NO302119B1 - Imidazolforbindelser, farmasöytiske preparater som omfatter en slik forbindelse, samt anvendelser derav for fremstilling av farmasöytiske preparater - Google Patents
Imidazolforbindelser, farmasöytiske preparater som omfatter en slik forbindelse, samt anvendelser derav for fremstilling av farmasöytiske preparater Download PDFInfo
- Publication number
- NO302119B1 NO302119B1 NO922475A NO922475A NO302119B1 NO 302119 B1 NO302119 B1 NO 302119B1 NO 922475 A NO922475 A NO 922475A NO 922475 A NO922475 A NO 922475A NO 302119 B1 NO302119 B1 NO 302119B1
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- Prior art keywords
- branched
- alkyl
- chain
- straight
- hydrogen
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Classifications
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- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
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- C07D235/30—Nitrogen atoms not forming part of a nitro radical
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- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Lubricants (AREA)
- Eye Examination Apparatus (AREA)
- Magnetic Resonance Imaging Apparatus (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US72002191A | 1991-06-24 | 1991-06-24 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO922475D0 NO922475D0 (no) | 1992-06-23 |
| NO922475L NO922475L (no) | 1992-12-28 |
| NO302119B1 true NO302119B1 (no) | 1998-01-26 |
Family
ID=24892332
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO922475A NO302119B1 (no) | 1991-06-24 | 1992-06-23 | Imidazolforbindelser, farmasöytiske preparater som omfatter en slik forbindelse, samt anvendelser derav for fremstilling av farmasöytiske preparater |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP0520200B1 (el) |
| JP (1) | JPH05186432A (el) |
| AT (1) | ATE163290T1 (el) |
| AU (1) | AU653816B2 (el) |
| CA (1) | CA2071793A1 (el) |
| DE (1) | DE69224448T2 (el) |
| DK (1) | DK0520200T3 (el) |
| ES (1) | ES2113898T3 (el) |
| FI (1) | FI922905L (el) |
| GR (1) | GR3026467T3 (el) |
| IE (1) | IE921650A1 (el) |
| NO (1) | NO302119B1 (el) |
| NZ (1) | NZ242951A (el) |
| ZA (1) | ZA924117B (el) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK40192D0 (da) * | 1992-03-26 | 1992-03-26 | Neurosearch As | Imidazolforbindelser, deres fremstilling og anvendelse |
| DK154092D0 (da) * | 1992-12-23 | 1992-12-23 | Neurosearch As | Imidazolforbindelser, deres fremstilling og anvendelse |
| AU675484B2 (en) * | 1993-03-24 | 1997-02-06 | Neurosearch A/S | Benzimidazole compounds, their use and preparation |
| US5554630A (en) * | 1993-03-24 | 1996-09-10 | Neurosearch A/S | Benzimidazole compounds |
| US5496826A (en) * | 1994-09-02 | 1996-03-05 | Bristol-Myers Squibb Company | Pharmaceutical methods of using heterocyclic derivatives of N-phenylamides |
| TR199701219T1 (xx) * | 1995-04-21 | 1998-03-21 | Neurosearch A/S | Benzimidazol bile�ikleri, bu bile�ikleri i�eren ispen�iyar� bile�ikler. |
| EP0997147B1 (en) * | 1997-07-08 | 2006-03-15 | Ono Pharmaceutical Co., Ltd. | Amino acid derivatives |
| CA2315910A1 (en) * | 1997-12-22 | 1999-07-01 | Ajinomoto Co., Inc. | Novel dihydropyridine derivative |
| TWI245035B (en) | 1998-06-26 | 2005-12-11 | Ono Pharmaceutical Co | Amino acid derivatives and a pharmaceutical composition comprising the derivatives |
