NO305025B1 - FremgangsmÕte for fremstilling av piperidinderivater - Google Patents

FremgangsmÕte for fremstilling av piperidinderivater

Info

Publication number: NO305025B1
Authority: NO; Norway
Prior art keywords: preparation; piperidine derivatives; piperidine; derivatives
Prior art date: 1992-04-10

Application number

NO981434A

Other languages

English (en)

Other versions

NO981434L (no

NO981434D0 (no

Inventor

Michele Ann Kaminski

Chi-Hsin Richard King

Original Assignee

Merrell Dow Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-04-10

Filing date

1998-03-30

Publication date

1999-03-22

1994-12-09 Publication of NO981434L publication Critical patent/NO981434L/no

1998-03-30 Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma

1998-03-30 Publication of NO981434D0 publication Critical patent/NO981434D0/no

1999-03-22 Publication of NO305025B1 publication Critical patent/NO305025B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Hydrogenated Pyridines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

NO981434A 1992-04-10 1998-03-30 FremgangsmÕte for fremstilling av piperidinderivater NO305025B1 (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US86726192A	1992-04-10	1992-04-10
US1725193A	1993-02-25	1993-02-25
PCT/US1993/002103 WO1993021156A1 (en)	1992-04-10	1993-03-10	4-diphenylmethyl piperidine derivatives and process for their preparation

Publications (3)

Publication Number	Publication Date
NO981434L NO981434L (no)	1994-12-09
NO981434D0 NO981434D0 (no)	1998-03-30
NO305025B1 true NO305025B1 (no)	1999-03-22

Family

ID=26689638

Family Applications (5)

Application Number	Title	Priority Date	Filing Date
NO943794A NO305076B1 (no)	1992-04-10	1994-10-07	FremgangsmÕte for fremstilling av en piperidinformylfenylketonforbindelse
NO981434A NO305025B1 (no)	1992-04-10	1998-03-30	FremgangsmÕte for fremstilling av piperidinderivater
NO981431A NO305023B1 (no)	1992-04-10	1998-03-30	FremgangsmÕte for fremstilling av piperidinderivater
NO981433A NO305024B1 (no)	1992-04-10	1998-03-30	FremgangsmÕte for fremstilling av piperidinderivater
NO981432A NO305077B1 (no)	1992-04-10	1998-03-30	FremgangsmÕte for fremstilling av piperidinderivater

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
NO943794A NO305076B1 (no)	1992-04-10	1994-10-07	FremgangsmÕte for fremstilling av en piperidinformylfenylketonforbindelse

Family Applications After (3)

Application Number	Title	Priority Date	Filing Date
NO981431A NO305023B1 (no)	1992-04-10	1998-03-30	FremgangsmÕte for fremstilling av piperidinderivater
NO981433A NO305024B1 (no)	1992-04-10	1998-03-30	FremgangsmÕte for fremstilling av piperidinderivater
NO981432A NO305077B1 (no)	1992-04-10	1998-03-30	FremgangsmÕte for fremstilling av piperidinderivater

Country Status (19)

