NO970831L - Nye substituerte piperidiner som er anvendbare for behandling av allergiske sykdommer - Google Patents
Nye substituerte piperidiner som er anvendbare for behandling av allergiske sykdommerInfo
- Publication number
- NO970831L NO970831L NO970831A NO970831A NO970831L NO 970831 L NO970831 L NO 970831L NO 970831 A NO970831 A NO 970831A NO 970831 A NO970831 A NO 970831A NO 970831 L NO970831 L NO 970831L
- Authority
- NO
- Norway
- Prior art keywords
- treatment
- allergic diseases
- useful
- new substituted
- substituted piperidines
- Prior art date
Links
- 208000026935 allergic disease Diseases 0.000 title abstract 2
- 150000003053 piperidines Chemical class 0.000 title abstract 2
- 208000036284 Rhinitis seasonal Diseases 0.000 abstract 2
- 208000035285 Allergic Seasonal Rhinitis Diseases 0.000 abstract 1
- 206010049153 Allergic sinusitis Diseases 0.000 abstract 1
- 229940122236 Histamine receptor antagonist Drugs 0.000 abstract 1
- 201000010105 allergic rhinitis Diseases 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 208000017022 seasonal allergic rhinitis Diseases 0.000 abstract 1
- 239000002462 tachykinin receptor antagonist Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Epidemiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29596094A | 1994-08-25 | 1994-08-25 | |
| US50191495A | 1995-07-13 | 1995-07-13 | |
| PCT/US1995/010640 WO1996006094A1 (en) | 1994-08-25 | 1995-08-17 | Novel substituted piperidines useful for the treatment of allergic diseases |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO970831D0 NO970831D0 (no) | 1997-02-24 |
| NO970831L true NO970831L (no) | 1997-04-18 |
| NO313237B1 NO313237B1 (no) | 2002-09-02 |
Family
ID=26969426
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19970831A NO313237B1 (no) | 1994-08-25 | 1997-02-24 | Nye substituerte piperidiner som er anvendbare for behandling av allergiske sykdommer og farmasöytisk preparat |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US6329392B1 (no) |
| EP (1) | EP0777666B1 (no) |
| JP (1) | JPH10504580A (no) |
| KR (1) | KR100362620B1 (no) |
| CN (1) | CN1067385C (no) |
| AT (1) | ATE177095T1 (no) |
| AU (1) | AU693936B2 (no) |
| CA (1) | CA2198084C (no) |
| DE (1) | DE69508093T2 (no) |
| DK (1) | DK0777666T3 (no) |
| ES (1) | ES2132709T3 (no) |
| FI (1) | FI114470B (no) |
| GR (1) | GR3030253T3 (no) |
| HU (1) | HU221434B (no) |
| IL (1) | IL115040A (no) |
| MX (1) | MX9701305A (no) |
| NO (1) | NO313237B1 (no) |
| NZ (1) | NZ292683A (no) |
| TW (1) | TW430663B (no) |
| WO (1) | WO1996006094A1 (no) |
Families Citing this family (68)
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| US6211199B1 (en) | 1995-11-17 | 2001-04-03 | Aventis Pharmaceuticals Inc. | Substituted 4-(1H-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases |
| NZ325581A (en) * | 1995-12-20 | 2000-03-27 | Hoechst Marion Roussel Inc | Substituted 4-(1h-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases |
| US6423704B2 (en) | 1995-12-20 | 2002-07-23 | Aventis Pharmaceuticals Inc. | Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases |
| US6194406B1 (en) | 1995-12-20 | 2001-02-27 | Aventis Pharmaceuticals Inc. | Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic disease |
| CN1143856C (zh) * | 1996-02-21 | 2004-03-31 | 阿温蒂斯药物公司 | 可用于治疗过敏性疾病的新的取代的 n－甲基 － n － ( 4 － ( 4 － ( 1 h－苯并咪唑 － 2 －基 ) [ 1 , 4 ]二氮杂环庚烷－1－基)－2－(芳基)丁基)苯甲酰胺类化合物 |
| US5932571A (en) * | 1996-02-21 | 1999-08-03 | Hoechst Marion Roussel, Inc. | Substituted N-methyl-N-(4-(4-(1H-benzimidazol-2-yl) {1,4}diazepan-1-yl)-2-(aryl) butyl) benzamides useful for the treatment of allergic diseases |
