JPS55105666A - Piperidine derivative - Google Patents
Piperidine derivativeInfo
- Publication number
- JPS55105666A JPS55105666A JP1411179A JP1411179A JPS55105666A JP S55105666 A JPS55105666 A JP S55105666A JP 1411179 A JP1411179 A JP 1411179A JP 1411179 A JP1411179 A JP 1411179A JP S55105666 A JPS55105666 A JP S55105666A
- Authority
- JP
- Japan
- Prior art keywords
- benzyl
- formula
- benzoyl
- compound shown
- tetra
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A piperidine derivative shown by the formula I (R<1> is benzyl or benzoyl; R<2> is H or 1-3C lower alkyl) and its acid addition salt. EXAMPLE:A compound shown by the formula II (Bn is benzyl). USE:Useful as a starting material of moranoline, an N-lower alkylmoranoline, much available as a drug. PROCESS:For example, 2,3,4,6-tetra-O-benzyl (or benzoyl)-gamma-gluconic lactone is subjected to ammonolysis to give 2,3,4,6-tetra-O-benzyl (or benzoyl)-5-ketogluconic acid amide, which undergoes ring closure by an acidic catalyst to prepare a compound shown by the formula III. The compound is reduced by lithium aluminum hydride to give the desired compound shown by the formula I.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1411179A JPS55105666A (en) | 1979-02-08 | 1979-02-08 | Piperidine derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1411179A JPS55105666A (en) | 1979-02-08 | 1979-02-08 | Piperidine derivative |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS55105666A true JPS55105666A (en) | 1980-08-13 |
JPS6156228B2 JPS6156228B2 (en) | 1986-12-01 |
Family
ID=11851996
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP1411179A Granted JPS55105666A (en) | 1979-02-08 | 1979-02-08 | Piperidine derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS55105666A (en) |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5252587A (en) * | 1990-04-27 | 1993-10-12 | Merrell Dow Pharmaceuticals, Inc. | N-derivatives of 1-deoxy nojirimycin |
US5536732A (en) * | 1990-04-27 | 1996-07-16 | Merrell Pharmaceuticals Inc. | N-derivatives of 1-deoxy nojirimycin |
JP2008001711A (en) * | 2000-03-31 | 2008-01-10 | Univ Michigan State | Preparation of 1,5-dideoxy-1,5-iminohexitol from oxime or imine |
-
1979
- 1979-02-08 JP JP1411179A patent/JPS55105666A/en active Granted
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5252587A (en) * | 1990-04-27 | 1993-10-12 | Merrell Dow Pharmaceuticals, Inc. | N-derivatives of 1-deoxy nojirimycin |
US5536732A (en) * | 1990-04-27 | 1996-07-16 | Merrell Pharmaceuticals Inc. | N-derivatives of 1-deoxy nojirimycin |
JP2008001711A (en) * | 2000-03-31 | 2008-01-10 | Univ Michigan State | Preparation of 1,5-dideoxy-1,5-iminohexitol from oxime or imine |
Also Published As
Publication number | Publication date |
---|---|
JPS6156228B2 (en) | 1986-12-01 |
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