IL148837A0 - Isoxazolecarboxamide derivatives - Google Patents

Isoxazolecarboxamide derivatives

Info

Publication number: IL148837A0
Authority: IL; Israel
Prior art keywords: isoxazolecarboxamide; derivatives; isoxazolecarboxamide derivatives
Prior art date: 1999-10-18

Application number

IL14883700A

Other languages

English (en)

Original Assignee

Recordati Chem Pharm

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-10-18

Filing date

2000-10-16

Publication date

2002-09-12

2000-10-16 Application filed by Recordati Chem Pharm filed Critical Recordati Chem Pharm

2002-09-12 Publication of IL148837A0 publication Critical patent/IL148837A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Urology & Nephrology (AREA)
Ophthalmology & Optometry (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Cardiology (AREA)
Gynecology & Obstetrics (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Heart & Thoracic Surgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

IL14883700A 1999-10-18 2000-10-16 Isoxazolecarboxamide derivatives IL148837A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IT1999MI002173A IT1314191B1 (it)	1999-10-18	1999-10-18	Derivati isossazolcarbossamidici
PCT/EP2000/010144 WO2001029015A2 (en)	1999-10-18	2000-10-16	Isoxazolecarboxamide derivatives as alpha1-adrenergic receptor antagonists

Publications (1)

Publication Number	Publication Date
IL148837A0 true IL148837A0 (en)	2002-09-12

Family

ID=11383797

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL14883700A IL148837A0 (en)	1999-10-18	2000-10-16	Isoxazolecarboxamide derivatives

Country Status (25)

Country	Link
EP (1)	EP1226131B1 (xx)
JP (1)	JP2003512362A (xx)
KR (1)	KR20020038944A (xx)
CN (1)	CN1139579C (xx)
AR (1)	AR029400A1 (xx)
AT (1)	ATE256670T1 (xx)
AU (1)	AU757614B2 (xx)
BR (1)	BR0014851A (xx)
CA (1)	CA2385472A1 (xx)
DE (1)	DE60007347T2 (xx)
DK (1)	DK1226131T3 (xx)
ES (1)	ES2210033T3 (xx)
HK (1)	HK1044940A1 (xx)
HU (1)	HUP0203184A3 (xx)
IL (1)	IL148837A0 (xx)
IT (1)	IT1314191B1 (xx)
MX (1)	MXPA02003432A (xx)
MY (1)	MY120400A (xx)
NO (1)	NO20021803L (xx)
NZ (1)	NZ517884A (xx)
PL (1)	PL356990A1 (xx)
PT (1)	PT1226131E (xx)
RU (1)	RU2002113096A (xx)
WO (1)	WO2001029015A2 (xx)
ZA (1)	ZA200203942B (xx)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN101277952B (zh)	2005-10-11	2011-09-28	弗·哈夫曼-拉罗切有限公司	异*唑衍生物
BRPI0618383A2 (pt)	2005-11-09	2011-08-30	Hoffmann La Roche	derivados de 3-aril-isoxazol-4-carbonil-benzofurano
RU2426731C2 (ru)	2005-12-23	2011-08-20	Ф. Хоффманн-Ля Рош Аг	Производные арил-изоксазоло-4-ил-оксадиазола
ES2371935T3 (es)	2005-12-27	2012-01-11	F. Hoffmann-La Roche Ag	Derivados de aril-isoxazol-4-il-imidazol.
BRPI0706560A2 (pt)	2006-01-17	2011-03-29	Hoffmann La Roche	derivados de aril-isoxazol-4-il-imidazo [1,2-a] piridina úteis para o tratamento de doença de alzheimer por intermédio de receptores gaba
AU2007267183B2 (en)	2006-05-31	2011-10-20	F. Hoffmann-La Roche Ag	Aryl-4-ethynyl-isoxazole derivatives
BRPI0814718A2 (pt)	2007-06-22	2015-02-24	Hoffmann La Roche	Derivados de isoxazol-imidazol
MX2010005753A (es)	2007-12-04	2010-06-15	Hoffmann La Roche	Derivados de isoxazolo-pirazina.
US7902201B2 (en)	2007-12-04	2011-03-08	Hoffmann-La Roche Inc.	Isoxazolo-pyrazine derivatives
US7943619B2 (en)	2007-12-04	2011-05-17	Hoffmann-La Roche Inc.	Isoxazolo-pyridazine derivatives
WO2010081851A1 (en)	2009-01-14	2010-07-22	Genoscience Pharma	Piperidin-4-ylpiperazine compounds for the treatment of hcv infection
TW201033201A (en)	2009-02-19	2010-09-16	Hoffmann La Roche	Isoxazole-isoxazole and isoxazole-isothiazole derivatives
US8389550B2 (en)	2009-02-25	2013-03-05	Hoffmann-La Roche Inc.	Isoxazoles / O-pyridines with ethyl and ethenyl linker
US8222246B2 (en)	2009-04-02	2012-07-17	Hoffmann-La Roche Inc.	Substituted isoxazoles
US20100280019A1 (en)	2009-04-30	2010-11-04	Roland Jakob-Roetne	Isoxazoles
CN102414206B (zh)	2009-05-05	2014-11-05	霍夫曼-拉罗奇有限公司	异*唑-吡啶衍生物
KR101384829B1 (ko)	2009-05-05	2014-04-15	에프. 호프만-라 로슈 아게	이속사졸-피라졸 유도체
US8410104B2 (en)	2009-05-05	2013-04-02	Hoffmann-La Roche Inc.	Pyridazines
AU2010244551A1 (en)	2009-05-05	2011-12-01	F. Hoffmann-La Roche Ag	Isoxazole-thiazole derivatives as GABA A receptor inverse agonists for use in the treatment of cognitive disorders
KR101354416B1 (ko)	2009-05-07	2014-02-19	에프. 호프만-라 로슈 아게	감마-아미노부티르산 조절제로서 이속사졸-피리딘 유도체
US8785435B2 (en)	2011-10-20	2014-07-22	Hoffmann-La Roche Inc.	Solid forms
CN113121540B (zh) *	2020-01-15	2024-01-26	鲁南制药集团股份有限公司	一种西格列汀游离碱的合成方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IT1254469B (it) *	1992-02-25	1995-09-25	Recordati Chem Pharm	Derivati benzopiranici e benzotiopiranici
IT1266582B1 (it) *	1993-07-30	1997-01-09	Recordati Chem Pharm	Derivati (di)azacicloesanici e diazacicloeptanici
DE4425146A1 (de) *	1994-07-15	1996-01-18	Basf Ag	Verwendung heterocyclischer Verbindungen

