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LT3386997T - Monomaleimidu funkcionalizuoti platinos junginiai, skirti vėžio terapijai - Google Patents

Monomaleimidu funkcionalizuoti platinos junginiai, skirti vėžio terapijai

Info

Publication number
LT3386997T
LT3386997T LTEPPCT/EP2016/080453T LT16080453T LT3386997T LT 3386997 T LT3386997 T LT 3386997T LT 16080453 T LT16080453 T LT 16080453T LT 3386997 T LT3386997 T LT 3386997T
Authority
LT
Lithuania
Prior art keywords
monomaleimide
functioned
cancer therapy
platinum compounds
platinum
Prior art date
Application number
LTEPPCT/EP2016/080453T
Other languages
English (en)
Inventor
Christian KOWOL
Petra Heffeter
Walter Berger
Bernhard K. Keppler
Josef Mayr
Verena PICHLER
Original Assignee
Medizinische Universität Wien
Universität Wien
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medizinische Universität Wien, Universität Wien filed Critical Medizinische Universität Wien
Publication of LT3386997T publication Critical patent/LT3386997T/lt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/0006Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
    • C07F15/0086Platinum compounds
    • C07F15/0093Platinum compounds without a metal-carbon linkage
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/555Heterocyclic compounds containing heavy metals, e.g. hemin, hematin, melarsoprol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
LTEPPCT/EP2016/080453T 2015-12-09 2016-12-09 Monomaleimidu funkcionalizuoti platinos junginiai, skirti vėžio terapijai LT3386997T (lt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP15198739 2015-12-09
PCT/EP2016/080453 WO2017097986A1 (en) 2015-12-09 2016-12-09 Monomaleimide-functionalized platinum compounds for cancer therapy

Publications (1)

Publication Number Publication Date
LT3386997T true LT3386997T (lt) 2021-12-10

Family

ID=54849106

Family Applications (1)

Application Number Title Priority Date Filing Date
LTEPPCT/EP2016/080453T LT3386997T (lt) 2015-12-09 2016-12-09 Monomaleimidu funkcionalizuoti platinos junginiai, skirti vėžio terapijai

Country Status (21)

Country Link
US (2) US10723748B2 (lt)
EP (1) EP3386997B1 (lt)
JP (1) JP6867652B2 (lt)
CN (1) CN108368143B (lt)
AU (1) AU2016367306B2 (lt)
CA (1) CA3004630A1 (lt)
CY (1) CY1124529T1 (lt)
DK (1) DK3386997T3 (lt)
ES (1) ES2898704T3 (lt)
HR (1) HRP20211466T1 (lt)
HU (1) HUE056897T2 (lt)
IL (1) IL259864B (lt)
LT (1) LT3386997T (lt)
MX (1) MX2018006953A (lt)
PL (1) PL3386997T3 (lt)
PT (1) PT3386997T (lt)
RS (1) RS62412B1 (lt)
SG (1) SG11201804885TA (lt)
SI (1) SI3386997T1 (lt)
SM (1) SMT202100709T1 (lt)
WO (1) WO2017097986A1 (lt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101915452B1 (ko) * 2014-06-23 2018-11-06 플라콘 테라퓨틱스 인코포레이티드 백금 화합물, 조성물 및 이의 용도
TWI808055B (zh) 2016-05-11 2023-07-11 美商滬亞生物國際有限公司 Hdac 抑制劑與 pd-1 抑制劑之組合治療
TWI794171B (zh) 2016-05-11 2023-03-01 美商滬亞生物國際有限公司 Hdac抑制劑與pd-l1抑制劑之組合治療
CN109171001A (zh) * 2018-09-14 2019-01-11 上海烟草集团有限责任公司 草酸钠在降低卷烟烟气中TSNAs释放量中的应用
US20230339997A1 (en) * 2020-09-11 2023-10-26 Shanghai Haiju Biological Technology Co., Ltd. Class of platinum compounds for treating cancer, and method for preparation thereof
CN114163479A (zh) * 2020-09-11 2022-03-11 上海海聚生物科技有限公司 一类治疗癌症用的铂类化合物及其制备方法
CN114539320A (zh) * 2020-11-25 2022-05-27 北京大学 辐射激活的四价铂配合物及其用途

