IL123551A0 - Tricyclic erythromycin derivatives - Google Patents
Tricyclic erythromycin derivativesInfo
- Publication number
- IL123551A0 IL123551A0 IL12355196A IL12355196A IL123551A0 IL 123551 A0 IL123551 A0 IL 123551A0 IL 12355196 A IL12355196 A IL 12355196A IL 12355196 A IL12355196 A IL 12355196A IL 123551 A0 IL123551 A0 IL 123551A0
- Authority
- IL
- Israel
- Prior art keywords
- compounds
- erythromycin derivatives
- tricyclic
- tricyclic erythromycin
- antibacterial
- Prior art date
Links
- ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 230000000844 anti-bacterial effect Effects 0.000 abstract 2
- 150000002148 esters Chemical class 0.000 abstract 1
- 208000015181 infectious disease Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US55524695A | 1995-11-08 | 1995-11-08 | |
| PCT/US1996/016585 WO1997017356A1 (en) | 1995-11-08 | 1996-10-17 | Tricyclic erythromycin derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL123551A0 true IL123551A0 (en) | 1998-10-30 |
Family
ID=24216555
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL12355196A IL123551A0 (en) | 1995-11-08 | 1996-10-17 | Tricyclic erythromycin derivatives |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP0876388B1 (xx) |
| JP (1) | JP2000500133A (xx) |
| KR (1) | KR19990067492A (xx) |
| AT (1) | ATE259823T1 (xx) |
| AU (1) | AU7447096A (xx) |
| DE (1) | DE69631609T2 (xx) |
| DK (1) | DK0876388T3 (xx) |
| ES (1) | ES2218604T3 (xx) |
| IL (1) | IL123551A0 (xx) |
| MX (1) | MX9803692A (xx) |
| PT (1) | PT876388E (xx) |
| WO (1) | WO1997017356A1 (xx) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6274715B1 (en) * | 1995-11-08 | 2001-08-14 | Abbott Laboratories | Tricyclic erythromycin derivatives |
| ES2244716T3 (es) * | 1996-09-04 | 2005-12-16 | Abbott Laboratories | Cetolidos 6-o-sustituidos que tienen actividad antibacteriana. |
| UA51730C2 (uk) * | 1996-09-04 | 2002-12-16 | Ебботт Лабораторіз | 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців |
| US5922683A (en) * | 1997-05-29 | 1999-07-13 | Abbott Laboratories | Multicyclic erythromycin derivatives |
| PL337066A1 (en) * | 1997-05-29 | 2000-07-31 | Abbott Lab | Polycyclic derivatives of erythromycin |
| ZA987689B (en) * | 1997-09-02 | 1999-02-24 | Abbott Lab | 3-descladinose 6-O substituted erythromycin derivatives |
| EP1025114B1 (en) * | 1997-09-30 | 2004-02-25 | Abbott Laboratories | 3'-n-modified 6-o-substituted erythromycin ketolide derivatives having antibacterial activity |
| US6034069A (en) * | 1997-09-30 | 2000-03-07 | Abbott Laboratories | 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity |
| CO4990972A1 (es) * | 1997-10-29 | 2000-12-26 | Abbott Lab | Derivados de eritromicina en puente 6,11 |
| US6046171A (en) * | 1997-10-29 | 2000-04-04 | Abbott Laboratories | 6,11-bridged erythromycin derivatives |
| US6124269A (en) * | 1997-10-29 | 2000-09-26 | Abbott Laboratories | 2-Halo-6-O-substituted ketolide derivatives |
| PA8461401A1 (es) * | 1997-10-29 | 2000-05-24 | Pfizer Prod Inc | Derivados de eritromicina triciclicos |
| AP1060A (en) | 1998-01-02 | 2002-04-23 | Pfizer Prod Inc | Novel erythromycin derivatives. |