1999
- 1999-10-18 IT IT1999MI002173A patent/IT1314191B1/it active
2000
- 2000-10-10 MY MYPI20004718A patent/MY120400A/en unknown
- 2000-10-16 DK DK00992436T patent/DK1226131T3/da active
- 2000-10-16 DE DE60007347T patent/DE60007347T2/de not_active Expired - Fee Related
- 2000-10-16 KR KR1020027004663A patent/KR20020038944A/ko not_active Application Discontinuation
- 2000-10-16 AT AT00992436T patent/ATE256670T1/de not_active IP Right Cessation
- 2000-10-16 RU RU2002113096/04A patent/RU2002113096A/ru not_active Application Discontinuation
- 2000-10-16 CA CA002385472A patent/CA2385472A1/en not_active Abandoned
- 2000-10-16 WO PCT/EP2000/010144 patent/WO2001029015A2/en active IP Right Grant
- 2000-10-16 NZ NZ517884A patent/NZ517884A/en unknown
- 2000-10-16 AU AU28347/01A patent/AU757614B2/en not_active Ceased
- 2000-10-16 ES ES00992436T patent/ES2210033T3/es not_active Expired - Lifetime
- 2000-10-16 HU HU0203184A patent/HUP0203184A3/hu unknown
- 2000-10-16 EP EP00992436A patent/EP1226131B1/en not_active Expired - Lifetime
- 2000-10-16 BR BR0014851-2A patent/BR0014851A/pt not_active IP Right Cessation
- 2000-10-16 PT PT00992436T patent/PT1226131E/pt unknown
- 2000-10-16 PL PL00356990A patent/PL356990A1/xx not_active Application Discontinuation
- 2000-10-16 MX MXPA02003432A patent/MXPA02003432A/es not_active Application Discontinuation
- 2000-10-16 IL IL14883700A patent/IL148837A0/xx unknown
- 2000-10-16 JP JP2001531815A patent/JP2003512362A/ja active Pending
- 2000-10-16 CN CNB008143226A patent/CN1139579C/zh not_active Expired - Fee Related
- 2000-10-18 AR ARP000105475A patent/AR029400A1/es not_active Application Discontinuation
2002
- 2002-04-17 NO NO20021803A patent/NO20021803L/no not_active Application Discontinuation
- 2002-05-17 ZA ZA200203942A patent/ZA200203942B/en unknown
- 2002-08-13 HK HK02105918.6A patent/HK1044940A1/zh unknown

Also Published As

Publication number	Publication date
DK1226131T3 (da)	2004-04-19
AU2834701A (en)	2001-04-30
AR029400A1 (es)	2003-06-25
EP1226131A2 (en)	2002-07-31
BR0014851A (pt)	2002-06-11
ZA200203942B (en)	2003-01-02
DE60007347T2 (de)	2004-09-02
HK1044940A1 (zh)	2002-11-08
PT1226131E (pt)	2004-05-31
HUP0203184A2 (hu)	2003-01-28
MY120400A (en)	2005-10-31
HUP0203184A3 (en)	2004-12-28
CN1379767A (zh)	2002-11-13
NZ517884A (en)	2003-08-29
ITMI992173A1 (it)	2001-04-18
DE60007347D1 (de)	2004-01-29
ATE256670T1 (de)	2004-01-15
NO20021803D0 (no)	2002-04-17
CA2385472A1 (en)	2001-04-26
NO20021803L (no)	2002-06-17
IT1314191B1 (it)	2002-12-06
ES2210033T3 (es)	2004-07-01
WO2001029015A3 (en)	2001-11-01
KR20020038944A (ko)	2002-05-24
WO2001029015A2 (en)	2001-04-26
RU2002113096A (ru)	2003-11-10
ITMI992173A0 (it)	1999-10-18
EP1226131B1 (en)	2003-12-17
AU757614B2 (en)	2003-02-27
CN1139579C (zh)	2004-02-25
PL356990A1 (en)	2004-07-12
MXPA02003432A (es)	2002-08-20
JP2003512362A (ja)	2003-04-02

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PL351407A1 (en)	2003-04-22	Thio-oxindole derivatives
IL146282A0 (en)	2002-07-25	Thio-oxindole derivatives
GB9907134D0 (en)	1999-05-19	Antimor napthylcombretastatin derivatives
SI1226131T1 (en)	2004-04-30	Isoxazolecarboxamide derivatives
SI1178984T1 (en)	2003-08-31	1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives
HK1043987A1 (zh)	2002-10-04	硫-羥吲衍生物
SI1200445T1 (en)	2004-02-29	Thienopyranecarboxamide derivatives