IL155841A0 - Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same - Google Patents

Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same

Info

Publication number: IL155841A0
Authority: IL; Israel
Prior art keywords: preparation; compositions containing; containing same; piperidine derivatives; heterocyclylalkyl piperidine
Prior art date: 2000-11-15

Application number

IL15584101A

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-15

Filing date

2001-11-14

Publication date

2003-12-23

2001-11-14 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2003-12-23 Publication of IL155841A0 publication Critical patent/IL155841A0/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

IL15584101A 2000-11-15 2001-11-14 Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same IL155841A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR0014738A FR2816618B1 (en)	2000-11-15	2000-11-15	HETEROCYCLYLALCOYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM
PCT/FR2001/003559 WO2002040474A2 (en)	2000-11-15	2001-11-14	Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents

Publications (1)

Publication Number	Publication Date
IL155841A0 true IL155841A0 (en)	2003-12-23

Family

ID=8856503

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL15584101A IL155841A0 (en)	2000-11-15	2001-11-14	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same

Country Status (28)

Country	Link
EP (2)	EP1695964A1 (en)
JP (1)	JP2004514661A (en)
KR (1)	KR100849608B1 (en)
CN (1)	CN1483031A (en)
AR (1)	AR034006A1 (en)
AT (1)	ATE337311T1 (en)
AU (2)	AU2002218365B2 (en)
BG (1)	BG107793A (en)
BR (1)	BR0115312A (en)
CA (1)	CA2429311A1 (en)
CZ (1)	CZ20031316A3 (en)
DE (1)	DE60122567T2 (en)
DK (1)	DK1337529T3 (en)
EA (1)	EA200300568A1 (en)
EE (1)	EE200300207A (en)
ES (1)	ES2271119T3 (en)
FR (1)	FR2816618B1 (en)
HR (1)	HRP20030379A2 (en)
HU (1)	HUP0303758A3 (en)
IL (1)	IL155841A0 (en)
NO (2)	NO20032187L (en)
PL (1)	PL363004A1 (en)
PT (1)	PT1337529E (en)
SK (1)	SK5822003A3 (en)
TN (1)	TNSN01160A1 (en)
WO (1)	WO2002040474A2 (en)
YU (1)	YU46803A (en)
ZA (1)	ZA200303794B (en)

Families Citing this family (37)

