LTIP1718A - New heterocyclic compounds as antagonists of exitatory amino acids receptors, process for their preparation and their use - Google Patents

New heterocyclic compounds as antagonists of exitatory amino acids receptors, process for their preparation and their use

Info

Publication number: LTIP1718A
Authority: LT; Lithuania
Prior art keywords: antagonists; preparation; amino acids; heterocyclic compounds; new heterocyclic
Prior art date: 1990-11-15

Application number

LTIP1718A

Inventor

Britt-Marie Eva Swahn

Alf Erling Albert Claesson

Original Assignee

Astra Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-11-15

Filing date

1993-12-30

Publication date

1995-07-25

1993-12-30 Application filed by Astra Ab filed Critical Astra Ab

1995-07-25 Publication of LTIP1718A publication Critical patent/LTIP1718A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
- C07F9/6509—Six-membered rings
- C07F9/650952—Six-membered rings having the nitrogen atoms in the positions 1 and 4
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/59—Hydrogenated pyridine rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pain & Pain Management (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

LTIP1718A 1990-11-15 1993-12-30 New heterocyclic compounds as antagonists of exitatory amino acids receptors, process for their preparation and their use LTIP1718A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
SE9003652A SE9003652D0 (en)	1990-11-15	1990-11-15	NEW HETEROCYCLIC COMPOUNDS

Publications (1)

Publication Number	Publication Date
LTIP1718A true LTIP1718A (en)	1995-07-25

Family

ID=20380925

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
LTIP1718A LTIP1718A (en)	1990-11-15	1993-12-30	New heterocyclic compounds as antagonists of exitatory amino acids receptors, process for their preparation and their use

Country Status (17)

Country	Link
EP (1)	EP0557375A1 (en)
JP (1)	JPH06502421A (en)
CN (1)	CN1061595A (en)
AU (1)	AU652399B2 (en)
CA (1)	CA2095224A1 (en)
CZ (1)	CZ80993A3 (en)
FI (1)	FI932206L (en)
HU (1)	HU9301417D0 (en)
IE (1)	IE913922A1 (en)
IS (1)	IS3782A7 (en)
LT (1)	LTIP1718A (en)
MX (1)	MX9101979A (en)
NO (1)	NO931679D0 (en)
PT (1)	PT99515A (en)
SE (1)	SE9003652D0 (en)
SK (1)	SK46993A3 (en)
WO (1)	WO1992008724A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5194430A (en) *	1990-05-17	1993-03-16	Merrell Dow Pharmaceuticals Inc.	Heterocyclic-nmda antagonists
TW281670B (en) *	1993-09-02	1996-07-21	Hoffmann La Roche
US5491241A (en) *	1993-10-18	1996-02-13	Eli Lilly And Company	Bicyclic intermediates for excitatory amino acid receptor antagonists
RS65984B1 (en)	2016-02-04	2024-10-31	Takeda Pharmaceuticals Co	Substituted piperidine compound as orexin type 2 agonist for the treatment of narcolepsy

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1248531A (en) *	1984-04-17	1989-01-10	Jeffrey C. Watkins	4-substituted piperazine-2-carboxylic acids
JPS612519A (en) *	1984-04-24	1986-01-08	Aron Kasei Co Ltd	Method of injection molding
US4906621A (en) *	1985-05-24	1990-03-06	Ciba-Geigy Corporation	Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade
US4740346A (en) *	1986-02-26	1988-04-26	The Budd Company	Perimeter resin feeding of composite structures
JPS63112129A (en) *	1986-10-30	1988-05-17	Toyoda Gosei Co Ltd	Multi-color resin molding die
EP0275820B1 (en) *	1986-11-21	1991-02-06	Ciba-Geigy Ag	Unsaturated phosphonic acids and derivatives

1990
- 1990-11-15 SE SE9003652A patent/SE9003652D0/en unknown
1991
- 1991-11-05 CN CN91110925A patent/CN1061595A/en active Pending
- 1991-11-07 WO PCT/SE1991/000753 patent/WO1992008724A1/en not_active Application Discontinuation
- 1991-11-07 CZ CS93809A patent/CZ80993A3/en unknown
- 1991-11-07 CA CA002095224A patent/CA2095224A1/en not_active Abandoned
- 1991-11-07 AU AU89391/91A patent/AU652399B2/en not_active Ceased
- 1991-11-07 JP JP4500566A patent/JPH06502421A/en active Pending
- 1991-11-07 HU HU931417A patent/HU9301417D0/en unknown
- 1991-11-07 SK SK46993A patent/SK46993A3/en unknown
- 1991-11-07 EP EP91920264A patent/EP0557375A1/en not_active Withdrawn
- 1991-11-08 MX MX9101979A patent/MX9101979A/en unknown
- 1991-11-12 IE IE392291A patent/IE913922A1/en unknown
- 1991-11-14 IS IS3782A patent/IS3782A7/en unknown
- 1991-11-14 PT PT99515A patent/PT99515A/en not_active Application Discontinuation
1993
- 1993-05-07 NO NO931679A patent/NO931679D0/en unknown
- 1993-05-14 FI FI932206A patent/FI932206L/en not_active Application Discontinuation
- 1993-12-30 LT LTIP1718A patent/LTIP1718A/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
MX9101979A (en)	1992-07-08
AU8939191A (en)	1992-06-11
JPH06502421A (en)	1994-03-17
SE9003652D0 (en)	1990-11-15
AU652399B2 (en)	1994-08-25
NO931679L (en)	1993-05-07
FI932206A0 (en)	1993-05-14
WO1992008724A1 (en)	1992-05-29
IE913922A1 (en)	1992-05-20
SK46993A3 (en)	1993-10-06
HU9301417D0 (en)	1993-09-28
EP0557375A1 (en)	1993-09-01
CZ80993A3 (en)	1994-02-16
CA2095224A1 (en)	1992-05-16
NO931679D0 (en)	1993-05-07
FI932206L (en)	1993-05-14
IS3782A7 (en)	1992-05-16
PT99515A (en)	1992-09-30
CN1061595A (en)	1992-06-03

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Legal Events

Date	Code	Title	Description
1996-02-26	FD9A	Withdrawn applications	Free format text: 951228