MA28363A1 - Antagonistes des recepteurs muscariniques de l'acetylcholine - Google Patents
Antagonistes des recepteurs muscariniques de l'acetylcholineInfo
- Publication number
- MA28363A1 MA28363A1 MA29273A MA29273A MA28363A1 MA 28363 A1 MA28363 A1 MA 28363A1 MA 29273 A MA29273 A MA 29273A MA 29273 A MA29273 A MA 29273A MA 28363 A1 MA28363 A1 MA 28363A1
- Authority
- MA
- Morocco
- Prior art keywords
- antagonists
- acetylcholine receptors
- muscarinic acetylcholine
- muscarinic
- receptors
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US53609204P | 2004-01-13 | 2004-01-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
MA28363A1 true MA28363A1 (fr) | 2006-12-01 |
Family
ID=34794385
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA29273A MA28363A1 (fr) | 2004-01-13 | 2006-08-15 | Antagonistes des recepteurs muscariniques de l'acetylcholine |
Country Status (16)
Country | Link |
---|---|
US (1) | US20080249127A1 (fr) |
EP (1) | EP1711183A4 (fr) |
JP (1) | JP2007518740A (fr) |
KR (1) | KR20060129017A (fr) |
CN (1) | CN1929844A (fr) |
AR (1) | AR049464A1 (fr) |
AU (1) | AU2005204935A1 (fr) |
BR (1) | BRPI0506777A (fr) |
CA (1) | CA2552880A1 (fr) |
IL (1) | IL176775A0 (fr) |
MA (1) | MA28363A1 (fr) |
NO (1) | NO20063636L (fr) |
PE (1) | PE20050898A1 (fr) |
RU (1) | RU2006129289A (fr) |
TW (1) | TW200534855A (fr) |
WO (1) | WO2005067537A2 (fr) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2007528420A (ja) * | 2004-03-11 | 2007-10-11 | グラクソ グループ リミテッド | 新規m3ムスカリン性アセチルコリン受容体アンタゴニスト |
TWI363759B (en) | 2004-04-27 | 2012-05-11 | Glaxo Group Ltd | Muscarinic acetylcholine receptor antagonists |
EP1747219A4 (fr) * | 2004-05-13 | 2010-05-26 | Glaxo Group Ltd | Domaine de l'invention antagonistes récepteurs d'acétyle choline muscarinique |
JP2008505118A (ja) * | 2004-06-30 | 2008-02-21 | グラクソ グループ リミテッド | ムスカリン性アセチルコリン受容体アンタゴニスト |
US7932247B2 (en) * | 2004-11-15 | 2011-04-26 | Glaxo Group Limited | M3 muscarinic acetylcholine receptor antagonists |
EP1856049A1 (fr) | 2005-03-10 | 2007-11-21 | Theravance, Inc. | Composes biphenyles utiles en tant qu'antagonistes des recepteurs muscariniques |
EP1904446A2 (fr) * | 2005-07-11 | 2008-04-02 | Ranbaxy Laboratories Limited | Antagonistes des recepteurs muscariniques |
UY31637A1 (es) | 2008-02-06 | 2009-08-03 | Farmacoforos duales-antagonistas muscarinicos de pde4 | |
PE20091563A1 (es) | 2008-02-06 | 2009-11-05 | Glaxo Group Ltd | Farmacoforos duales - antagonistas muscarinicos de pde4 |
CL2009000248A1 (es) | 2008-02-06 | 2009-09-11 | Glaxo Group Ltd | Compuestos derivados de pirazolo [3,4-b] piridin-5-il, inhibidores de la fosfodiesterasa de tipo iv (pde4) y antagonista de receptores muscarinicos de acetilcolina (machr); composicion farmaceutica que los comprende; y su uso en la preparacion de medicamentos utiles en el tratamiento de enferemedades respiratorias y alergicas |
WO2010094643A1 (fr) | 2009-02-17 | 2010-08-26 | Glaxo Group Limited | Dérivés de quinoline et applications associées dans la rhinite et l'urticaire |
BRPI1014390A2 (pt) | 2009-04-30 | 2016-04-05 | Teijin Pharma Ltd | composto de sal de amônio quaternário, composição medicinal, e, agente preventivo ou terapêutico |
WO2014023325A1 (fr) * | 2012-08-06 | 2014-02-13 | Fondazione Istituto Italiano Di Tecnologia | Inhibiteurs de faah et de cox multicibles et leurs utilisations thérapeutiques |
KR101538846B1 (ko) * | 2013-07-30 | 2015-07-22 | 동아에스티 주식회사 | 신규한 바이페닐 유도체 및 그의 제조방법 |
KR102239776B1 (ko) * | 2016-08-26 | 2021-04-13 | 동아에스티 주식회사 | (r)-(1-메틸피롤리딘-3-일)메틸(3'-클로로-4'-플루오로-[1,1'-비페닐]-2-일)카바메이트의 신규염 및 이의 결정형 |