Family Cites Families (44)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3773919A (en) 1969-10-23 1973-11-20 Du Pont Polylactide-drug mixtures
CH588505A5 (lt) 1972-06-08 1977-06-15 Research Corp
US4263428A (en) 1978-03-24 1981-04-21 The Regents Of The University Of California Bis-anthracycline nucleic acid function inhibitors and improved method for administering the same
ATE12348T1 (de) 1980-11-10 1985-04-15 Gersonde Klaus Prof Dr Verfahren zur herstellung von lipid-vesikeln durch ultraschallbehandlung, anwendung des verfahrens und vorrichtung zur durchfuehrung des verfahrens.
US4485045A (en) 1981-07-06 1984-11-27 Research Corporation Synthetic phosphatidyl cholines useful in forming liposomes
EP0088046B1 (de) 1982-02-17 1987-12-09 Ciba-Geigy Ag Lipide in wässriger Phase
DE3218121A1 (de) 1982-05-14 1983-11-17 Leskovar, Peter, Dr.-Ing., 8000 München Arzneimittel zur tumorbehandlung
EP0102324A3 (de) 1982-07-29 1984-11-07 Ciba-Geigy Ag Lipide und Tenside in wässriger Phase
US4544545A (en) 1983-06-20 1985-10-01 Trustees University Of Massachusetts Liposomes containing modified cholesterol for organ targeting
JPS607934A (ja) 1983-06-29 1985-01-16 Dai Ichi Seiyaku Co Ltd リポソ−ムの製造方法
HUT35524A (en) 1983-08-02 1985-07-29 Hoechst Ag Process for preparing pharmaceutical compositions containing regulatory /regulative/ peptides providing for the retarded release of the active substance
ATE159858T1 (de) 1983-09-26 1997-11-15 Ehrenfeld Udo Mittel und erzeugnis für die diagnose und therapie von tumoren sowie zur behandlung von schwächen der zelligen und humoralen immunabwehr
US4615885A (en) 1983-11-01 1986-10-07 Terumo Kabushiki Kaisha Pharmaceutical composition containing urokinase
CS269719B1 (en) 1986-12-29 1990-05-14 Kiss Frantisek Platinum cytostatic
US6051256A (en) 1994-03-07 2000-04-18 Inhale Therapeutic Systems Dispersible macromolecule compositions and methods for their preparation and use
DE19636889A1 (de) 1996-09-11 1998-03-12 Felix Dr Kratz Antineoplastisch wirkende Transferrin- und Albuminkonjugate zytostatischer Verbindungen aus der Gruppe der Anthrazykline, Alkylantien, Antimetabolite und Cisplatin-Analoga und diese enthaltende Arzneimittel
WO1999016422A1 (en) 1997-09-29 1999-04-08 Inhale Therapeutic Systems, Inc. Stabilized preparations for use in metered dose inhalers
AU761587B2 (en) 1998-04-21 2003-06-05 Amgen Research (Munich) Gmbh CD19xCD3 specific polypeptides and uses thereof
DE19926154A1 (de) 1999-06-09 2000-12-14 Ktb Tumorforschungs Gmbh Verfahren zur Herstellung einer injizierbaren Arzneimittelzubereitung
AUPQ641100A0 (en) 2000-03-23 2000-04-15 Australia Nuclear Science & Technology Organisation Methods of synthesis and use of radiolabelled platinum chemotherapeutic ag ents
PT1280520E (pt) 2000-05-10 2014-12-16 Novartis Ag Pós à base de fosfolípidos para administração de fármacos
TWI324518B (en) 2001-12-19 2010-05-11 Nektar Therapeutics Pulmonary delivery of aminoglycosides
DE10314780A1 (de) 2003-03-19 2004-09-30 Ktb Tumorforschungsgesellschaft Mbh Proteinbindende Derivate von Platinkomplexen mit Cyclobutan-1,1-dicarboxylatliganden
RU2343913C2 (ru) 2003-03-31 2009-01-20 Плива-Лахема А.С. Фармацевтическая композиция, содержащая комплекс платины в качестве активного вещества, и способ ее получения
CZ296169B6 (cs) 2004-09-08 2006-01-11 Pliva - Lachema A. S. Farmaceutická kompozice pro rektální nebo vaginální podání, zpusob její prípravy a tato kompozice pro pouzití jako lécivo
CZ296459B6 (cs) 2004-09-14 2006-03-15 Pliva-Lachema A. S. Perorální farmaceutická kompozice pro cílený transport komplexu platiny do kolorektální oblasti, zpusob její prípravy a tato kompozice pro pouzití jako lécivo
US20060205810A1 (en) 2004-11-24 2006-09-14 Schering Corporation Platinum therapeutic combinations
CZ300120B6 (cs) 2006-06-20 2009-02-11 Pliva - Lachema A. S. Farmaceutická kompozice pro injekcní podání
CZ300590B6 (cs) 2006-06-20 2009-06-24 Pliva - Lachema A. S. Farmaceutická kompozice pro injekcní podání
CZ300424B6 (cs) 2006-06-20 2009-05-13 Pliva - Lachema A. S. Farmaceutická kompozice pro perorální podání
EP2793585A4 (en) 2011-12-05 2015-12-09 Igenica Biotherapeutics Inc Antibody-Agent Conjugates and Related Compounds, Compositions and Methods
MX366864B (es) * 2012-02-27 2019-07-26 Amunix Operating Inc Composiciones de conjugados de xten y métodos para realizarlas.
EA201690434A1 (ru) * 2013-10-08 2016-08-31 Этлас Дженетикс Лимитед Маркирующие соединения и их применение в анализах
EP3089745A4 (en) 2013-12-31 2017-05-17 Placon Therapeutics, Inc. Compounds, compositions, and methods for the treatment of cancers
KR101915452B1 (ko) * 2014-06-23 2018-11-06 플라콘 테라퓨틱스 인코포레이티드 백금 화합물, 조성물 및 이의 용도
WO2016209935A1 (en) 2015-06-23 2016-12-29 Placon Therapeutics, Inc. Platinum compounds, compositions, and uses thereof
US10342801B2 (en) 2015-06-23 2019-07-09 Placon Therapeutics, Inc. Platinum compounds, compositions, and uses thereof
EP3313527B1 (en) 2015-06-29 2021-02-24 Case Western Reserve University Anticancer drug-containing plant virus particles
JP6759326B2 (ja) 2015-07-12 2020-09-23 ハンジョウ ディーエーシー バイオテック シーオー.,エルティディ.Hangzhou Dac Biotech Co.,Ltd. 細胞結合分子の共役のための架橋連結体
JP7043425B2 (ja) 2016-06-06 2022-03-29 ジェネンテック, インコーポレイテッド シルベストロール抗体-薬物コンジュゲート及び使用方法
CN109690315A (zh) 2016-07-08 2019-04-26 豪夫迈·罗氏有限公司 人附睾蛋白4(he4)用于评估muc16阳性癌症治疗的响应性的用途
WO2018026742A1 (en) 2016-08-01 2018-02-08 Askgene Pharma Inc. Novel antibody-albumin-drug conjugates (aadc) and methods for using them
CN108164512B (zh) 2017-12-27 2021-05-25 沈阳药科大学 一类具有生物粘附作用的马来酰亚胺型前药及其在口服药物传递中的应用
CN108187063B (zh) 2018-01-09 2020-09-08 沈阳药科大学 白蛋白结合型抗肿瘤药-马来酰亚胺分子前药

