NO326497B1 - Arylsulfonylderivater med 5-HT6 reseptor affinitet, farmasoytisk medikament omfattende slike, fremgangsmate for fremstilling av slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom - Google Patents

Arylsulfonylderivater med 5-HT6 reseptor affinitet, farmasoytisk medikament omfattende slike, fremgangsmate for fremstilling av slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom Download PDF

Info

Publication number: NO326497B1
Authority: NO; Norway
Prior art keywords: methoxy; phenyl; compound; piperazine; benzenesulfonyl
Prior art date: 2001-08-10

Application number

NO20040589A

Other languages

English (en)

Norwegian (no)

Other versions

NO20040589L (no

Inventor

Jacob Berger

Shu-Hai Zhao

Robin Douglas Clark

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-08-10

Filing date

2004-02-09

Publication date

2008-12-15

2004-02-09 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2004-03-19 Publication of NO20040589L publication Critical patent/NO20040589L/no

2008-12-15 Publication of NO326497B1 publication Critical patent/NO326497B1/no

Links

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Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
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Addiction (AREA)
Psychiatry (AREA)
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Psychology (AREA)
Obesity (AREA)
Orthopedic Medicine & Surgery (AREA)
Hematology (AREA)
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Child & Adolescent Psychology (AREA)
Anesthesiology (AREA)
Nutrition Science (AREA)
Hospice & Palliative Care (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Compositions Of Macromolecular Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Photoreceptors In Electrophotography (AREA)

NO20040589A 2001-08-10 2004-02-09 Arylsulfonylderivater med 5-HT6 reseptor affinitet, farmasoytisk medikament omfattende slike, fremgangsmate for fremstilling av slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom NO326497B1 (no)

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US31150401P	2001-08-10	2001-08-10
US38471102P	2002-05-31	2002-05-31
PCT/EP2002/008696 WO2003014097A1 (en)	2001-08-10	2002-08-05	Arylsulfonyl derivatives with 5-ht6 receptor affinity

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NO326497B1 true NO326497B1 (no)	2008-12-15

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US (1)	US6825202B2 (ru)
EP (1)	EP1423106B1 (ru)
JP (1)	JP4187650B2 (ru)
KR (1)	KR100608417B1 (ru)
CN (1)	CN1254469C (ru)
AT (1)	ATE417838T1 (ru)
AU (1)	AU2002340804B2 (ru)
CA (1)	CA2456250A1 (ru)
CO (1)	CO5550439A2 (ru)
DE (1)	DE60230424D1 (ru)
ES (1)	ES2316619T3 (ru)
HK (1)	HK1070054A1 (ru)
HR (1)	HRP20040090A2 (ru)
HU (1)	HUP0401235A2 (ru)
IL (1)	IL159880A0 (ru)
MX (1)	MXPA04001250A (ru)
NO (1)	NO326497B1 (ru)
NZ (1)	NZ530742A (ru)
PL (1)	PL373397A1 (ru)
RU (1)	RU2268884C2 (ru)
WO (1)	WO2003014097A1 (ru)