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Publication number	Priority date	Publication date	Assignee	Title
AU8974901A (en)	2000-07-26	2002-02-05	Smithkline Beecham Plc	Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0118238D0 (en) *	2001-07-26	2001-09-19	Smithkline Beecham Plc	Medicaments
EP2181996A1 (en)	2002-01-29	2010-05-05	Glaxo Group Limited	Aminopiperidine derivatives
US7109213B2 (en)	2002-01-29	2006-09-19	Glaxo Group Limited	Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
AR040336A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE TO PREPARE SUCH COMPOUND
AR040335A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	CYCLLOHEXAN OR CYCLHEXENE COMPOUND, USE OF THE SAME TO PREPARE A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, PROCEDURE AND INTERMEDIATE COMPOUNDS OF UTILITY TO PREPARE SUCH COMPOUND
FR2842807A1 (en) *	2002-07-23	2004-01-30	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME
GB0217294D0 (en) *	2002-07-25	2002-09-04	Glaxo Group Ltd	Medicaments
FR2844270B1 (en) *	2002-09-11	2006-05-19	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM
FR2844268B1 (en) *	2002-09-11	2004-10-22	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM
DE10256405A1 (en) *	2002-12-02	2004-06-17	Morphochem Aktiengesellschaft für kombinatorische Chemie	New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
EP1560821B8 (en)	2002-11-05	2010-05-19	Glaxo Group Limited	Antibacterial agents
JP2006515862A (en)	2002-12-04	2006-06-08	グラクソ　グループ　リミテッド	Quinolines and their nitrogenated derivatives and their use as antibacterial agents
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
US7232833B2 (en)	2003-03-28	2007-06-19	Novexel	4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2862301B1 (en) *	2003-11-17	2007-12-21	Aventis Pharma Sa	NEW PROCESS FOR THE PREPARATION OF 3-FLUORINATED QUINOLINES
FR2867472B1 (en) *	2004-03-12	2008-07-18	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
EP1846418A4 (en)	2005-01-25	2009-12-23	Glaxo Group Ltd	Antibacterial agents
WO2006081178A2 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
WO2006081179A1 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
EP1846417A4 (en)	2005-01-25	2009-12-23	Glaxo Group Ltd	Antibacterial agents
CA2599688A1 (en)	2005-03-01	2006-09-08	Wyeth	Cinnoline compounds and their use as liver x receptor modulators
MY150958A (en)	2005-06-16	2014-03-31	Astrazeneca Ab	Compounds for the treatment of multi-drug resistant bacterial infections
WO2007086016A1 (en)	2006-01-26	2007-08-02	Actelion Pharmaceuticals Ltd	Tetrahydropyrane antibiotics
ATE481406T1 (en)	2006-04-06	2010-10-15	Glaxo Group Ltd	PYRROLOQUINOXALINONE DERIVATIVES AS ANTIBACTERIAL AGENTS
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
WO2008152603A1 (en)	2007-06-15	2008-12-18	Actelion Pharmaceuticals Ltd	3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
US20110275661A1 (en)	2008-10-17	2011-11-10	Glaxo Group Limited	Tricyclic nitrogen compounds used as antibacterials
ES2561631T3 (en)	2009-01-15	2016-02-29	Glaxo Group Limited	Naphthyridine-2 (1H) -one compounds useful as antibacterial agents
CA2881935A1 (en) *	2012-08-15	2014-02-20	Glaxo Group Limited	Process for preparing a 1-(2-haolethyl)-4-piperidine carboxylate intermediate useful in the synthesis of umeclidinium bromide
WO2016027249A1 (en)	2014-08-22	2016-02-25	Glaxosmithkline Intellectual Property Development Limited	Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection
WO2016138988A1 (en) *	2015-03-02	2016-09-09	University Of Copenhagen	Piperazine inhibitors of bacterial gyrase and topoisomerase iv
TW201722965A (en)	2015-08-16	2017-07-01	葛蘭素史密斯克藍智慧財產發展有限公司	Compounds for use in antibacterial applications

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7908031A (en)	1979-11-01	1981-06-01	Acf Chemiefarma Nv	NEW QUINOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH A COMPOUND AND METHOD FOR PREPARING THESE COMPOUNDS.
JPH0239546A (en)	1988-07-29	1990-02-08	Origin Electric Co Ltd	Manufacture of hybrid integrated circuit
NZ232091A (en)	1989-01-16	1990-12-21	Bellon Labor Sa Roger	7-fluoro-8-(piperazin-1-yl)-4-oxo-1,4-dihydro-benzo(b)(1,8)naphthyridine-3-carboxylic acid derivatives, preparation and pharmaceutical compositions thereof
JP2002501061A (en) *	1998-01-26	2002-01-15	スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー	Quinoline derivatives for antibacterial agents
EP1144404A1 (en) *	1999-01-20	2001-10-17	Smithkline Beecham Plc	Piperidinylquinolines as protein tyrosine kinase inhibitors
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

