HK1139399A1 - - Google Patents

Info

Publication number: HK1139399A1
Authority: HK; Hong Kong

Application number

HK10106008.5A

Inventor

Sean Dalziel

Leticia M Preza

Miroslav Rapta

Pierre-Jean Colson

Original Assignee

Theravance Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-02-28

Filing date

2010-06-15

Publication date

2010-09-17

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39620376&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1139399(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2010-06-15 Application filed by Theravance Inc filed Critical Theravance Inc

2010-09-17 Publication of HK1139399A1 publication Critical patent/HK1139399A1/xx

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Emergency Medicine (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pain & Pain Management (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

HK10106008.5A 2007-02-28 2010-06-15 HK1139399A1 (xx)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US90409007P	2007-02-28	2007-02-28
PCT/US2008/002583 WO2008106159A1 (en)	2007-02-28	2008-02-27	Crystalline forms of an 8-azabicyclo[3.2.1]octane compound

Publications (1)

Publication Number	Publication Date
HK1139399A1 true HK1139399A1 (xx)	2010-09-17

Family

ID=39620376

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HK10106008.5A HK1139399A1 (xx)	2007-02-28	2010-06-15

Country Status (27)

Country	Link
US (7)	US7943772B2 (xx)
EP (1)	EP2132204B1 (xx)
JP (2)	JP5512289B2 (xx)
KR (1)	KR101480530B1 (xx)
CN (1)	CN101616916B (xx)
AR (2)	AR065554A1 (xx)
AU (1)	AU2008219615B2 (xx)
BR (1)	BRPI0807974B8 (xx)
CA (1)	CA2678073C (xx)
CL (1)	CL2008000573A1 (xx)
CO (1)	CO6220856A2 (xx)
CY (1)	CY1115077T1 (xx)
DK (1)	DK2132204T3 (xx)
ES (1)	ES2402031T3 (xx)
HK (1)	HK1139399A1 (xx)
HR (1)	HRP20130193T1 (xx)
IL (1)	IL200131A (xx)
MX (1)	MX2009009141A (xx)
MY (1)	MY148318A (xx)
NZ (1)	NZ578871A (xx)
PL (1)	PL2132204T3 (xx)
PT (1)	PT2132204E (xx)
RU (1)	RU2458061C2 (xx)
SI (1)	SI2132204T1 (xx)
TW (1)	TWI409067B (xx)
WO (1)	WO2008106159A1 (xx)
ZA (1)	ZA200905832B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
MY145633A (en) *	2006-03-01	2012-03-15	Theravance Inc	8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
TWI409067B (zh)	2007-02-28	2013-09-21	Theravance Inc	８-氮雜雙環〔３．２．１〕辛烷化合物之結晶型
TWI415850B (zh) *	2007-07-20	2013-11-21	Theravance Inc	製備ｍｕ類鴉片受體拮抗劑之中間物的方法
US7902221B2 (en) *	2007-08-27	2011-03-08	Theravance, Inc.	Amidoalkyl-8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
ATE502939T1 (de) *	2007-08-27	2011-04-15	Theravance Inc	Disubstituierte alkyl-8-azabicycloä3.2.1üoktan- verbindungen als mu-opioid-rezeptorantagonisten
TWI423801B (zh)	2007-08-27	2014-01-21	Theravance Inc	作為μ類鴉片受體拮抗劑之８－氮雜雙環〔３．２．１〕辛基－２－羥基苯甲醯胺化合物
WO2009029253A1 (en) *	2007-08-27	2009-03-05	Theravance, Inc.	Heteroarylalkyl-8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
TW201118084A (en) *	2009-09-18	2011-06-01	Adolor Corp	The use of an opioid receptor antagonist for the treatment or prevention of gastrointestinal tract disorders
DK3277278T3 (da)	2015-04-02	2020-04-06	Theravance Biopharma R&D Ip Llc	Kombinationsdoseringsform af en my-opioid receptorantagonist og et opioid

