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IL163870A0 - Antiparasitic artemisinin derivatives (endoperoxides) - Google Patents

Antiparasitic artemisinin derivatives (endoperoxides)

Info

Publication number
IL163870A0
IL163870A0 IL16387003A IL16387003A IL163870A0 IL 163870 A0 IL163870 A0 IL 163870A0 IL 16387003 A IL16387003 A IL 16387003A IL 16387003 A IL16387003 A IL 16387003A IL 163870 A0 IL163870 A0 IL 163870A0
Authority
IL
Israel
Prior art keywords
endoperoxides
artemisinin derivatives
antiparasitic
antiparasitic artemisinin
derivatives
Prior art date
Application number
IL16387003A
Other languages
English (en)
Original Assignee
Bayer Business Services Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Business Services Gmbh filed Critical Bayer Business Services Gmbh
Publication of IL163870A0 publication Critical patent/IL163870A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/12Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains three hetero rings
    • C07D493/20Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/12Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains three hetero rings
    • C07D493/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL16387003A 2002-03-08 2003-02-24 Antiparasitic artemisinin derivatives (endoperoxides) IL163870A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02005233 2002-03-08
PCT/EP2003/001839 WO2003076446A1 (en) 2002-03-08 2003-02-24 Antiparasitic artemisinin derivatives (endoperoxides)

Publications (1)

Publication Number Publication Date
IL163870A0 true IL163870A0 (en) 2005-12-18

Family

ID=27798779

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16387003A IL163870A0 (en) 2002-03-08 2003-02-24 Antiparasitic artemisinin derivatives (endoperoxides)

Country Status (21)

Country Link
US (1) US20050119232A1 (pt)
EP (1) EP1485389B1 (pt)
JP (1) JP2005526073A (pt)
KR (1) KR20040104493A (pt)
CN (1) CN1649874A (pt)
AR (1) AR038842A1 (pt)
AT (1) ATE334987T1 (pt)
AU (1) AU2003215584A1 (pt)
BR (1) BR0308291A (pt)
CA (1) CA2478600A1 (pt)
DE (1) DE60307239D1 (pt)
HR (1) HRP20040927A2 (pt)
IL (1) IL163870A0 (pt)
MX (1) MXPA04008638A (pt)
NZ (1) NZ535084A (pt)
PL (1) PL372341A1 (pt)
RU (1) RU2004130284A (pt)
TW (1) TW200400964A (pt)
WO (1) WO2003076446A1 (pt)
YU (1) YU79304A (pt)
ZA (1) ZA200407102B (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004027871B3 (de) * 2004-06-08 2006-03-16 Lanxess Deutschland Gmbh Verfahren zur Herstellung von 10α-[4'-(S,S-Dioxothiomorpholin-1'-yl)]-10-desoxo-10-dihydroartemisinin
EP1714967A1 (en) * 2005-04-22 2006-10-25 Bayer HealthCare AG Antiparasitic artemisinin derivatives
KR101496988B1 (ko) * 2005-10-20 2015-03-03 에피팜 게엠베하 아르테미시닌 및 그의 유도체를 이용한 양성 착색점(반점)의 처치 및 예방
US8431611B2 (en) 2006-10-20 2013-04-30 Johns Hopkins University Artemisinin derivatives
US20100286154A1 (en) * 2007-11-15 2010-11-11 Susanne Christine Wieland-Berghausen Antihelmintic paste
US8815942B2 (en) 2010-10-20 2014-08-26 The Royal Institution For The Advancement Of Learning/Mcgill University Combination therapy and uses thereof for treatment and prevention of parasitic infection and disease
CN102010422B (zh) * 2010-11-23 2014-11-26 沈阳药科大学 含有胍基的青蒿素类衍生物及其应用
US8232417B1 (en) 2010-12-01 2012-07-31 Bioderm Research Artemisinin derivatives with natural amino acids, peptides, and amino sugars for skin imperfections and infection in mammals
CN103183682B (zh) * 2011-12-31 2015-10-14 沈阳药科大学 C-10位脲基取代的青蒿素衍生物及其制备方法和用途
AU2013250714A1 (en) * 2012-04-18 2014-11-27 Hadasit Medical Research Services And Development Ltd. Methods and compositions for treating viral infections

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5726203A (en) * 1993-07-19 1998-03-10 Li; Zelin Qinghaosu derivatives against AIDS
EP0974594A1 (en) * 1998-07-14 2000-01-26 The Hong Kong University of Science & Technology Artemisinin derivatives as anti-infective agent
DE69929203T2 (de) * 1998-07-14 2006-08-31 Bayer Healthcare Ag Antiparasitische artemisinin derivate (endoperoxide)

Also Published As

Publication number Publication date
NZ535084A (en) 2006-05-26
AR038842A1 (es) 2005-01-26
HRP20040927A2 (en) 2005-06-30
RU2004130284A (ru) 2005-05-10
KR20040104493A (ko) 2004-12-10
BR0308291A (pt) 2005-01-11
YU79304A (sh) 2006-08-17
CN1649874A (zh) 2005-08-03
JP2005526073A (ja) 2005-09-02
MXPA04008638A (es) 2005-04-19
WO2003076446A1 (en) 2003-09-18
AU2003215584A1 (en) 2003-09-22
US20050119232A1 (en) 2005-06-02
WO2003076446A8 (en) 2004-10-07
PL372341A1 (en) 2005-07-11
DE60307239D1 (de) 2006-09-14
ZA200407102B (en) 2005-09-06
EP1485389B1 (en) 2006-08-02
TW200400964A (en) 2004-01-16
EP1485389A1 (en) 2004-12-15
ATE334987T1 (de) 2006-08-15
CA2478600A1 (en) 2003-09-18

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