2000
- 2000-11-15 FR FR0014738A patent/FR2816618B1/en not_active Expired - Fee Related
2001
- 2001-11-13 AR ARP010105289A patent/AR034006A1/en unknown
- 2001-11-14 CZ CZ20031316A patent/CZ20031316A3/en unknown
- 2001-11-14 AU AU2002218365A patent/AU2002218365B2/en not_active Ceased
- 2001-11-14 CN CNA018210996A patent/CN1483031A/en active Pending
- 2001-11-14 AT AT01996538T patent/ATE337311T1/en not_active IP Right Cessation
- 2001-11-14 EP EP06010725A patent/EP1695964A1/en not_active Withdrawn
- 2001-11-14 CA CA002429311A patent/CA2429311A1/en not_active Abandoned
- 2001-11-14 SK SK582-2003A patent/SK5822003A3/en unknown
- 2001-11-14 TN TNTNSN01160A patent/TNSN01160A1/en unknown
- 2001-11-14 AU AU1836502A patent/AU1836502A/en active Pending
- 2001-11-14 EE EEP200300207A patent/EE200300207A/en unknown
- 2001-11-14 HU HU0303758A patent/HUP0303758A3/en unknown
- 2001-11-14 WO PCT/FR2001/003559 patent/WO2002040474A2/en active IP Right Grant
- 2001-11-14 KR KR1020037006600A patent/KR100849608B1/en not_active IP Right Cessation
- 2001-11-14 DE DE60122567T patent/DE60122567T2/en not_active Expired - Fee Related
- 2001-11-14 ES ES01996538T patent/ES2271119T3/en not_active Expired - Lifetime
- 2001-11-14 PL PL01363004A patent/PL363004A1/en not_active Application Discontinuation
- 2001-11-14 DK DK01996538T patent/DK1337529T3/en active
- 2001-11-14 BR BR0115312-9A patent/BR0115312A/en not_active Application Discontinuation
- 2001-11-14 EP EP01996538A patent/EP1337529B1/en not_active Expired - Lifetime
- 2001-11-14 IL IL15584101A patent/IL155841A0/en unknown
- 2001-11-14 EA EA200300568A patent/EA200300568A1/en unknown
- 2001-11-14 JP JP2002543484A patent/JP2004514661A/en active Pending
- 2001-11-14 PT PT01996538T patent/PT1337529E/en unknown
- 2001-11-14 YU YU46803A patent/YU46803A/en unknown
2003
- 2003-05-09 BG BG107793A patent/BG107793A/en unknown
- 2003-05-13 HR HR20030379A patent/HRP20030379A2/en not_active Application Discontinuation
- 2003-05-14 NO NO20032187A patent/NO20032187L/en unknown
- 2003-05-15 ZA ZA200303794A patent/ZA200303794B/en unknown
2007
- 2007-04-25 NO NO20072142A patent/NO20072142L/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
HRP20030379A2 (en)	2005-04-30
EP1695964A1 (en)	2006-08-30
HUP0303758A3 (en)	2009-08-28
EP1337529A2 (en)	2003-08-27
YU46803A (en)	2006-05-25
AU1836502A (en)	2002-05-27
NO20072142L (en)	2007-04-25
AR034006A1 (en)	2004-01-21
BR0115312A (en)	2003-09-23
CA2429311A1 (en)	2002-05-23
WO2002040474A2 (en)	2002-05-23
ATE337311T1 (en)	2006-09-15
AU2002218365B2 (en)	2007-07-05
KR100849608B1 (en)	2008-07-31
NO20032187D0 (en)	2003-05-14
SK5822003A3 (en)	2004-06-08
TNSN01160A1 (en)	2005-11-10
DE60122567D1 (en)	2006-10-05
HUP0303758A2 (en)	2004-03-01
CN1483031A (en)	2004-03-17
ES2271119T3 (en)	2007-04-16
FR2816618A1 (en)	2002-05-17
EP1337529B1 (en)	2006-08-23
CZ20031316A3 (en)	2003-10-15
ZA200303794B (en)	2004-06-29
FR2816618B1 (en)	2002-12-27
KR20030060934A (en)	2003-07-16
EA200300568A1 (en)	2003-12-25
PT1337529E (en)	2006-12-29
BG107793A (en)	2004-08-31
EE200300207A (en)	2003-08-15
PL363004A1 (en)	2004-11-15
DE60122567T2 (en)	2007-08-23
WO2002040474A3 (en)	2002-10-31
NO20032187L (en)	2003-06-26
JP2004514661A (en)	2004-05-20
DK1337529T3 (en)	2006-12-18

Publication	Publication Date	Title
IL155841A0 (en)	2003-12-23	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same
IL151209A0 (en)	2003-04-10	Pharmaceutical compositions containing 3-aminoazetidine derivatives, novel derivatives and their preparation
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