NO329559B1 - Fremgangsmate for a fremstille modafinil - Google Patents

Fremgangsmate for a fremstille modafinil Download PDF

Info

Publication number: NO329559B1
Authority: NO; Norway
Prior art keywords: equivalents; modafinil; acid; reacting; aqueous
Prior art date: 2002-05-23

Application number

NO20044916A

Other languages

English (en)

Norwegian (no)

Other versions

NO20044916L (no

Inventor

Denis Largeau

Gilles Oddon

Original Assignee

Cephalon Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-05-23

Filing date

2004-11-11

Publication date

2010-11-15

2004-11-11 Application filed by Cephalon Inc filed Critical Cephalon Inc

2004-12-16 Publication of NO20044916L publication Critical patent/NO20044916L/no

2010-11-15 Publication of NO329559B1 publication Critical patent/NO329559B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/02—Preparation of sulfones; Preparation of sulfoxides by formation of sulfone or sulfoxide groups by oxidation of sulfides, or by formation of sulfone groups by oxidation of sulfoxides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
- A61K31/10—Sulfides; Sulfoxides; Sulfones
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
- C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

NO20044916A 2002-05-23 2004-11-11 Fremgangsmate for a fremstille modafinil NO329559B1 (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US38317302P	2002-05-23	2002-05-23
US10/443,327 US6875893B2 (en)	2002-05-23	2003-05-22	Preparations of a sulfinyl acetamide
PCT/US2003/016379 WO2003099774A1 (en)	2002-05-23	2003-05-23	Preparations of a sulfinyl acetamide

Publications (2)

Publication Number	Publication Date
NO20044916L NO20044916L (no)	2004-12-16
NO329559B1 true NO329559B1 (no)	2010-11-15

Family

ID=29586987

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20044916A NO329559B1 (no)	2002-05-23	2004-11-11	Fremgangsmate for a fremstille modafinil

Country Status (29)

Country	Link
US (2)	US6875893B2 (zh)
EP (1)	EP1506171B1 (zh)
JP (1)	JP4351627B2 (zh)
KR (1)	KR100984571B1 (zh)
CN (1)	CN100379721C (zh)
AR (1)	AR039857A1 (zh)
AT (1)	ATE414058T1 (zh)
BR (1)	BR0311242A (zh)
CA (1)	CA2486533C (zh)
CY (1)	CY1108747T1 (zh)
DE (1)	DE60324671D1 (zh)
DK (1)	DK1506171T3 (zh)
EA (1)	EA007561B1 (zh)
EG (1)	EG23693A (zh)
ES (1)	ES2316755T3 (zh)
HK (1)	HK1072596A1 (zh)
IL (2)	IL165095A0 (zh)
IS (1)	IS2650B (zh)
MX (1)	MXPA04011459A (zh)
MY (1)	MY129141A (zh)
NO (1)	NO329559B1 (zh)
NZ (1)	NZ536747A (zh)
PL (1)	PL211695B1 (zh)
PT (1)	PT1506171E (zh)
SI (1)	SI1506171T1 (zh)
TW (1)	TWI317733B (zh)
UA (1)	UA79790C2 (zh)
WO (1)	WO2003099774A1 (zh)
ZA (1)	ZA200409400B (zh)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
MXPA03000747A (es) *	2000-07-27	2003-06-04	Teva Pharma	Modafinilo cristalino y puro y proceso para prepararlo.
US6875893B2 (en) *	2002-05-23	2005-04-05	Cephalon, Inc.	Preparations of a sulfinyl acetamide
US6992219B2 (en) *	2002-08-09	2006-01-31	Cephalon France	Modafinil polymorphic forms
FR2849029B1 (fr) *	2002-12-20	2005-03-18	Lafon Labor	Procede de preparation et formes cristallines des enantiomeres optiques du modafinil.
JP2006518754A (ja) *	2003-02-24	2006-08-17	マリンクロッド・インコーポレイテッド	ベンズヒドリルチオアセトアミドの改良製法
US20040253308A1 (en) *	2003-04-29	2004-12-16	Barr Laboratories, Inc.	Surface-treated modafinil particles
US7368591B2 (en)	2003-09-19	2008-05-06	Cephalon France	Process for enantioselective synthesis of single enantiomers of modafinil by asymmetric oxidation
DK1678129T3 (da) *	2003-10-23	2009-02-09	Mallinckrodt Inc	Forbedret fremgangsmåde til fremstilling af benzhydrylthioacetamid
US20060086667A1 (en) *	2004-09-13	2006-04-27	Cephalon, Inc., U.S. Corporation	Methods for the separation of enantiomeric sulfinylacetamides
US7939629B2 (en)	2004-10-19	2011-05-10	Lonza Ag	Method for solid phase peptide synthesis
US20090123545A1 (en) *	2005-07-21	2009-05-14	Ron Eyal S	Rapid Onset and Short Term Modafinil Compositions and Methods of Use Thereof
US7553646B2 (en) *	2005-07-28	2009-06-30	University Of Iowa Research Foundation	Microbial sulfoxidation and amidation of benzhdrylsulfanyl carboxylic acids and uses thereof
CA2618494A1 (en) *	2005-09-14	2007-03-22	Novetide, Ltd.	Process for production of bivalirudin
CN101326159A (zh) *	2005-12-09	2008-12-17	马林克罗特公司	制备莫达非尼及其类似物的方法
CN100343228C (zh) *	2006-02-17	2007-10-17	中国科学院上海有机化学研究所	高对映体选择性制备 2－二苯甲基亚磺酰基－乙酰胺单一对映体的方法
KR20070119037A (ko) *	2006-02-21	2007-12-18	테바 파마슈티컬 인더스트리즈 리미티드	아르모다피닐의 신규한 결정질 형태 및 이것의 제조 방법
CA2634133A1 (en) *	2006-03-01	2007-09-13	Teva Pharmaceutical Industries Ltd.	An improved process for the preparation of armodafinil
GB0604233D0 (en) *	2006-03-02	2006-04-12	Syngenta Participations Ag	Process
JP2009543803A (ja) *	2006-07-12	2009-12-10	エラン・ファルマ・インターナショナル・リミテッド	モダフィニルのナノ粒子製剤
EP2056811B8 (en) *	2006-08-14	2018-03-21	Neurohealing Pharmaceuticals, Inc.	Modafinil-based treatment for premature ejaculation
US7960586B2 (en) *	2007-08-16	2011-06-14	Teva Pharmaceutical Industries Ltd.	Purification of armodafinil
US20100036164A1 (en) *	2008-08-06	2010-02-11	Srinivas Areveli	Preparation of armodafinil form i
CN102976985A (zh) *	2011-09-07	2013-03-20	大连大学	一锅法合成二苯甲基亚磺酰基乙酰胺及其类似物的方法
CN105992734A (zh) *	2014-02-06	2016-10-05	比勒鲁迪克斯那斯公司	由可拉伸的纸构成的直立袋