Also Published As

Publication number Publication date
HUE056897T2 (hu) 2022-03-28
CN108368143B (zh) 2022-02-01
HRP20211466T1 (hr) 2021-12-24
IL259864A (en) 2018-07-31
JP6867652B2 (ja) 2021-05-12
SMT202100709T1 (it) 2022-01-10
PL3386997T3 (pl) 2021-12-13
CA3004630A1 (en) 2017-06-15
MX2018006953A (es) 2019-05-16
CN108368143A (zh) 2018-08-03
SG11201804885TA (en) 2018-07-30
EP3386997A1 (en) 2018-10-17
US20210002313A1 (en) 2021-01-07
JP2018538292A (ja) 2018-12-27
US20180354979A1 (en) 2018-12-13
US10723748B2 (en) 2020-07-28
ES2898704T3 (es) 2022-03-08
PT3386997T (pt) 2021-11-04
US11572379B2 (en) 2023-02-07
CY1124529T1 (el) 2022-07-22
IL259864B (en) 2022-07-01
AU2016367306B2 (en) 2021-04-22
AU2016367306A1 (en) 2018-06-14
RS62412B1 (sr) 2021-10-29
WO2017097986A1 (en) 2017-06-15
EP3386997B1 (en) 2021-06-30
DK3386997T3 (da) 2021-09-20
SI3386997T1 (sl) 2021-11-30

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