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IT1205349B - Determinate pirazolo-chinoline sostituite,procedimento per la loro preparazione,preparati farmaceutici contenenti questi composti e loro impiego terapeutico - Google Patents

Determinate pirazolo-chinoline sostituite,procedimento per la loro preparazione,preparati farmaceutici contenenti questi composti e loro impiego terapeutico

Info

Publication number
IT1205349B
IT1205349B IT49450/83A IT4945083A IT1205349B IT 1205349 B IT1205349 B IT 1205349B IT 49450/83 A IT49450/83 A IT 49450/83A IT 4945083 A IT4945083 A IT 4945083A IT 1205349 B IT1205349 B IT 1205349B
Authority
IT
Italy
Prior art keywords
kinolines
pyrazol
compounds
replaced
procedure
Prior art date
Application number
IT49450/83A
Other languages
English (en)
Other versions
IT8349450A0 (it
Inventor
Naokata Yokoyama
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of IT8349450A0 publication Critical patent/IT8349450A0/it
Application granted granted Critical
Publication of IT1205349B publication Critical patent/IT1205349B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A61P39/02—Antidotes

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Toxicology (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IT49450/83A 1982-12-08 1983-12-06 Determinate pirazolo-chinoline sostituite,procedimento per la loro preparazione,preparati farmaceutici contenenti questi composti e loro impiego terapeutico IT1205349B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/447,825 US4524146A (en) 1982-12-08 1982-12-08 Certain -2-heterocycle substituted pyrazoloquinolines

Publications (2)

Publication Number Publication Date
IT8349450A0 IT8349450A0 (it) 1983-12-06
IT1205349B true IT1205349B (it) 1989-03-15

Family

ID=23777905

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49450/83A IT1205349B (it) 1982-12-08 1983-12-06 Determinate pirazolo-chinoline sostituite,procedimento per la loro preparazione,preparati farmaceutici contenenti questi composti e loro impiego terapeutico

Country Status (9)

Country Link
US (1) US4524146A (it)
JP (1) JPS59110694A (it)
BE (1) BE898383A (it)
CH (1) CH656127A5 (it)
DE (1) DE3343922A1 (it)
FR (1) FR2537584B1 (it)
GB (1) GB2131801B (it)
IT (1) IT1205349B (it)
NL (1) NL8304224A (it)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2549833B1 (fr) * 1983-07-26 1985-11-08 Roussel Uclaf Derives de la pyrazolo /4,3-c/ cinnolin-3-one, leurs sels, procede de preparation, application a titre de medicaments, compositions les renfermant et produits intermediaires
CA1263651A (en) * 1984-07-09 1989-12-05 Ciba-Geigy Ag Certain ring-fused pyrazolo ¬3,4-d|-pyridin-3-one derivatives
US4602014A (en) * 1984-07-09 1986-07-22 Ciba-Geigy Corporation Ring-fused pyrazolo[3,4-d]-pyridin-3-one derivatives as benzodiazepine receptor modulators
PH21213A (en) * 1984-10-26 1987-08-21 Fujisawa Pharmaceutical Co Benzene- and pyrazole- fused heterocyclic compound and pharmaceutical composition comprising the same
JPS61112075A (ja) * 1984-11-05 1986-05-30 Shionogi & Co Ltd チエニルピラゾロキノリン誘導体
US4591589A (en) * 1985-01-16 1986-05-27 Roussel Uclaf 2-aryl pyrazolo[4,3-c]cinnolin-3-ones
US4758427A (en) * 1985-08-08 1988-07-19 Ciba-Geigy Corporation Enhanced absorption of psychoactive 2-aryl-pyrazolo quinolines as a solid molecular dispersion in polyvinylpyrrolidone
US4831013A (en) * 1986-03-20 1989-05-16 Ciba-Geigy Corporation 2-substituted-e-fused-[1,2,4]triazolo[1,5-c]pyrimidines, pharmaceutical compositions, and uses thereof
US4826854A (en) * 1986-11-25 1989-05-02 Ciba-Geigy Corporation Certain cycloalka-(b)-pyrazolo(3,4-d)-pyridin-3-one derivatives
US5192768A (en) * 1990-09-14 1993-03-09 Kyowa Hakko Kogyo Co., Ltd. Pyrazoloquinoline derivatives
US5334595A (en) * 1992-10-23 1994-08-02 Sterling Winthrop Inc. Pyrazoloquinolones as anticancer agents
ID16283A (id) * 1996-03-20 1997-09-18 Astra Pharma Prod Senyawa yang berguna dibidang farmasi
WO2001038329A1 (fr) * 1999-11-24 2001-05-31 Sumika Fine Chemicals Co., Ltd. Cristaux de mirtazapine anhydre et leur procede d'obtention
EP2164328B8 (en) * 2007-06-08 2013-09-11 Dart Neuroscience (Cayman) Ltd Therapeutic pyrazoloquinoline urea derivatives
US20110212053A1 (en) * 2008-06-19 2011-09-01 Dapeng Qian Phosphatidylinositol 3 kinase inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2009079A1 (it) * 1968-05-22 1970-01-30 Sandoz Sa
US4312870A (en) * 1979-06-21 1982-01-26 Ciba-Geigy Corporation Pyrazoloquinolines
DE3068673D1 (en) * 1979-06-21 1984-08-30 Ciba Geigy Ag Pyrazolo-quinolines, processes for their production, and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
FR2537584A1 (fr) 1984-06-15
IT8349450A0 (it) 1983-12-06
DE3343922A1 (de) 1984-06-28
CH656127A5 (de) 1986-06-13
NL8304224A (nl) 1984-07-02
GB2131801A (en) 1984-06-27
GB8332274D0 (en) 1984-01-11
US4524146A (en) 1985-06-18
JPS59110694A (ja) 1984-06-26
BE898383A (fr) 1984-06-06
FR2537584B1 (fr) 1987-01-16
GB2131801B (en) 1986-01-22

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