JPS5536456A - 1,2-benzodiazepine derivative and its preparation - Google Patents
1,2-benzodiazepine derivative and its preparationInfo
- Publication number
- JPS5536456A JPS5536456A JP11059378A JP11059378A JPS5536456A JP S5536456 A JPS5536456 A JP S5536456A JP 11059378 A JP11059378 A JP 11059378A JP 11059378 A JP11059378 A JP 11059378A JP S5536456 A JPS5536456 A JP S5536456A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- benzodiazepine
- preparation
- give
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- SVUOLADPCWQTTE-UHFFFAOYSA-N 1h-1,2-benzodiazepine Chemical class N1N=CC=CC2=CC=CC=C12 SVUOLADPCWQTTE-UHFFFAOYSA-N 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 2
- QOXHHGWPFLSWRJ-UHFFFAOYSA-N 1-methyl-2H-1,2-benzodiazepin-3-one Chemical compound CN1NC(=O)C=CC2=CC=CC=C12 QOXHHGWPFLSWRJ-UHFFFAOYSA-N 0.000 abstract 1
- MYMOFIZGZYHOMD-UHFFFAOYSA-N Dioxygen Chemical compound O=O MYMOFIZGZYHOMD-UHFFFAOYSA-N 0.000 abstract 1
- 150000001350 alkyl halides Chemical class 0.000 abstract 1
- 229940100198 alkylating agent Drugs 0.000 abstract 1
- 239000002168 alkylating agent Substances 0.000 abstract 1
- 229910001882 dioxygen Inorganic materials 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 230000001678 irradiating effect Effects 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A 1, 2-benzodiazepine devivative of formula I: (R1 is H or lower alkyl group; R2 is lower alkyl group).
EXAMPLE: 1-Methyl-3-oxo-1, 2-benzodiazepine.
USE: Central nervous depressants and their intermediates.
PROCESS: A compound of formula II is irradiated with light in the presence of oxygen gas to give the compound of formula I. The compound of formula II can be obtained by irradiating an N-iminoquinoline derivative of formula IV with light to give a compound of formula III, which is alkylated with an alkylating agent, e.g. an alkyl halide.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP53110593A JPS6033392B2 (en) | 1978-09-08 | 1978-09-08 | 1,2-benzodiazepine derivative and method for producing the same |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP53110593A JPS6033392B2 (en) | 1978-09-08 | 1978-09-08 | 1,2-benzodiazepine derivative and method for producing the same |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5536456A true JPS5536456A (en) | 1980-03-14 |
JPS6033392B2 JPS6033392B2 (en) | 1985-08-02 |
Family
ID=14539781
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP53110593A Expired JPS6033392B2 (en) | 1978-09-08 | 1978-09-08 | 1,2-benzodiazepine derivative and method for producing the same |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS6033392B2 (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001021969A1 (en) | 1999-09-17 | 2001-03-29 | Sumitomo Electric Industries, Ltd. | Dynamic pressure bearing with improved starting characteristics |
US6749339B1 (en) | 1999-09-03 | 2004-06-15 | Sumitomo Electric Industries, Ltd. | Hydrodynamic bearing assembly and spindle motor having the same |
-
1978
- 1978-09-08 JP JP53110593A patent/JPS6033392B2/en not_active Expired
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6749339B1 (en) | 1999-09-03 | 2004-06-15 | Sumitomo Electric Industries, Ltd. | Hydrodynamic bearing assembly and spindle motor having the same |
US7033078B2 (en) | 1999-09-03 | 2006-04-25 | Sumitomo Electric Industries, Ltd. | Hydrodynamic bearing assembly and spindle motor having the same |
US7360950B2 (en) | 1999-09-03 | 2008-04-22 | Sumitomo Electric Industries, Ltd. | Hydrodynamic bearing assembly |
WO2001021969A1 (en) | 1999-09-17 | 2001-03-29 | Sumitomo Electric Industries, Ltd. | Dynamic pressure bearing with improved starting characteristics |
US6702464B1 (en) | 1999-09-17 | 2004-03-09 | Sumitomo Electric Industries, Ltd. | Dynamic pressure bearing with improved starting characteristics |
Also Published As
Publication number | Publication date |
---|---|
JPS6033392B2 (en) | 1985-08-02 |
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