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1520812A (en) *	1975-10-02	1978-08-09	Lafon Labor	Benzhydrylsulphinyl derivatives
GB1584462A (en) *	1977-03-31	1981-02-11	Lafon Labor	N-diaryl-malonamide and diarylmethyl-sulphinyl-acetamide derivatives and pharmaceutical compositions containing them
FR2593809B1 (fr) *	1986-01-31	1988-07-22	Lafon Labor	Benzhydrylsulfinylacetamide, procede de preparation et utilisation en therapeutique
US20030187023A1 (en)	2000-07-17	2003-10-02	Keiji Kubo	Sulfone derivatives, process for their production and use thereof
MXPA03000747A (es)	2000-07-27	2003-06-04	Teva Pharma	Modafinilo cristalino y puro y proceso para prepararlo.
IL143106A (en)	2001-05-13	2005-11-20	Chemagis Ltd	Process for the preparation of diphenylmethylthioacetamide
US6875893B2 (en) *	2002-05-23	2005-04-05	Cephalon, Inc.	Preparations of a sulfinyl acetamide
DE10245546B3 (de) *	2002-09-30	2004-05-13	Infineon Technologies Ag	Pseudostatische Speicherschaltung
JP3838972B2 (ja) *	2002-12-25	2006-10-25	Ｎｅｃエレクトロニクス株式会社	周波数検出回路及びデータ処理装置