Country	Link
EP (1)	EP0635004B1 (no)
JP (3)	JP3686950B2 (no)
KR (1)	KR100257805B1 (no)
AR (1)	AR253777A1 (no)
AT (1)	ATE220666T1 (no)
AU (1)	AU671822B2 (no)
CA (1)	CA2117892C (no)
DE (1)	DE69332117T2 (no)
DK (1)	DK0635004T3 (no)
ES (1)	ES2176201T3 (no)
FI (2)	FI106454B (no)
HU (1)	HU226561B1 (no)
IL (1)	IL105328A (no)
MX (1)	MX9302076A (no)
NO (5)	NO305076B1 (no)
NZ (1)	NZ251132A (no)
PT (1)	PT635004E (no)
TW (1)	TW362096B (no)
WO (1)	WO1993021156A1 (no)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
RU2167657C2 (ru) *	1992-08-03	2001-05-27	Сепракор, Инк.	Фармацевтическая композиция для лечения аллергических заболеваний, способ антигистаминного лечения, применение композиции для получения лекарственного препарата
EP0723958A1 (en) *	1993-06-24	1996-07-31	Albany Molecular Research, Inc.	Synthesis of substantially pure terfenadine derivatives
US20020007068A1 (en)	1999-07-16	2002-01-17	D'ambra Thomas E.	Piperidine derivatives and process for their production
AU699559B2 (en)	1993-06-25	1998-12-10	Aventisub Ii Inc.	Novel intermediates for the preparation of antihistaminic piperidine derivatives
US6147216A (en) *	1993-06-25	2000-11-14	Merrell Pharmaceuticals Inc.	Intermediates useful for the preparation of antihistaminic piperidine derivatives
JPH10500134A (ja)	1994-05-18	1998-01-06	ヘキスト・マリオン・ルセル・インコーポレイテツド	抗ヒスタミン性ピペリジン誘導体の無水および水和形態、それらの多形態および擬似形態の製造方法
EP0812195B1 (en)	1995-02-28	2002-10-30	Aventis Pharmaceuticals Inc.	Pharmaceutical composition for piperidinoalkanol compounds
US6201124B1 (en)	1995-12-21	2001-03-13	Albany Molecular Research, Inc.	Process for production of piperidine derivatives
US6153754A (en) *	1995-12-21	2000-11-28	Albany Molecular Research, Inc.	Process for production of piperidine derivatives
DK1091938T3 (da) *	1998-07-02	2011-02-07	Aventisub Ii Inc	Antihistamin piperidinderivativer og mellemprodukter til fremstilling af disse
AU2002305162A1 (en) *	2001-04-09	2002-10-21	Teva Pharmaceutical Industries Ltd.	Polymorphs of fexofenadine hydrochloride
ITRM20010260A1 (it)	2001-05-17	2002-11-18	Dinamite Dipharma S P A In For	Processo per la preparazione della fexofenadina o acido 4 1-idrossi-4-4- (idrossidifenilmetil)-1-piperidinil\|-butil\|-alfa,alfa-dimetilbenz
US6743941B2 (en) *	2001-06-15	2004-06-01	Aventis Pharma Deutschland Gmbh	Process for the production of piperidine derivatives
DE03757471T1 (de)	2002-06-10	2005-09-01	Teva Pharmaceutical Industries Ltd.	Polymorphe form xvi von fexofenadin-hydrochlorid
GB0319935D0 (en)	2003-08-26	2003-09-24	Cipla Ltd	Polymorphs
ITMI20061492A1 (it) *	2006-07-27	2008-01-28	Archimica Srl	Processo per la preparazione di fexofenadina.
ITMI20070987A1 (it)	2007-05-16	2008-11-17	Dipharma Francis Srl	Procedimento per la preparazione di composti chetonici
EP2289867A3 (en)	2009-08-19	2012-04-25	Jubilant Organosys Limited	A process for producing 4-(4-halo-1-oxybutyl)-alpha,alpha-dimethylbenzene acetic acid or alkyl esters thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4254129A (en) *	1979-04-10	1981-03-03	Richardson-Merrell Inc.	Piperidine derivatives
US4254130A (en) *	1979-04-10	1981-03-03	Richardson-Merrell Inc.	Piperidine derivatives

1993
- 1993-03-10 WO PCT/US1993/002103 patent/WO1993021156A1/en active IP Right Grant
- 1993-03-10 ES ES93907333T patent/ES2176201T3/es not_active Expired - Lifetime
- 1993-03-10 AU AU37973/93A patent/AU671822B2/en not_active Expired
- 1993-03-10 AT AT93907333T patent/ATE220666T1/de active
- 1993-03-10 JP JP51831393A patent/JP3686950B2/ja not_active Expired - Lifetime
- 1993-03-10 KR KR1019940703575A patent/KR100257805B1/ko not_active IP Right Cessation
- 1993-03-10 DK DK93907333T patent/DK0635004T3/da active
- 1993-03-10 CA CA002117892A patent/CA2117892C/en not_active Expired - Lifetime
- 1993-03-10 MX MX9302076A patent/MX9302076A/es unknown
- 1993-03-10 HU HU9402913A patent/HU226561B1/hu unknown
- 1993-03-10 PT PT93907333T patent/PT635004E/pt unknown
- 1993-03-10 NZ NZ251132A patent/NZ251132A/en not_active IP Right Cessation
- 1993-03-10 DE DE69332117T patent/DE69332117T2/de not_active Expired - Lifetime
- 1993-03-10 EP EP93907333A patent/EP0635004B1/en not_active Expired - Lifetime
- 1993-04-07 AR AR25377793A patent/AR253777A1/es unknown
- 1993-04-07 TW TW082102558A patent/TW362096B/zh not_active IP Right Cessation
- 1993-04-07 IL IL105328A patent/IL105328A/en not_active IP Right Cessation
1994
- 1994-10-07 FI FI944713A patent/FI106454B/fi not_active IP Right Cessation
- 1994-10-07 NO NO943794A patent/NO305076B1/no not_active IP Right Cessation
1998
- 1998-03-30 NO NO981434A patent/NO305025B1/no not_active IP Right Cessation
- 1998-03-30 NO NO981431A patent/NO305023B1/no not_active IP Right Cessation
- 1998-03-30 NO NO981433A patent/NO305024B1/no not_active IP Right Cessation
- 1998-03-30 NO NO981432A patent/NO305077B1/no not_active IP Right Cessation
2000
- 2000-11-09 FI FI20002460A patent/FI20002460A/fi unknown
2004
- 2004-05-06 JP JP2004137675A patent/JP4266184B2/ja not_active Expired - Lifetime
2005
- 2005-04-01 JP JP2005105603A patent/JP2005213268A/ja active Pending