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5159081A (en) *	1991-03-29	1992-10-27	Eli Lilly And Company	Intermediates of peripherally selective n-carbonyl-3,4,4-trisubstituted piperidine opioid antagonists
US6900228B1 (en) *	1998-03-10	2005-05-31	Research Triangle Institute	Opiate compounds, methods of making and methods of use
GB9810671D0 (en) *	1998-05-18	1998-07-15	Pfizer Ltd	Anti-pruritic agents
TWI244481B (en) *	1998-12-23	2005-12-01	Pfizer	3-azabicyclo[3.1.0]hexane derivatives useful in therapy
GB9912410D0 (en) *	1999-05-28	1999-07-28	Pfizer Ltd	Compounds useful in therapy
US6469030B2 (en) *	1999-11-29	2002-10-22	Adolor Corporation	Methods for the treatment and prevention of ileus
US6467084B1 (en) *	1999-12-16	2002-10-15	Emware, Inc.	Systems and methods for reprogramming an embedded device with program code using relocatable program code
IL151550A0 (en)	2000-03-03	2003-04-10	Ortho Mcneil Pharm Inc	3-(diarylmethylene)-8-azabicyclo [3.2.1] octane derivatives
US20020025948A1 (en) *	2000-06-23	2002-02-28	Banks Bernard Joseph	3-azabicyclo[3.1.0]hexane derivatives useful in therapy
UA75714C2 (en) *	2001-10-22	2006-05-15	Pfizer Prod Inc	3-azabicyclo [3.1.0] hexane derivatives as opioid receptor antagonists and pharmaceutical composition based thereon
US7381721B2 (en) *	2003-03-17	2008-06-03	Adolor Corporation	Substituted piperidine compounds
US7056930B2 (en) *	2003-04-14	2006-06-06	Pfizer Inc.	2-Azabicyclo[3.3.1]nonane derivatives
US20040204453A1 (en) *	2003-04-14	2004-10-14	Pfizer Inc	4-Phenyl-piperidine compounds and their use as modulators of opioid receptors
CA2522323C (en) *	2003-04-14	2009-09-15	Pfizer Products Inc.	3-azabicyclo[3.2.1]octane derivatives as opioid receptor ligands
EP1615920A1 (en)	2003-04-15	2006-01-18	Pfizer Products Inc.	3-benzhydrylidene-8-aza-bicyclo [3.2.1] octane derivatives with opioid receptor activity
US6992090B2 (en) *	2003-06-16	2006-01-31	Adolor Corporation	Substituted piperidine compounds and methods of their use
US7435822B2 (en)	2004-02-03	2008-10-14	Janssen Pharmaceutica N.V.	3-(diheteroarylmethylene)-8-azabicyclo[3.2.1]octane and 3-((aryl)(heteroaryl)methylene)-8-azabicyclo[3.2.1]octane derivatives
US7087749B2 (en) *	2004-03-11	2006-08-08	Adolor Corporation	Substituted piperidine compounds and methods of their use
MY145633A (en)	2006-03-01	2012-03-15	Theravance Inc	8-azabicyclo[3.2.1]octane compounds as mu opioid receptor antagonists
US20100284960A1 (en)	2006-11-07	2010-11-11	Nektar Therapeutics Al, Corporation	Dosage Forms and Co-Administration of Opioid Agonist and Opioid Antagonist
TWI409067B (zh) *	2007-02-28	2013-09-21	Theravance Inc	８-氮雜雙環〔３．２．１〕辛烷化合物之結晶型

