KR20050088291A - 아데노신 ａ３ 수용체 리간드로서의 이미다조퀴놀린 유도체 - Google Patents

아데노신 ａ３ 수용체 리간드로서의 이미다조퀴놀린 유도체 Download PDF

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Publication number: KR20050088291A
Authority: KR; South Korea
Prior art keywords: group; formula; branched; straight; salts
Prior art date: 2002-11-15
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

KR1020057008683A

Other languages

English (en)

Korean (ko)

Inventor

페터 아라니

라슬로 발라주

마리아 발로그

산도르 바토리

나기 러이오시 티.

게자 티마리

킨가 보에르

졸탄 카푸이

엔드레 미쿠스

카탈린 게르베르

세레디 유디트 바르가네

카탈린 우르반-사보

에르즈세베트 왈츠

Original Assignee

사노피-아벤티스

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-11-15

Filing date

2003-11-11

Publication date

2005-09-05

2003-11-11 Application filed by 사노피-아벤티스 filed Critical 사노피-아벤티스

2005-09-05 Publication of KR20050088291A publication Critical patent/KR20050088291A/ko

Status Abandoned legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
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- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Psychiatry (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Immunology (AREA)
Dermatology (AREA)
Rheumatology (AREA)
Ophthalmology & Optometry (AREA)
Pain & Pain Management (AREA)
Epidemiology (AREA)
Psychology (AREA)
Hematology (AREA)
Obesity (AREA)
Emergency Medicine (AREA)
Physical Education & Sports Medicine (AREA)
Endocrinology (AREA)
Orthopedic Medicine & Surgery (AREA)
Vascular Medicine (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)

KR1020057008683A 2002-11-15 2003-11-11 아데노신 ａ３ 수용체 리간드로서의 이미다조퀴놀린 유도체 Abandoned KR20050088291A (ko)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
HUP0203976		2002-11-15
HU0203976A HUP0203976A3 (en)	2002-11-15	2002-11-15	Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them

Publications (1)

Publication Number	Publication Date
KR20050088291A true KR20050088291A (ko)	2005-09-05

Family

ID=90001561

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
KR1020057008683A Abandoned KR20050088291A (ko)	2002-11-15	2003-11-11	아데노신 ａ３ 수용체 리간드로서의 이미다조퀴놀린 유도체

Country Status (35)

Country	Link
US (2)	US7419977B2 (is)
EP (1)	EP1560828B9 (is)
JP (1)	JP4533148B2 (is)
KR (1)	KR20050088291A (is)
CN (1)	CN1332960C (is)
AR (1)	AR041968A1 (is)
AT (1)	ATE325123T1 (is)
AU (1)	AU2003282263B2 (is)
BR (1)	BR0316355A (is)
CA (1)	CA2505910C (is)
CO (1)	CO5690577A2 (is)
CY (1)	CY1105180T1 (is)
DE (1)	DE60305058T2 (is)
DK (1)	DK1560828T3 (is)
EA (1)	EA007595B1 (is)
ES (1)	ES2263039T3 (is)
HK (1)	HK1077819A1 (is)
HR (1)	HRP20050540A2 (is)
HU (1)	HUP0203976A3 (is)
IL (1)	IL168516A (is)
IS (1)	IS2456B (is)
MA (1)	MA27501A1 (is)
ME (1)	MEP19008A (is)
MX (1)	MXPA05005198A (is)
NO (1)	NO20052866D0 (is)
NZ (1)	NZ540029A (is)
PL (1)	PL376837A1 (is)
PT (1)	PT1560828E (is)
RS (1)	RS51320B (is)
SI (1)	SI1560828T1 (is)
TN (1)	TNSN05133A1 (is)
TW (1)	TWI248934B (is)
UA (1)	UA78889C2 (is)
WO (1)	WO2004046146A1 (is)
ZA (1)	ZA200503807B (is)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HUP0105406A3 (en) *	2001-12-21	2003-12-29	Sanofi Aventis	Imidazo[1,2-a]quinolin derivatives, process for their preparation, pharmaceutical compositions thereof and intermediates
HUP0203976A3 (en) *	2002-11-15	2004-08-30	Sanofi Aventis	Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them
HUP0400812A2 (en) *	2004-04-19	2006-02-28	Sanofi Aventis	Crystalline forms of 2-amino-3-cyano-quinoline derivatives, process for their preparation and pharmaceutical compositions containing them
GT200600381A (es)	2005-08-25	2007-03-28		Compuestos organicos
US20090088403A1 (en) *	2007-05-07	2009-04-02	Randy Blakely	A3 adenosine receptors as targets for the modulation of central serotonergic signaling
HUP0700395A2 (en) *	2007-06-07	2009-03-02	Sanofi Aventis	Substituted [1,2,4] triazolo [1,5-a] quinolines, process for their preparation, pharmaceutical compositions thereof, and intermediates
EP2456419B1 (en)	2009-07-21	2016-11-23	Oradin Pharmaceutical Ltd.	A3 adenosine receptor ligands for modulation of pigmentation
CA2898018C (en)	2013-02-01	2021-02-09	Wellstat Therapeutics Corporation	Substituted quinolin-4-amine compounds and pharmaceutical compositions thereof having anti-inflammatory, antifungal, antiparasitic and anticancer activity
KR101820909B1 (ko) *	2017-07-07	2018-01-23	퓨쳐메디신 주식회사	아데노신 유도체를 포함하는 만성신장질환 예방 및 치료용 약학적 조성물
AU2018334272B2 (en)	2017-09-15	2023-06-15	Forma Therapeutics, Inc.	Tetrahydro-imidazo quinoline compositions as CBP/p300 inhibitors
AU2019295790B2 (en)	2018-06-29	2023-07-13	Forma Therapeutics, Inc.	Inhibiting creb binding protein (CBP)
MX2021010829A (es) *	2019-03-15	2021-12-10	Forma Therapeutics Inc	Inhibición de la proteína de unión al elemento de respuesta a adenosín monofosfato (amp) cíclica (creb).
US11801243B2 (en)	2020-09-23	2023-10-31	Forma Therapeutics, Inc.	Bromodomain inhibitors for androgen receptor-driven cancers
US11795168B2 (en)	2020-09-23	2023-10-24	Forma Therapeutics, Inc.	Inhibiting cyclic amp-responsive element-binding protein (CREB) binding protein (CBP)

