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MA28048A1 - Amino-acides a affinite pour la proteine alpha-2-delta - Google Patents

Amino-acides a affinite pour la proteine alpha-2-delta

Info

Publication number
MA28048A1
MA28048A1 MA28887A MA28887A MA28048A1 MA 28048 A1 MA28048 A1 MA 28048A1 MA 28887 A MA28887 A MA 28887A MA 28887 A MA28887 A MA 28887A MA 28048 A1 MA28048 A1 MA 28048A1
Authority
MA
Morocco
Prior art keywords
affinity
alpha
amino acids
delta
delta protein
Prior art date
Application number
MA28887A
Other languages
English (en)
Inventor
Christopher James Deur
Christine Nylund Kolz
Augustine Tobi Osuma
Mark Stephen Plummer
Jacob Bradley Schwarz
Andrew John Thorpe
David Juergen Wustrow
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34396281&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA28048(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of MA28048A1 publication Critical patent/MA28048A1/fr

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    • C—CHEMISTRY; METALLURGY
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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
    • C07C229/08—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to hydrogen atoms
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • C07C229/20—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
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    • C07D263/18—Oxygen atoms
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Abstract

DEPOSANT Société dite : WARNER-LAMBERT COMPANY LLC REVENDICATION DE PRIORITES US 25 Septembre 2003 60/505,953 US 30 Septembre 2003 60/507,443 Voir en annexe le titre de l'invention et le texte de l'abrégé Amino-acides à affinité pour la protéine alpha-2-delta Certains (beta)-amino-acides qui se lient à la sous-unité alpha-2-delta (a2S) d'un canal calcium sont décrits. Ces composés et leurs sels pharmaceutiquement acceptables sont utiles dans le traitement de divers troubles psychiatriques, de la douleur et d'autres troubles.
MA28887A 2003-09-25 2006-03-24 Amino-acides a affinite pour la proteine alpha-2-delta MA28048A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50595303P 2003-09-25 2003-09-25
US50744303P 2003-09-30 2003-09-30

Publications (1)

Publication Number Publication Date
MA28048A1 true MA28048A1 (fr) 2006-07-03

Family

ID=34396281

Family Applications (1)

Application Number Title Priority Date Filing Date
MA28887A MA28048A1 (fr) 2003-09-25 2006-03-24 Amino-acides a affinite pour la proteine alpha-2-delta

Country Status (27)

Country Link
US (3) US20050124668A1 (fr)
EP (1) EP1667957A2 (fr)
JP (2) JP4001349B2 (fr)
KR (2) KR20070039986A (fr)
AP (1) AP2006003544A0 (fr)
AR (1) AR046022A1 (fr)
AU (1) AU2004276072A1 (fr)
BR (1) BRPI0414781A (fr)
CA (1) CA2540208A1 (fr)
CO (1) CO5680413A2 (fr)
CR (1) CR8290A (fr)
EA (1) EA200600467A1 (fr)
EC (1) ECSP066450A (fr)
IL (1) IL173764A0 (fr)
IS (1) IS8308A (fr)
MA (1) MA28048A1 (fr)
MX (1) MXPA06003395A (fr)
NL (2) NL1027115C2 (fr)
NO (1) NO20061812L (fr)
OA (1) OA13258A (fr)
PA (1) PA8613101A1 (fr)
PE (1) PE20050434A1 (fr)
RS (1) RS20060210A (fr)
TN (1) TNSN06095A1 (fr)
TW (1) TW200528420A (fr)
UY (1) UY28533A1 (fr)
WO (1) WO2005030700A2 (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090247743A1 (en) * 2004-07-09 2009-10-01 Pfizer Inc Preparation of beta-amino acids having affinity for the alpha-2-delta protein
KR20070107147A (ko) * 2005-03-24 2007-11-06 파마시아 앤드 업존 캄파니 엘엘씨 알파-2-델타 단백질에 친화성을 갖는 광학적으로 순수한베타-아미노산의 제조
JP2009516675A (ja) * 2005-11-17 2009-04-23 ファイザー・リミテッド 疼痛を治療するためのイソシステイン誘導体
EP1993529A1 (fr) * 2006-03-06 2008-11-26 Pfizer Products Inc. Ligands alpha-2-delta pour sommeil non réparateur
AR061728A1 (es) * 2006-06-30 2008-09-17 Pfizer Prod Inc Composicion para tratamiento usando compuestos selectivos alfa-2-delta-1
EP1903027A1 (fr) * 2006-09-13 2008-03-26 Novartis AG Procédé de préparation de l' acide amino-4 butyrique ou de ses derivés et leur utilisation pour la préparation des inhibiteurs NEP
US20110124705A1 (en) * 2009-11-24 2011-05-26 Xenoport, Inc. Prodrugs of alpha-2-delta ligands, pharmaceutical compositions and uses thereof
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