| WO2000001676A1 (en) * | 1998-07-02 | 2000-01-13 | Neurosearch A/S | Potassium channel blocking agents |
| US6194447B1 (en) | 1998-07-02 | 2001-02-27 | Neurosearch A/S | Bis (benzimidazole) derivatives serving as potassium blocking agents |
| KR100633349B1 (ko) | 1998-07-14 | 2006-10-16 | 오노 야꾸힝 고교 가부시키가이샤 | 아미노산 유도체 및 이들을 유효 성분으로서 함유하는 약제 |
| US6316440B1 (en) | 1998-07-30 | 2001-11-13 | Warner-Lambert Company | Reduced dipeptide analogues as calcium channel antagonists |
| WO2000078719A1 (fr) | 1999-06-23 | 2000-12-28 | Ajinomoto Co., Inc. | Derive de la dihydropyridine |
| SK287527B6 (sk) * | 2000-01-14 | 2011-01-04 | Bayer Schering Pharma Aktiengesellschaft | 1,2-Diarylbenzimidazoly a ich farmaceutické použitie |
| US7115645B2 (en) | 2000-01-14 | 2006-10-03 | Schering Aktiengesellschaft | 1,2 diarylbenzimidazoles and their pharmaceutical use |
| US7329679B2 (en) | 2000-01-27 | 2008-02-12 | Schering Aktiengesellschaft | 1,2 Diarylbenzimidazoles and their pharmaceutical use |
| DE10135050A1 (de) * | 2001-07-09 | 2003-02-06 | Schering Ag | 1-Ary1-2-N-, S- oder O-substituierte Benzimidazolderivate, deren Verwendung zur Herstellung von Arzneimitteln sowie diese Derivate enthaltende pharmazeutische Präparate |
| KR100873400B1 (ko) * | 2002-10-17 | 2008-12-11 | 한국과학기술연구원 | Ｎ-타입 칼슘 채널의 활성을 억제함으로써 우울증을감소시키는 방법 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4492708A (en) * | 1982-09-27 | 1985-01-08 | Eli Lilly And Company | Antiviral benzimidazoles |
| JPH0772181B2 (ja) * | 1989-06-26 | 1995-08-02 | 株式会社大塚製薬工場 | ベンズイミダゾール誘導体 |
| NZ239540A (en) * | 1990-09-24 | 1993-11-25 | Neurosearch As | 1-phenyl benzimidazole derivatives and medicaments |
-
1992
- 1992-05-27 EP EP92108983A patent/EP0520200B1/en not_active Expired - Lifetime
- 1992-05-27 DK DK92108983T patent/DK0520200T3/da active
- 1992-05-27 AT AT92108983T patent/ATE163290T1/de active
- 1992-05-27 DE DE69224448T patent/DE69224448T2/de not_active Expired - Lifetime
- 1992-05-27 ES ES92108983T patent/ES2113898T3/es not_active Expired - Lifetime
- 1992-05-29 NZ NZ242951A patent/NZ242951A/en not_active IP Right Cessation
- 1992-05-29 AU AU17267/92A patent/AU653816B2/en not_active Ceased
- 1992-06-05 ZA ZA924117A patent/ZA924117B/xx unknown
- 1992-06-22 CA CA002071793A patent/CA2071793A1/en not_active Abandoned
- 1992-06-22 FI FI922905A patent/FI922905L/fi unknown
- 1992-06-23 JP JP4165075A patent/JPH05186432A/ja active Pending
- 1992-06-23 NO NO922475A patent/NO302119B1/no not_active IP Right Cessation
- 1992-07-01 IE IE165092A patent/IE921650A1/en unknown
-
1998
- 1998-03-27 GR GR980400651T patent/GR3026467T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0520200A2 (en) | 1992-12-30 |
| ZA924117B (en) | 1993-03-31 |
| NZ242951A (en) | 1994-12-22 |
| NO922475L (no) | 1992-12-28 |
| FI922905A0 (fi) | 1992-06-22 |
| FI922905L (fi) | 1992-12-25 |
| AU653816B2 (en) | 1994-10-13 |
| AU1726792A (en) | 1993-01-07 |
| CA2071793A1 (en) | 1992-12-25 |
| DE69224448T2 (de) | 1998-06-10 |
| ES2113898T3 (es) | 1998-05-16 |
| EP0520200B1 (en) | 1998-02-18 |
| DK0520200T3 (da) | 1998-09-23 |
| EP0520200A3 (en) | 1993-05-12 |
| DE69224448D1 (de) | 1998-03-26 |
| JPH05186432A (ja) | 1993-07-27 |
| GR3026467T3 (en) | 1998-06-30 |
| IE921650A1 (en) | 1992-12-30 |
| ATE163290T1 (de) | 1998-03-15 |
| NO922475D0 (no) | 1992-06-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |
Free format text: LAPSED IN DECEMBER 2000 |