PH12019500380B1 (en) * | 2016-08-26 | 2024-04-17 | Dong A St Co Ltd | Novel salt of (r)-(1-methylpyrrolidine-3-yl)methyl(3`-chloro-4`fluoro-[1,1`-biphenyl]-2-yl)carbamate and a crystal form thereof |
EP3710483A4 (fr) | 2017-11-16 | 2021-10-20 | XL-protein GmbH | Protéines de fusion vegfr/pdgfr pasylées et leur utilisation en thérapie |
JP2021505569A (ja) * | 2017-12-04 | 2021-02-18 | フリードリヒ−アレクサンダー−ウニヴェルシテート エアランゲン−ニュルンベルク | M2よりもm3に対して選択性を有するフルオロフェニル置換ムスカリン受容体リガンド |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1140998B (it) * | 1980-06-18 | 1986-10-10 | Valeas Ind Chimica E Farmaceut | Sali di endo-8-metil-8-sin-alchil-8-azoniabiciclo aperta par. quadrata 3.2.1. chiusa par. quadrata-ottan-3-alchilcarbossilati, processo per la loro preparazione e composizioni terapeutiche che li contengono come principio attivo |
WO1995021820A1 (fr) * | 1994-02-10 | 1995-08-17 | Yamanouchi Pharmaceutical Co., Ltd. | Nouveau derive du carbamate et composition correspondante |
AU2001271027B2 (en) * | 2000-07-11 | 2005-07-07 | Msd K.K. | Ester derivatives |
US7365167B2 (en) * | 2001-11-26 | 2008-04-29 | Cell Matrix, Inc. | Humanized collagen antibodies and related methods |
WO2003094831A2 (fr) * | 2002-05-07 | 2003-11-20 | Neurosearch A/S | Nouveaux derives de biaryle diazabicyclique |
US7041674B2 (en) * | 2002-11-26 | 2006-05-09 | Boehringer Ingelhiem Pharma Gmbh & Co. Kg | Carbamic acid esters with anticholinergic activity |
DE10255040A1 (de) * | 2002-11-26 | 2004-06-03 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Carbaminsäureester mit anticholinerger Wirksamkeit |
EP1613307A4 (fr) * | 2003-04-07 | 2008-03-12 | Glaxo Group Ltd | Antagonistes du recepteur muscarinique m sb 3 /sb de l'acetylcholine |
-
2005
- 2005-01-11 TW TW094100746A patent/TW200534855A/zh unknown
- 2005-01-13 AU AU2005204935A patent/AU2005204935A1/en not_active Abandoned
- 2005-01-13 EP EP05711495A patent/EP1711183A4/fr not_active Withdrawn
- 2005-01-13 AR ARP050100118A patent/AR049464A1/es not_active Application Discontinuation
- 2005-01-13 CA CA002552880A patent/CA2552880A1/fr not_active Abandoned
- 2005-01-13 PE PE2005000059A patent/PE20050898A1/es not_active Application Discontinuation
- 2005-01-13 WO PCT/US2005/001333 patent/WO2005067537A2/fr active Application Filing
- 2005-01-13 US US10/585,830 patent/US20080249127A1/en not_active Abandoned
- 2005-01-13 RU RU2006129289/04A patent/RU2006129289A/ru not_active Application Discontinuation
- 2005-01-13 BR BRPI0506777-4A patent/BRPI0506777A/pt not_active Application Discontinuation
- 2005-01-13 JP JP2006549649A patent/JP2007518740A/ja active Pending
- 2005-01-13 KR KR1020067016188A patent/KR20060129017A/ko not_active Application Discontinuation
- 2005-01-13 CN CNA2005800081262A patent/CN1929844A/zh active Pending
-
2006
- 2006-07-10 IL IL176775A patent/IL176775A0/en unknown
- 2006-08-11 NO NO20063636A patent/NO20063636L/no not_active Application Discontinuation
- 2006-08-15 MA MA29273A patent/MA28363A1/fr unknown
Also Published As
Publication number | Publication date |
---|---|
PE20050898A1 (es) | 2005-11-06 |
KR20060129017A (ko) | 2006-12-14 |
RU2006129289A (ru) | 2008-02-20 |
WO2005067537A3 (fr) | 2006-05-18 |
JP2007518740A (ja) | 2007-07-12 |
TW200534855A (en) | 2005-11-01 |
CA2552880A1 (fr) | 2005-07-28 |
EP1711183A2 (fr) | 2006-10-18 |
CN1929844A (zh) | 2007-03-14 |
AU2005204935A1 (en) | 2005-07-28 |
NO20063636L (no) | 2006-10-04 |
BRPI0506777A (pt) | 2007-05-22 |
IL176775A0 (en) | 2006-10-31 |
AR049464A1 (es) | 2006-08-09 |
EP1711183A4 (fr) | 2009-04-01 |
WO2005067537A2 (fr) | 2005-07-28 |
US20080249127A1 (en) | 2008-10-09 |
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