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DK1497266T3 (da)	2002-03-27	2008-10-06	Glaxo Group Ltd	Quinolinderivater og deres anvendelse som 5HT6-ligander
TWI285639B (en) *	2002-11-08	2007-08-21	Roche Palo Alto Llc	Substituted benzoxazinones and uses thereof
TWI289141B (en)	2003-03-11	2007-11-01	Hoffmann La Roche F. Ag.	Quinolinone derivatives and uses thereof
GB0305575D0 (en) *	2003-03-11	2003-04-16	Glaxo Group Ltd	Novel compounds
ATE313532T1 (de)	2003-07-22	2006-01-15	Arena Pharm Inc	Diaryl- und arylheteroarylharnstoffderivate als modulatoren des 5-ht2a-serotoninrezeptors, die sich zur prophylaxe und behandlung von damit im zusammenhang stehenden erkrankungen eignen
WO2006062481A1 (en) *	2004-12-09	2006-06-15	Biovitrum Ab	New benzofuran derivatives and their use in the treatment of obesity, type ii diabetes and cns disorders .
ES2337482T3 (es) *	2004-12-21	2010-04-26	F. Hoffmann-La Roche Ag	Derivados de tetralina y de indano y usos de los mismos.
EP1695971A1 (en) *	2004-12-30	2006-08-30	Laboratorios Del Dr. Esteve, S.A.	Substituted phenyl-piperazine compounds, their preparation and use in medicaments
EP2254564A1 (en)	2007-12-12	2010-12-01	Glaxo Group Limited	Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline
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2002
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Publication number	Publication date
US6825202B2 (en)	2004-11-30
IL159880A0 (en)	2004-06-20
JP2005502649A (ja)	2005-01-27
CN1254469C (zh)	2006-05-03
HK1070054A1 (en)	2005-06-10
KR20040023738A (ko)	2004-03-18
AU2002340804B2 (en)	2008-04-03
NZ530742A (en)	2007-07-27
EP1423106B1 (en)	2008-12-17
JP4187650B2 (ja)	2008-11-26
ES2316619T3 (es)	2009-04-16
PL373397A1 (en)	2005-08-22
CO5550439A2 (es)	2005-08-31
CN1541210A (zh)	2004-10-27
MXPA04001250A (es)	2004-05-27
DE60230424D1 (en)	2009-01-29
WO2003014097A1 (en)	2003-02-20
ATE417838T1 (de)	2009-01-15
RU2268884C2 (ru)	2006-01-27
US20030069254A1 (en)	2003-04-10
KR100608417B1 (ko)	2006-08-02
HRP20040090A2 (en)	2004-12-31
HUP0401235A2 (hu)	2004-10-28
RU2004107261A (ru)	2005-09-10
CA2456250A1 (en)	2003-02-20
EP1423106A1 (en)	2004-06-02
NO20040589L (no)	2004-03-19

Publication	Publication Date	Title
NO326497B1 (no)	2008-12-15	Arylsulfonylderivater med 5-HT6 reseptor affinitet, farmasoytisk medikament omfattende slike, fremgangsmate for fremstilling av slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom
EP1401812B1 (en)	2006-06-28	4-piperazinylindole derivatives with 5-ht6 receptor affinity
KR20090092832A (ko)	2009-09-01	비만, 제 ⅱ 형 당뇨병 및 ｃｎｓ 장애의 치료를 위한 신규한 아릴술폰아미드 화합물
US6774241B2 (en)	2004-08-10	1-sulfonyl-4-aminoalkoxy indole derivatives and uses thereof
AU2002340804A1 (en)	2003-06-19	Arylsulfonyl derivatives with 5-HT6 receptor affinity
MX2011011520A (es)	2012-06-19	Compuestos de n-fenil-(piperazinil u homopiperazinil)-bencensulfon amida o bencensulfonil-fenil-(piperazina u homopiperazina) adecuados para tratar trastornos que responden a la modulacion del receptor de serotonina 5-ht6.
JP4339795B2 (ja)	2009-10-07	Ｃｎｓ障害の治療のための５−ｈｔ６レセプターリガンドとしてのアミノアルコキシインドール
JP2008524277A (ja)	2008-07-10	テトラリン及びインダン誘導体、並びにそれらの５−ｈｔ拮抗薬としての使用
EP1910296B1 (en)	2010-04-21	4-aryloxy quinoline derivatives as 5-ht6 modulators
SK137597A3 (en)	1998-05-06	1-£'omega'-(3,4-dihydro-2-naphthalenyl)alkyl\| cyclic amine derivatives, process for producing the same, and medicinal composition containing the same
ZA200400749B (en)	2005-04-29	Arylsulfonyl derivatives with 5-HT6 receptor affinity.
KR100922486B1 (ko)	2009-10-20	비만, 제 ⅱ 형 당뇨병 및 ｃｎｓ 장애의 치료를 위한신규한 아릴술폰아미드 화합물
JP2008524274A (ja)	2008-07-10	テトラリン及びインダン誘導体、並びにそれらの使用
AU2002345587A1 (en)	2003-01-02	4-Piperazinylindole derivatives with 5-HT6 receptor affinity
MXPA06005840A (en)	2006-10-17	Benzoxazine derivatives and uses thereof

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