| US5998439A (en) | 1996-02-21 | 1999-12-07 | Hoescht Marion Roussel, Inc. | Substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases |
| PT888336E (pt) * | 1996-02-21 | 2002-12-31 | Aventis Pharma Inc | Novas n-metil-n-(4-(4-(1h-benzimidazol-2-il-amino)-piperidina-1-il)-2-(aril)-butil)-benzamidas substituidas uteis para o tratamento de doencas alergicas |
| FR2755133B1 (fr) * | 1996-10-31 | 1999-01-15 | Sanofi Sa | Nouveaux derives d'amides cycliques diversement substitues antagonistes selectifs du recepteur nk3 humain, procede pour leur obtention et compositions pharmaceutiques les contenant |
| FR2759584B1 (fr) * | 1997-02-17 | 1999-06-11 | Sanofi Sa | Composition pharmaceutique pour l'administration orale de composes heterocycliques sous forme ammonium quaternaire |
| FR2759585B1 (fr) | 1997-02-17 | 1999-06-11 | Sanofi Sa | Formulations pharmaceutiques presentees sous forme seche pour l'administration orale d'un compose ammonium quaternaire cyclique |
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-
1995
- 1995-08-17 ES ES95931551T patent/ES2132709T3/es not_active Expired - Lifetime
- 1995-08-17 NZ NZ292683A patent/NZ292683A/en unknown
- 1995-08-17 WO PCT/US1995/010640 patent/WO1996006094A1/en not_active Ceased
- 1995-08-17 AT AT95931551T patent/ATE177095T1/de not_active IP Right Cessation
- 1995-08-17 CA CA002198084A patent/CA2198084C/en not_active Expired - Fee Related
- 1995-08-17 AU AU34928/95A patent/AU693936B2/en not_active Ceased
- 1995-08-17 MX MX9701305A patent/MX9701305A/es unknown
- 1995-08-17 EP EP95931551A patent/EP0777666B1/en not_active Expired - Lifetime
- 1995-08-17 DE DE69508093T patent/DE69508093T2/de not_active Expired - Fee Related
- 1995-08-17 HU HU9701257A patent/HU221434B/hu not_active IP Right Cessation
- 1995-08-17 DK DK95931551T patent/DK0777666T3/da active
- 1995-08-17 KR KR1019970701189A patent/KR100362620B1/ko not_active Expired - Fee Related
- 1995-08-17 CN CN95195283A patent/CN1067385C/zh not_active Expired - Fee Related
- 1995-08-17 JP JP8508257A patent/JPH10504580A/ja not_active Ceased
- 1995-08-23 TW TW084108797A patent/TW430663B/zh not_active IP Right Cessation
- 1995-08-23 IL IL11504095A patent/IL115040A/xx not_active IP Right Cessation
-
1997
- 1997-02-24 NO NO19970831A patent/NO313237B1/no unknown
- 1997-02-24 FI FI970771A patent/FI114470B/fi not_active IP Right Cessation
-
1998
- 1998-05-15 US US09/079,924 patent/US6329392B1/en not_active Expired - Fee Related
-
1999
- 1999-05-19 GR GR990401346T patent/GR3030253T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| HUT76644A (en) | 1997-10-28 |
| WO1996006094A1 (en) | 1996-02-29 |
| JPH10504580A (ja) | 1998-05-06 |
| MX9701305A (es) | 1998-05-31 |
| ATE177095T1 (de) | 1999-03-15 |
| EP0777666B1 (en) | 1999-03-03 |
| CA2198084C (en) | 2000-03-28 |
| HU221434B (en) | 2002-10-28 |
| FI970771L (fi) | 1997-02-24 |
| IL115040A0 (en) | 1995-12-08 |
| KR970705556A (ko) | 1997-10-09 |
| GR3030253T3 (en) | 1999-08-31 |
| DK0777666T3 (da) | 1999-09-27 |
| AU693936B2 (en) | 1998-07-09 |
| CN1067385C (zh) | 2001-06-20 |
| FI114470B (fi) | 2004-10-29 |
| US6329392B1 (en) | 2001-12-11 |
| NO313237B1 (no) | 2002-09-02 |
| AU3492895A (en) | 1996-03-14 |
| NO970831D0 (no) | 1997-02-24 |
| IL115040A (en) | 2000-02-29 |
| TW430663B (en) | 2001-04-21 |
| NZ292683A (en) | 1998-07-28 |
| DE69508093T2 (de) | 1999-07-15 |
| FI970771A0 (fi) | 1997-02-24 |
| KR100362620B1 (ko) | 2003-02-14 |
| ES2132709T3 (es) | 1999-08-16 |
| DE69508093D1 (de) | 1999-04-08 |
| EP0777666A1 (en) | 1997-06-11 |
| CN1158612A (zh) | 1997-09-03 |
| CA2198084A1 (en) | 1996-02-29 |
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