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ITMI910255A0 - Processo per la preparazione di acidi 3 acilammino-4- carbamoilossimetil-2-azetidinone-l-solfonici ed intermedi per la loro preparazione - Google Patents

Processo per la preparazione di acidi 3 acilammino-4- carbamoilossimetil-2-azetidinone-l-solfonici ed intermedi per la loro preparazione

Info

Publication number
ITMI910255A0
ITMI910255A0 IT91MI255A ITMI910255A ITMI910255A0 IT MI910255 A0 ITMI910255 A0 IT MI910255A0 IT 91MI255 A IT91MI255 A IT 91MI255A IT MI910255 A ITMI910255 A IT MI910255A IT MI910255 A0 ITMI910255 A0 IT MI910255A0
Authority
IT
Italy
Prior art keywords
preparation
carbamoyloxymethyl
azetidinone
acylamino
intermediates
Prior art date
Application number
IT91MI255A
Other languages
English (en)
Inventor
Giuseppe Guanti
Luca Banfi
Enrica Narisano
Renata Riva
Elso Manghisi
Giuseppe Cascio
Original Assignee
Luso Farmaco Inst
Stituto Luso Farmaco D Italia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Luso Farmaco Inst, Stituto Luso Farmaco D Italia filed Critical Luso Farmaco Inst
Priority to ITMI910255A priority Critical patent/IT1244699B/it
Publication of ITMI910255A0 publication Critical patent/ITMI910255A0/it
Priority to AU11873/92A priority patent/AU1187392A/en
Priority to PCT/EP1992/000175 priority patent/WO1992013837A1/en
Publication of ITMI910255A1 publication Critical patent/ITMI910255A1/it
Application granted granted Critical
Publication of IT1244699B publication Critical patent/IT1244699B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ITMI910255A 1991-02-01 1991-02-01 Processo per la preparazione di acidi 3 acilammino-4- carbamoilossimetil-2-azetidinone-l-solfonici ed intermedi per la loro preparazione IT1244699B (it)

Priority Applications (3)

Application Number Priority Date Filing Date Title
ITMI910255A IT1244699B (it) 1991-02-01 1991-02-01 Processo per la preparazione di acidi 3 acilammino-4- carbamoilossimetil-2-azetidinone-l-solfonici ed intermedi per la loro preparazione
AU11873/92A AU1187392A (en) 1991-02-01 1992-01-28 A process for the preparation of 3-acylamino-4-carbamoyloxymethyl-2-azetidinone-1-sulphonic acids and intermediates for the preparation thereof
PCT/EP1992/000175 WO1992013837A1 (en) 1991-02-01 1992-01-28 A process for the preparation of 3-acylamino-4-carbamoyloxymethyl-2-azetidinone-1-sulphonic acids and intermediates for the preparation thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITMI910255A IT1244699B (it) 1991-02-01 1991-02-01 Processo per la preparazione di acidi 3 acilammino-4- carbamoilossimetil-2-azetidinone-l-solfonici ed intermedi per la loro preparazione

Publications (3)

Publication Number Publication Date
ITMI910255A0 true ITMI910255A0 (it) 1991-02-01
ITMI910255A1 ITMI910255A1 (it) 1992-08-01
IT1244699B IT1244699B (it) 1994-08-08

Family

ID=11358378

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI910255A IT1244699B (it) 1991-02-01 1991-02-01 Processo per la preparazione di acidi 3 acilammino-4- carbamoilossimetil-2-azetidinone-l-solfonici ed intermedi per la loro preparazione

Country Status (3)

Country Link
AU (1) AU1187392A (it)
IT (1) IT1244699B (it)
WO (1) WO1992013837A1 (it)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6982251B2 (en) 2000-12-20 2006-01-03 Schering Corporation Substituted 2-azetidinones useful as hypocholesterolemic agents
SI1353696T1 (sl) 2001-01-26 2007-04-30 Schering Corp Kombinacije aktivatorja(-ev) peroksisomskega proliferatorja aktivirajocega receptorja (PPAR) in inhibitorja(-ev) absorpcije sterola in oblike zdravljenja za vaskularne indikacije
US7071181B2 (en) 2001-01-26 2006-07-04 Schering Corporation Methods and therapeutic combinations for the treatment of diabetes using sterol absorption inhibitors
AR035533A1 (es) 2001-01-26 2004-06-02 Schering Corp Uso de por lo menos un inhibidor de la absorcion de los esteroles o sus sales, solvatos, prodrogas farmaceuticamente aceptables o mezclas de los mismos para la preparacion de un medicamento para el tratamiento de la sitosterolemia, composiciones farmaceuticas, el uso de dichas composiciones para la
US7056906B2 (en) 2001-09-21 2006-06-06 Schering Corporation Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women
US7053080B2 (en) 2001-09-21 2006-05-30 Schering Corporation Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors
JP2005504091A (ja) 2001-09-21 2005-02-10 シェーリング コーポレイション ステロール吸収阻害剤としてアゼチジノンを用いる黄色腫の処置
JP2006508189A (ja) 2002-11-06 2006-03-09 シェーリング コーポレイション 自己免疫障害の処置のためのコレステロール吸収インヒビター
CN1756755A (zh) 2003-03-07 2006-04-05 先灵公司 取代的2-吖丁啶酮化合物、其制剂及其治疗高胆甾醇血症的用途
US7459442B2 (en) 2003-03-07 2008-12-02 Schering Corporation Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
US7208486B2 (en) 2003-03-07 2007-04-24 Schering Corporation Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
ATE406364T1 (de) 2003-03-07 2008-09-15 Schering Corp Substituierte azetidinon-derivate, deren pharmazeutische formulierungen und deren verwendung zur behandlung von hypercholesterolemia

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU564150B2 (en) * 1982-04-30 1987-08-06 Takeda Chemical Industries Ltd. 1-sulfo-2-azetidinone derivatives
US4502994A (en) * 1982-12-09 1985-03-05 Hoffmann-La Roche Inc. Enantiomeric synthesis of 3-amino-4-carbamoyloxymethyl-2-azetidonone-1-sulfate
IT1231770B (it) * 1989-08-02 1991-12-21 Consiglio Nazionale Ricerche Processo per la preparazione di monobattami ed intermedio di preparazione.

Also Published As

Publication number Publication date
ITMI910255A1 (it) 1992-08-01
IT1244699B (it) 1994-08-08
WO1992013837A1 (en) 1992-08-20
AU1187392A (en) 1992-09-07

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19970226