Also Published As

Publication number	Publication date
ES2176201T3 (es)	2002-12-01
NO943794D0 (no)	1994-10-07
DK0635004T3 (da)	2002-11-11
JP3686950B2 (ja)	2005-08-24
NO981433D0 (no)	1998-03-30
NO305023B1 (no)	1999-03-22
AR253777A1 (es)	2001-10-08
HU9402913D0 (en)	1995-01-30
NO981432D0 (no)	1998-03-30
AU671822B2 (en)	1996-09-12
FI944713A0 (fi)	1994-10-07
HU226561B1 (en)	2009-04-28
IL105328A (en)	2007-03-08
JP4266184B2 (ja)	2009-05-20
KR950700881A (ko)	1995-02-20
MX9302076A (es)	1994-03-31
WO1993021156A1 (en)	1993-10-28
HUT70517A (en)	1995-10-30
FI944713A (fi)	1994-12-02
JP2004285072A (ja)	2004-10-14
CA2117892C (en)	2001-12-18
NO981431L (no)	1994-12-09
DE69332117T2 (de)	2003-01-30
KR100257805B1 (ko)	2000-07-01
IL105328A0 (en)	1993-08-18
NO981434L (no)	1994-12-09
EP0635004A1 (en)	1995-01-25
DE69332117D1 (de)	2002-08-22
FI20002460A (fi)	2000-11-09
NO981434D0 (no)	1998-03-30
ATE220666T1 (de)	2002-08-15
TW362096B (en)	1999-06-21
NO305077B1 (no)	1999-03-29
CA2117892A1 (en)	1993-10-28
JPH08502022A (ja)	1996-03-05
NZ251132A (en)	1996-12-20
EP0635004B1 (en)	2002-07-17
NO943794L (no)	1994-12-09
NO981433L (no)	1994-12-09
FI106454B (fi)	2001-02-15
PT635004E (pt)	2002-12-31
NO981431D0 (no)	1998-03-30
AU3797393A (en)	1993-11-18
NO305076B1 (no)	1999-03-29
NO305024B1 (no)	1999-03-22
JP2005213268A (ja)	2005-08-11
NO981432L (no)	1994-12-09

Publication	Publication Date	Title
FI945441A0 (fi)	1994-11-18	Uusi menetelmä 7beta-substituoitu-4-atsa-5alfa-androstan-3-onien valmistamiseksi
NO981432L (no)	1994-12-09	FremgangsmÕte for fremstilling av piperidinderivater
FI940769A (fi)	1994-08-20	Menetelmä 2-aminoatsolijohdannaisten valmistamiseksi
NO931346D0 (no)	1993-04-07	Fremgangsmaate for fremstilling av et bifenylderivat
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NO306717B1 (no)	1999-12-13	Fremgangsmåte for fremstilling av piperidin-karbinoler
NO179517C (no)	1996-10-23	Fremgangsmåte for fremstilling av 8-klorkinolonderivater
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NO972129D0 (no)	1997-05-07	Fremgangsmåte for fremstilling av 1-halo-3-trialkylsilanyl-benzenderivater
FI943660A0 (fi)	1994-08-05	Menetelmä 3-karbonyyliandrostadieeni-17-karboksamidien valmistamiseksi
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NO911665D0 (no)	1991-04-26	Fremgangsmaate for fremstilling av nye nojirimycinderivater
NO177305C (no)	1995-08-23	Fremgangsmåte for fremstilling av 3-substituerte-2-oksindol-derivater
NO180301C (no)	1997-03-26	Fremgangsmåte for fremstilling av azaspiroalkanderivater
NO960829D0 (no)	1996-02-29	Fremgangsmåte for fresmtilling av 13-alkyl-11 r
FI932887A (fi)	1994-12-23	Parannettu menetelmä 4-nitro-3-trifluorometyylianiliinin valmistamiseksi
NO943237D0 (no)	1994-09-01	Fremgangsmåte for fremstilling av benzotiazepinderivater
NO950203D0 (no)	1995-01-19	Fremgangsmåte for fremstilling av propargylazetidion-forbindelser
FI902356A0 (fi)	1990-05-11	Tieno-triatsolo-diatsepiinijohdosten valmistusmenetelmä

Legal Events

Date	Code	Title	Description
2013-04-15	MK1K	Patent expired