary protection certificate

Free format text: PRODUCT NAME: MICAFUNGIN SODIUM; NAT. REG. NO/DATE: EU/1/08/448/001-002 20080521; FIRST REG. NO/DATE: 1/08/448/001-002 20080425

Spc suppl protection certif: 2010016

Filing date: 20100809

SPCG Granted supplementary protection certificate

Free format text: PRODUCT NAME: MICAFUNGIN SODIUM; NAT. REG. NO/DATE: EU/1/08/448/001-002 20080521; FIRST REG. NO/DATE: 1/08/448/001-002 20080425

Spc suppl protection certif: 2010016

Filing date: 20100809

Extension date: 20200929

MK1K Patent expired
SPCX Expiry of an spc

Spc suppl protection certif: 2010016

Effective date: 20201001