2003
- 2003-05-22 US US10/443,327 patent/US6875893B2/en not_active Expired - Lifetime
- 2003-05-23 CN CNB038118386A patent/CN100379721C/zh not_active Expired - Fee Related
- 2003-05-23 DE DE60324671T patent/DE60324671D1/de not_active Expired - Lifetime
- 2003-05-23 UA UA20041210602A patent/UA79790C2/uk unknown
- 2003-05-23 JP JP2004507432A patent/JP4351627B2/ja not_active Expired - Lifetime
- 2003-05-23 WO PCT/US2003/016379 patent/WO2003099774A1/en active Application Filing
- 2003-05-23 KR KR1020047018819A patent/KR100984571B1/ko not_active IP Right Cessation
- 2003-05-23 PL PL373792A patent/PL211695B1/pl unknown
- 2003-05-23 IL IL16509503A patent/IL165095A0/xx unknown
- 2003-05-23 AR ARP030101796A patent/AR039857A1/es not_active Application Discontinuation
- 2003-05-23 DK DK03729108T patent/DK1506171T3/da active
- 2003-05-23 CA CA2486533A patent/CA2486533C/en not_active Expired - Fee Related
- 2003-05-23 BR BR0311242-0A patent/BR0311242A/pt not_active Application Discontinuation
- 2003-05-23 TW TW092113924A patent/TWI317733B/zh not_active IP Right Cessation
- 2003-05-23 MY MYPI20031924A patent/MY129141A/en unknown
- 2003-05-23 EA EA200401551A patent/EA007561B1/ru not_active IP Right Cessation
- 2003-05-23 EP EP03729108A patent/EP1506171B1/en not_active Expired - Lifetime
- 2003-05-23 AT AT03729108T patent/ATE414058T1/de active
- 2003-05-23 SI SI200331442T patent/SI1506171T1/sl unknown
- 2003-05-23 NZ NZ536747A patent/NZ536747A/en not_active IP Right Cessation
- 2003-05-23 US US11/091,215 patent/US7057069B2/en not_active Expired - Fee Related
- 2003-05-23 ES ES03729108T patent/ES2316755T3/es not_active Expired - Lifetime
- 2003-05-23 MX MXPA04011459A patent/MXPA04011459A/es active IP Right Grant
- 2003-05-23 PT PT03729108T patent/PT1506171E/pt unknown
2004
- 2004-11-08 IL IL165095A patent/IL165095A/en active IP Right Grant
- 2004-11-09 IS IS7523A patent/IS2650B/is unknown
- 2004-11-11 NO NO20044916A patent/NO329559B1/no not_active IP Right Cessation
- 2004-11-21 EG EGNA2004000127 patent/EG23693A/xx active
- 2004-11-22 ZA ZA2004/09400A patent/ZA200409400B/en unknown
2005
- 2005-06-29 HK HK05105443.7A patent/HK1072596A1/xx not_active IP Right Cessation
2009
- 2009-02-04 CY CY20091100129T patent/CY1108747T1/el unknown

Also Published As

Publication number	Publication date
EG23693A (en)	2007-05-15
KR100984571B1 (ko)	2010-09-30
AR039857A1 (es)	2005-03-02
DK1506171T3 (da)	2009-01-19
EP1506171A1 (en)	2005-02-16
EA200401551A1 (ru)	2005-04-28
UA79790C2 (en)	2007-07-25
CA2486533C (en)	2011-01-04
SI1506171T1 (sl)	2009-06-30
IS7523A (is)	2004-11-09
ATE414058T1 (de)	2008-11-15
CN100379721C (zh)	2008-04-09
IS2650B (is)	2010-08-15
CA2486533A1 (en)	2003-12-04
US7057069B2 (en)	2006-06-06
PL211695B1 (pl)	2012-06-29
WO2003099774A1 (en)	2003-12-04
IL165095A (en)	2010-11-30
TWI317733B (en)	2009-12-01
US20040002547A1 (en)	2004-01-01
US6875893B2 (en)	2005-04-05
ES2316755T3 (es)	2009-04-16
AU2003233668A1 (en)	2003-12-12
KR20050016421A (ko)	2005-02-21
CN1656064A (zh)	2005-08-17
DE60324671D1 (de)	2008-12-24
US20050171209A1 (en)	2005-08-04
ZA200409400B (en)	2005-12-28
PL373792A1 (en)	2005-09-19
EP1506171B1 (en)	2008-11-12
TW200406196A (en)	2004-05-01
HK1072596A1 (en)	2005-09-02
JP2005527623A (ja)	2005-09-15
JP4351627B2 (ja)	2009-10-28
NZ536747A (en)	2006-11-30
MY129141A (en)	2007-03-30
MXPA04011459A (es)	2005-02-14
EA007561B1 (ru)	2006-12-29
BR0311242A (pt)	2005-03-15
CY1108747T1 (el)	2014-04-09
PT1506171E (pt)	2009-01-02
IL165095A0 (en)	2005-12-18
NO20044916L (no)	2004-12-16

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Legal Events

Date	Code	Title	Description
2018-12-27	MM1K	Lapsed by not paying the annual fees