2008
- 2008-02-15 TW TW097105472A patent/TWI409067B/zh active
- 2008-02-25 CL CL200800573A patent/CL2008000573A1/es unknown
- 2008-02-27 SI SI200830928T patent/SI2132204T1/sl unknown
- 2008-02-27 EP EP08726162A patent/EP2132204B1/en active Active
- 2008-02-27 MX MX2009009141A patent/MX2009009141A/es active IP Right Grant
- 2008-02-27 PL PL08726162T patent/PL2132204T3/pl unknown
- 2008-02-27 CN CN2008800059690A patent/CN101616916B/zh active Active
- 2008-02-27 US US12/072,534 patent/US7943772B2/en active Active
- 2008-02-27 WO PCT/US2008/002583 patent/WO2008106159A1/en active Application Filing
- 2008-02-27 AU AU2008219615A patent/AU2008219615B2/en not_active Ceased
- 2008-02-27 BR BRPI0807974A patent/BRPI0807974B8/pt not_active IP Right Cessation
- 2008-02-27 PT PT87261624T patent/PT2132204E/pt unknown
- 2008-02-27 MY MYPI20093401A patent/MY148318A/en unknown
- 2008-02-27 ES ES08726162T patent/ES2402031T3/es active Active
- 2008-02-27 JP JP2009551709A patent/JP5512289B2/ja active Active
- 2008-02-27 NZ NZ578871A patent/NZ578871A/en not_active IP Right Cessation
- 2008-02-27 CA CA2678073A patent/CA2678073C/en active Active
- 2008-02-27 RU RU2009135834/04A patent/RU2458061C2/ru active
- 2008-02-27 KR KR1020097020094A patent/KR101480530B1/ko active Active
- 2008-02-27 DK DK08726162.4T patent/DK2132204T3/da active
- 2008-02-28 AR ARP080100850A patent/AR065554A1/es not_active Application Discontinuation
2009
- 2009-07-29 IL IL200131A patent/IL200131A/en active IP Right Grant
- 2009-08-21 ZA ZA200905832A patent/ZA200905832B/xx unknown
- 2009-08-26 CO CO09089674A patent/CO6220856A2/es active IP Right Grant
2010
- 2010-06-15 HK HK10106008.5A patent/HK1139399A1/xx unknown
2011
- 2011-04-06 US US13/081,162 patent/US8247555B2/en active Active
2012
- 2012-07-17 US US13/550,781 patent/US8536335B2/en active Active
2013
- 2013-03-05 HR HRP20130193AT patent/HRP20130193T1/hr unknown
- 2013-04-08 CY CY20131100293T patent/CY1115077T1/el unknown
- 2013-05-10 JP JP2013099851A patent/JP2013151564A/ja not_active Withdrawn
- 2013-08-13 US US13/965,691 patent/US8816091B2/en active Active
2014
- 2014-07-16 US US14/333,003 patent/US9290491B2/en active Active
2016
- 2016-02-10 US US15/040,191 patent/US9949963B2/en active Active
2017
- 2017-07-31 AR ARP170102183A patent/AR109224A2/es unknown
2018
- 2018-03-13 US US15/919,678 patent/US10426766B2/en active Active

Also Published As

Publication number	Publication date
AU2008219615B2 (en)	2013-05-09
CY1115077T1 (el)	2016-12-14
CO6220856A2 (es)	2010-11-19
EP2132204B1 (en)	2013-01-23
EP2132204A1 (en)	2009-12-16
US8536335B2 (en)	2013-09-17
US20180200246A1 (en)	2018-07-19
MY148318A (en)	2013-03-29
ZA200905832B (en)	2010-05-26
TW200845984A (en)	2008-12-01
MX2009009141A (es)	2009-09-03
BRPI0807974A2 (pt)	2014-09-16
HRP20130193T1 (hr)	2013-03-31
JP5512289B2 (ja)	2014-06-04
IL200131A (en)	2013-03-24
US10426766B2 (en)	2019-10-01
SI2132204T1 (sl)	2013-05-31
BRPI0807974B1 (pt)	2020-11-24
ES2402031T3 (es)	2013-04-26
US20160287572A1 (en)	2016-10-06
CN101616916B (zh)	2011-10-12
TWI409067B (zh)	2013-09-21
KR101480530B1 (ko)	2015-01-08
IL200131A0 (en)	2010-04-15
CN101616916A (zh)	2009-12-30
US9949963B2 (en)	2018-04-24
PL2132204T3 (pl)	2013-06-28
CA2678073A1 (en)	2008-09-04
AR109224A2 (es)	2018-11-07
AU2008219615A1 (en)	2008-09-04
BRPI0807974B8 (pt)	2021-05-25
JP2013151564A (ja)	2013-08-08
CL2008000573A1 (es)	2008-05-16
US8816091B2 (en)	2014-08-26
US7943772B2 (en)	2011-05-17
US20130072515A1 (en)	2013-03-21
US20080207676A1 (en)	2008-08-28
WO2008106159A1 (en)	2008-09-04
US20150073014A1 (en)	2015-03-12
DK2132204T3 (da)	2013-04-29
US8247555B2 (en)	2012-08-21
NZ578871A (en)	2012-01-12
AR065554A1 (es)	2009-06-17
RU2009135834A (ru)	2011-04-10
US9290491B2 (en)	2016-03-22
RU2458061C2 (ru)	2012-08-10
CA2678073C (en)	2016-01-05
JP2010520198A (ja)	2010-06-10
US20140080856A1 (en)	2014-03-20
PT2132204E (pt)	2013-03-25
US20110184008A1 (en)	2011-07-28
KR20090115767A (ko)	2009-11-05

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