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4075343A (en) *	1976-09-13	1978-02-21	Pfizer Inc.	Anti-allergenic 5-alkoxyimidazo[1,2-A]quinoline-2-carboxylic acids and derivatives thereof
GB1596652A (en) *	1977-01-20	1981-08-26	Roussel Lab Ltd	Imidazo (1,2-a) quinoline-2-carboxylic acid and derivatives
US4644002A (en)	1979-02-09	1987-02-17	Roussel Uclaf	Imidazo[2,1-C]quinolines, useful as antiallergic agents
IL59104A (en) *	1979-02-09	1984-02-29	Roussel Uclaf	Heterotricyclic derivatives,process for their preparation and pharmaceutical compositions incorporating them
FR2448541A1 (fr)	1979-02-09	1980-09-05	Roussel Uclaf	Nouveaux derives de l'oxoimidazoquinoxaline et leurs sels, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
WO2000002861A1 (en)	1998-07-10	2000-01-20	The United States Of America, Represented By Secretary, Department Of Health And Human Services	A3 adenosine receptor antagonists
US6448253B1 (en) *	1998-09-16	2002-09-10	King Pharmaceuticals Research And Development, Inc.	Adenosine A3 receptor modulators
CN1207298C (zh)	1999-09-28	2005-06-22	株式会社大塚制药工厂	三唑并嘌呤衍生物、含有该衍生物的药物组合物和腺苷a3受体亲和剂
US7160890B2 (en) *	1999-12-02	2007-01-09	Osi Pharmaceuticals, Inc.	Compounds specific to adenosine A3 receptor and uses thereof
YU42703A (sh) *	2000-12-01	2006-03-03	Osi Pharmaceuticals Inc.	Jedinjenja specifična za dobijanje adenozinske a1,a2a i a3 receptore i njihove primene
RU2278112C2 (ru)	2001-05-31	2006-06-20	Санофи-Авентис	Производные аминохинолина и аминопиридина и их применение в качестве лигандов аденозина a3
HUP0105406A3 (en)	2001-12-21	2003-12-29	Sanofi Aventis	Imidazo[1,2-a]quinolin derivatives, process for their preparation, pharmaceutical compositions thereof and intermediates
HUP0105407A3 (en) *	2001-12-21	2004-04-28	Sanofi Aventis	Triazolo[1,5-a]quinolin derivatives, process for their preparation, pharmaceutical compositions thereof and intermediates
HUP0203976A3 (en)	2002-11-15	2004-08-30	Sanofi Aventis	Adenozine a3 receptors, process for their preparation and pharmaceutical compositions containing them

