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NO20072288L - Sulfonamid pert-substituerte bicykler for okklusly arteriesykdom - Google Patents

Sulfonamid pert-substituerte bicykler for okklusly arteriesykdom

Info

Publication number
NO20072288L
NO20072288L NO20072288A NO20072288A NO20072288L NO 20072288 L NO20072288 L NO 20072288L NO 20072288 A NO20072288 A NO 20072288A NO 20072288 A NO20072288 A NO 20072288A NO 20072288 L NO20072288 L NO 20072288L
Authority
NO
Norway
Prior art keywords
sulfonamide
occlusly
pert
artery disease
substituted
Prior art date
Application number
NO20072288A
Other languages
English (en)
Inventor
Jasbir Singh
Mark Gurney
Georgeta Hategan
Peng Yu
David Zembower
Nian Zhou
Original Assignee
Decode Chemistry Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Decode Chemistry Inc filed Critical Decode Chemistry Inc
Publication of NO20072288L publication Critical patent/NO20072288L/no

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
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    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
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Abstract

Det er beskrevet acylsulfonamid, peri-substituerte, fusjonerte bicykliske ring-forbindelser som er nyttige for behandling eller profylakse av en prostaglandinformidlet sykdom eller lidelse. Forbindelsene er av generell formel (I). Et representativt eksempel er formel (II):
NO20072288A 2004-10-12 2007-05-02 Sulfonamid pert-substituerte bicykler for okklusly arteriesykdom NO20072288L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61817204P 2004-10-12 2004-10-12
PCT/US2005/023009 WO2006044000A1 (en) 2004-10-12 2005-06-27 Sulfonamide pert-substituted bicyclics for occlusive artery disease

Publications (1)

Publication Number Publication Date
NO20072288L true NO20072288L (no) 2007-06-25

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Family Applications (1)

Application Number Title Priority Date Filing Date
NO20072288A NO20072288L (no) 2004-10-12 2007-05-02 Sulfonamid pert-substituerte bicykler for okklusly arteriesykdom

Country Status (16)

Country Link
US (2) US7598397B2 (no)
EP (1) EP1812388B1 (no)
JP (1) JP2008515971A (no)
KR (1) KR20070091607A (no)
CN (1) CN101142184A (no)
AT (1) ATE499344T1 (no)
AU (1) AU2005296305A1 (no)
BR (1) BRPI0516003A (no)
CA (1) CA2583667A1 (no)
DE (1) DE602005026553D1 (no)
IL (1) IL182488A0 (no)
MX (1) MX2007004525A (no)
NO (1) NO20072288L (no)
NZ (1) NZ554491A (no)
RU (1) RU2403240C2 (no)
WO (1) WO2006044000A1 (no)

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ATE499344T1 (de) * 2004-10-12 2011-03-15 Decode Genetics Ehf Peri-substituierte bicyclische sulfonamide gegen arterielle verschlusskrankheit
CA2583828A1 (en) * 2004-10-12 2006-04-27 Decode Genetics, Inc. Carboxylic acid peri-substituted bicyclics for occlusive artery disease
AU2006277231A1 (en) * 2005-08-10 2007-02-15 Takeda Pharmaceutical Company Limited Therapeutic agent for diabetes
US7579483B2 (en) * 2006-05-16 2009-08-25 Decode Genetics, Ehf. Process for preparing 7-(acryloyl)indoles
WO2007137040A2 (en) * 2006-05-16 2007-11-29 Decode Genetics Ehf 7-(acryloyl) indole compositions and methods for making and using same
CA2654811A1 (en) * 2006-06-12 2007-12-21 Merck Frosst Canada Ltd. Indoline amide derivatives as ep4 receptor ligands
WO2008127275A2 (en) * 2006-09-22 2008-10-23 Ptc Therapeutics, Inc. Pyrrolinone compounds as inhibitors of bacterial peptidyl trna hydrolase and uses thereof
JP5624762B2 (ja) 2007-03-30 2014-11-12 塩野義製薬株式会社 新規ピロリノン誘導体およびそれを含有する医薬組成物
EP2219648A4 (en) * 2007-11-09 2010-11-03 Cenomed Biosciences Llc TREATMENT OF POSTRAUMATIC STRESS WITH TETRAHYDROINDOLONE ARYLPIPERAZINE COMPOUNDS
US20090264443A1 (en) * 2008-04-18 2009-10-22 David Helton Treatment of organophosphate exposure with tetrahydroindolone arylpiperazine compounds
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IL182488A0 (en) 2007-09-20
US20090291948A1 (en) 2009-11-26
EP1812388A1 (en) 2007-08-01
RU2007115410A (ru) 2008-11-10
CA2583667A1 (en) 2006-04-27
NZ554491A (en) 2009-07-31
BRPI0516003A (pt) 2008-04-29
RU2403240C2 (ru) 2010-11-10
JP2008515971A (ja) 2008-05-15
EP1812388B1 (en) 2011-02-23
WO2006044000A1 (en) 2006-04-27
KR20070091607A (ko) 2007-09-11
CN101142184A (zh) 2008-03-12
US20060079520A1 (en) 2006-04-13
US7598397B2 (en) 2009-10-06
DE602005026553D1 (de) 2011-04-07
ATE499344T1 (de) 2011-03-15
AU2005296305A1 (en) 2006-04-27

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