| PT952157E (pt) * | 1998-04-24 | 2003-11-28 | Pfizer Prod Inc | Derivados 9a, 11b-desidro de 9-oxima-3-ceto-6-o-metileritromicina |
| US6248719B1 (en) | 1998-06-03 | 2001-06-19 | Pfizer Inc | Tricyclic 3-keto derivatives of 6-O-methylerthromycin |
| JP4573925B2 (ja) * | 1998-07-09 | 2010-11-04 | アベンティス・ファーマ・ソシエテ・アノニム | 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用 |
| FR2780977B1 (fr) * | 1998-07-09 | 2000-09-01 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| US6472372B1 (en) | 2000-12-06 | 2002-10-29 | Ortho-Mcneil Pharmaceuticals, Inc. | 6-O-Carbamoyl ketolide antibacterials |
| JP2005503416A (ja) | 2001-09-17 | 2005-02-03 | オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド | ６−ｏ−カルバメート−１１，１２−ラクト−ケトライド抗菌剤 |
| HUP0500018A3 (en) | 2001-12-05 | 2009-09-28 | Ortho Mcneil Pharm Inc | 6-o-acyl ketolide derivatives of erythromycine processes for preparing them and using them as antibacterials |
| CA2487918A1 (en) * | 2002-05-31 | 2003-12-11 | Janssen Pharmaceutica N.V. | 3-descladinosyl-6-o-carbamoyl and 6-o-carbonoyl macrolide antibacterial agents |
| ES2331867B1 (es) | 2008-07-17 | 2010-10-27 | Entrechem, S.L. | Sintesis enzimatica de derivados enantiomericamente enriquecidos de trans-ciclopentano- 1,2-diaminas. |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR0166096B1 (ko) * | 1990-11-28 | 1999-01-15 | 우에하라 아키라 | 6-0-메틸에리쓰로마이신 a 유도체 |
| US5523399A (en) * | 1991-12-27 | 1996-06-04 | Taisho Pharmaceutical Co., Ltd. | 5-O-desosaminylerythronolide derivatives |
| WO1993021200A1 (fr) * | 1992-04-22 | 1993-10-28 | Taisho Pharmaceutical Co., Ltd. | Derive de 5-o-desosaminylerythronolide a |
-
1996
- 1996-10-17 EP EP96936579A patent/EP0876388B1/en not_active Expired - Lifetime
- 1996-10-17 WO PCT/US1996/016585 patent/WO1997017356A1/en not_active Application Discontinuation
- 1996-10-17 PT PT96936579T patent/PT876388E/pt unknown
- 1996-10-17 DE DE69631609T patent/DE69631609T2/de not_active Expired - Lifetime
- 1996-10-17 AT AT96936579T patent/ATE259823T1/de not_active IP Right Cessation
- 1996-10-17 ES ES96936579T patent/ES2218604T3/es not_active Expired - Lifetime
- 1996-10-17 JP JP9518186A patent/JP2000500133A/ja active Pending
- 1996-10-17 KR KR1019980703512A patent/KR19990067492A/ko not_active Application Discontinuation
- 1996-10-17 AU AU74470/96A patent/AU7447096A/en not_active Abandoned
- 1996-10-17 DK DK96936579T patent/DK0876388T3/da active
- 1996-10-17 IL IL12355196A patent/IL123551A0/xx unknown
-
1998
- 1998-05-08 MX MX9803692A patent/MX9803692A/es not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| MX9803692A (es) | 1998-09-30 |
| PT876388E (pt) | 2004-07-30 |
| EP0876388B1 (en) | 2004-02-18 |
| KR19990067492A (ko) | 1999-08-25 |
| DE69631609D1 (en) | 2004-03-25 |
| ES2218604T3 (es) | 2004-11-16 |
| AU7447096A (en) | 1997-05-29 |
| DE69631609T2 (de) | 2005-01-05 |
| JP2000500133A (ja) | 2000-01-11 |
| DK0876388T3 (da) | 2004-06-07 |
| EP0876388A1 (en) | 1998-11-11 |
| ATE259823T1 (de) | 2004-03-15 |
| WO1997017356A1 (en) | 1997-05-15 |
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