2002
- 2002-11-15 HU HU0203976A patent/HUP0203976A3/hu unknown
2003
- 2003-11-11 CN CNB2003801062293A patent/CN1332960C/zh not_active Expired - Fee Related
- 2003-11-11 DK DK03773882T patent/DK1560828T3/da active
- 2003-11-11 AU AU2003282263A patent/AU2003282263B2/en not_active Ceased
- 2003-11-11 UA UAA200505875A patent/UA78889C2/uk unknown
- 2003-11-11 KR KR1020057008683A patent/KR20050088291A/ko not_active Abandoned
- 2003-11-11 ME MEP-190/08A patent/MEP19008A/xx unknown
- 2003-11-11 AT AT03773882T patent/ATE325123T1/de active
- 2003-11-11 ES ES03773882T patent/ES2263039T3/es not_active Expired - Lifetime
- 2003-11-11 CA CA2505910A patent/CA2505910C/en not_active Expired - Fee Related
- 2003-11-11 SI SI200330299T patent/SI1560828T1/sl unknown
- 2003-11-11 PT PT03773882T patent/PT1560828E/pt unknown
- 2003-11-11 DE DE60305058T patent/DE60305058T2/de not_active Expired - Lifetime
- 2003-11-11 BR BR0316355-5A patent/BR0316355A/pt not_active IP Right Cessation
- 2003-11-11 MX MXPA05005198A patent/MXPA05005198A/es active IP Right Grant
- 2003-11-11 WO PCT/HU2003/000095 patent/WO2004046146A1/en active IP Right Grant
- 2003-11-11 RS YUP-2005/0364A patent/RS51320B/sr unknown
- 2003-11-11 NZ NZ540029A patent/NZ540029A/en not_active IP Right Cessation
- 2003-11-11 PL PL376837A patent/PL376837A1/pl not_active Application Discontinuation
- 2003-11-11 EP EP03773882A patent/EP1560828B9/en not_active Expired - Lifetime
- 2003-11-11 EA EA200500830A patent/EA007595B1/ru unknown
- 2003-11-11 JP JP2004552920A patent/JP4533148B2/ja not_active Expired - Fee Related
- 2003-11-14 AR ARP030104200A patent/AR041968A1/es unknown
- 2003-11-14 TW TW092131901A patent/TWI248934B/zh not_active IP Right Cessation
2005
- 2005-05-10 IL IL168516A patent/IL168516A/en not_active IP Right Cessation
- 2005-05-10 TN TNP2005000133A patent/TNSN05133A1/en unknown
- 2005-05-11 ZA ZA200503807A patent/ZA200503807B/en unknown
- 2005-05-16 US US11/130,429 patent/US7419977B2/en not_active Expired - Fee Related
- 2005-05-31 IS IS7874A patent/IS2456B/is unknown
- 2005-06-13 MA MA28334A patent/MA27501A1/fr unknown
- 2005-06-13 NO NO20052866A patent/NO20052866D0/no not_active Application Discontinuation
- 2005-06-14 CO CO05057645A patent/CO5690577A2/es not_active Application Discontinuation
- 2005-06-14 HR HR20050540A patent/HRP20050540A2/xx not_active Application Discontinuation
- 2005-11-07 HK HK05109885A patent/HK1077819A1/xx not_active IP Right Cessation
2006
- 2006-07-28 CY CY20061101054T patent/CY1105180T1/el unknown
2008
- 2008-06-17 US US12/140,512 patent/US7709489B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
MXPA05005198A (es)	2005-08-18
TW200413369A (en)	2004-08-01
CO5690577A2 (es)	2006-10-31
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Publication	Publication Date	Title
US7709489B2 (en)	2010-05-04	Imidazoquinoline derivatives as adenosine A3 receptor ligands
JP2011042653A (ja)	2011-03-03	アデノシン受容体リガンドとして有用なトリアゾロ−キノリン誘導体
EP2173346A2 (en)	2010-04-14	Use of compounds for preparing anti-tuberculosis agents
EP2167470B1 (en)	2011-03-16	Triazolo [1, 5-a]quinolines as adenosine a3 receptor ligands
KR100745307B1 (ko)	2007-08-01	아미노퀴놀린 유도체 및 아데노신 ａ３ 리간드로서의 이의 용도
KR20060065662A (ko)	2006-06-14	아미노퀴놀린 유도체 및 아데노신 ａ3 리간드로서의 이의용도
JP4530663B2 (ja)	2010-08-25	イミダゾキノリン誘導体
KR20070020335A (ko)	2007-02-20	아미노퀴놀린 유도체 및 아데노신 ａ３ 리간드로서의 이의용도

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