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HRP20110558T1 - Malatne soli i polimorfi od (3s, 5s)-7-[3-amino-5-metil-piperidinil]-1-ciklopropil-1, 4-dihidro-8-metoksi-4-okso-3-kinolinkarboksilne kiseline - Google Patents

Malatne soli i polimorfi od (3s, 5s)-7-[3-amino-5-metil-piperidinil]-1-ciklopropil-1, 4-dihidro-8-metoksi-4-okso-3-kinolinkarboksilne kiseline Download PDF

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Publication number
HRP20110558T1
HRP20110558T1 HR20110558T HRP20110558T HRP20110558T1 HR P20110558 T1 HRP20110558 T1 HR P20110558T1 HR 20110558 T HR20110558 T HR 20110558T HR P20110558 T HRP20110558 T HR P20110558T HR P20110558 T1 HRP20110558 T1 HR P20110558T1
Authority
HR
Croatia
Prior art keywords
salt
malate
image
hydrate
pattern
Prior art date
Application number
HR20110558T
Other languages
English (en)
Croatian (hr)
Inventor
Lee Redman-Furey Nancy
Ellen Godlewski Jane
Lloyd Dicks Michael
Original Assignee
Warner Chilcott Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38441484&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20110558(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Warner Chilcott Company filed Critical Warner Chilcott Company
Publication of HRP20110558T1 publication Critical patent/HRP20110558T1/hr

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
HR20110558T 2006-03-28 2007-03-26 Malatne soli i polimorfi od (3s, 5s)-7-[3-amino-5-metil-piperidinil]-1-ciklopropil-1, 4-dihidro-8-metoksi-4-okso-3-kinolinkarboksilne kiseline HRP20110558T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78648306P 2006-03-28 2006-03-28
PCT/IB2007/051055 WO2007110834A2 (en) 2006-03-28 2007-03-26 Malate salts, and polymorphs of (3s,5s)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid

Publications (1)

Publication Number Publication Date
HRP20110558T1 true HRP20110558T1 (hr) 2011-09-30

Family

ID=38441484

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20110558T HRP20110558T1 (hr) 2006-03-28 2007-03-26 Malatne soli i polimorfi od (3s, 5s)-7-[3-amino-5-metil-piperidinil]-1-ciklopropil-1, 4-dihidro-8-metoksi-4-okso-3-kinolinkarboksilne kiseline

Country Status (27)

Country Link
US (1) US8039485B2 (pl)
EP (1) EP2001862B1 (pl)
JP (1) JP5097967B2 (pl)
KR (1) KR101102288B1 (pl)
AR (2) AR060189A1 (pl)
AT (1) ATE507219T1 (pl)
AU (1) AU2007230630B2 (pl)
BR (1) BRPI0709772B8 (pl)
CA (1) CA2647346C (pl)
CY (1) CY1111683T1 (pl)
DE (1) DE602007014191D1 (pl)
DK (1) DK2001862T3 (pl)
ES (1) ES2366150T3 (pl)
HR (1) HRP20110558T1 (pl)
IL (1) IL193990A (pl)
MA (1) MA30554B1 (pl)
MX (1) MX2008012328A (pl)
MY (1) MY148393A (pl)
NZ (1) NZ570494A (pl)
PE (1) PE20080175A1 (pl)
PL (1) PL2001862T3 (pl)
PT (1) PT2001862E (pl)
SI (1) SI2001862T1 (pl)
SM (1) SMP200800058B (pl)
TW (1) TWI364419B (pl)
WO (1) WO2007110834A2 (pl)
ZA (1) ZA200807158B (pl)

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US8658183B2 (en) * 2007-08-09 2014-02-25 Taigen Biotechnology Company, Ltd. Antimicrobial parenteral formulation
AU2008358909B2 (en) * 2008-07-01 2012-12-13 Taigen Biotechnology Co., Ltd. Treatment of antibiotic-resistant bacteria infection
CN101618039B (zh) * 2008-07-02 2012-04-11 太景生物科技股份有限公司 肺炎的治疗药物
US8553466B2 (en) 2010-03-04 2013-10-08 Samsung Electronics Co., Ltd. Non-volatile memory device, erasing method thereof, and memory system including the same
CZ304984B6 (cs) 2012-10-12 2015-03-11 Zentiva, K.S. Zlepšený způsob výroby a nové intermediáty syntézy elvitegraviru
CZ304983B6 (cs) * 2012-10-12 2015-03-11 Zentiva, K.S. Způsob výroby a nové intermediáty syntézy elvitegraviru
CN103145615B (zh) * 2013-03-20 2015-07-29 浙江医药股份有限公司 一种奈诺沙星螯合物的后处理方法
CN114437026A (zh) * 2021-10-26 2022-05-06 浙江医药股份有限公司新昌制药厂 一种低组合物杂质的苹果酸奈诺沙星原料药及其制备方法
CN116332831A (zh) * 2023-03-15 2023-06-27 浙江医药股份有限公司新昌制药厂 氨基被Boc保护的3-氨基-5-甲基哌啶的提纯方法

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Also Published As

Publication number Publication date
WO2007110834A2 (en) 2007-10-04
RU2008134544A (ru) 2010-05-10
SI2001862T1 (sl) 2011-10-28
MY148393A (en) 2013-04-15
JP5097967B2 (ja) 2012-12-12
MA30554B1 (fr) 2009-07-01
AU2007230630A1 (en) 2007-10-04
US8039485B2 (en) 2011-10-18
SMAP200800058A (it) 2008-10-29
US20070232650A1 (en) 2007-10-04
EP2001862A2 (en) 2008-12-17
RU2417222C2 (ru) 2011-04-27
EP2001862B1 (en) 2011-04-27
ZA200807158B (en) 2009-09-30
AR060189A1 (es) 2008-05-28
DE602007014191D1 (en) 2011-06-09
ATE507219T1 (de) 2011-05-15
PE20080175A1 (es) 2008-03-14
BRPI0709772B8 (pt) 2021-05-25
CA2647346C (en) 2011-07-19
MX2008012328A (es) 2008-10-09
IL193990A (en) 2014-12-31
TWI364419B (en) 2012-05-21
NZ570494A (en) 2011-09-30
BRPI0709772B1 (pt) 2019-10-15
SMP200800058B (it) 2009-09-07
BRPI0709772A2 (pt) 2011-07-26
TW200808759A (en) 2008-02-16
DK2001862T3 (da) 2011-08-08
PL2001862T3 (pl) 2011-09-30
JP2009531417A (ja) 2009-09-03
ES2366150T3 (es) 2011-10-17
KR20090004887A (ko) 2009-01-12
KR101102288B1 (ko) 2012-01-03
CA2647346A1 (en) 2007-10-04
CY1111683T1 (el) 2015-10-07
AR060377A1 (es) 2008-06-11
PT2001862E (pt) 2011-07-20
WO2007110834A3 (en) 2007-12-06
AU2007230630B2 (en) 2012-12-20

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