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GT200800218A - Compuestos organicos - Google Patents

Compuestos organicos

Info

Publication number
GT200800218A
GT200800218A GT200800218A GT200800218A GT200800218A GT 200800218 A GT200800218 A GT 200800218A GT 200800218 A GT200800218 A GT 200800218A GT 200800218 A GT200800218 A GT 200800218A GT 200800218 A GT200800218 A GT 200800218A
Authority
GT
Guatemala
Prior art keywords
organic compounds
compounds
useful
adenosine
allergic
Prior art date
Application number
GT200800218A
Other languages
English (en)
Inventor
Fairhurst Robin Alec
Taylor Roger John
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200800218A publication Critical patent/GT200800218A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

LA PRESENTE INVENCIÓN SE REFIERE A COMPUESTOS DE LA FÓRMULA GENERAL I EN LA QUE R1A,R2A,X1,X2,L,U1,R1B,U2, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS SON DE UTILIDAD EN LOS RECEPTORES DE ADENOSINA A2A POR LO QUE SON DE UTILIDAD EN CUADROS ALÉRGICOS E INFLAMATORIOS.
GT200800218A 2006-04-21 2008-10-17 Compuestos organicos GT200800218A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0607950.3A GB0607950D0 (en) 2006-04-21 2006-04-21 Organic compounds

Publications (1)

Publication Number Publication Date
GT200800218A true GT200800218A (es) 2008-12-15

Family

ID=36581047

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200800218A GT200800218A (es) 2006-04-21 2008-10-17 Compuestos organicos

Country Status (32)

Country Link
US (1) US8193164B2 (es)
EP (1) EP2018388B9 (es)
JP (1) JP2009534341A (es)
KR (1) KR20080112399A (es)
CN (1) CN101437829B (es)
AR (1) AR060606A1 (es)
AT (1) ATE502040T1 (es)
AU (1) AU2007241347A1 (es)
CA (1) CA2648037A1 (es)
CL (1) CL2007001132A1 (es)
CR (1) CR10328A (es)
CY (1) CY1111568T1 (es)
DE (1) DE602007013203D1 (es)
DK (1) DK2018388T3 (es)
EC (1) ECSP088837A (es)
ES (1) ES2363255T3 (es)
GB (1) GB0607950D0 (es)
GT (1) GT200800218A (es)
HR (1) HRP20110445T1 (es)
IL (1) IL194398A0 (es)
MA (1) MA30404B1 (es)
MX (1) MX2008013398A (es)
NO (1) NO20084456L (es)
PE (1) PE20071228A1 (es)
PL (1) PL2018388T3 (es)
PT (1) PT2018388E (es)
RU (1) RU2008145715A (es)
SI (1) SI2018388T1 (es)
TN (1) TNSN08409A1 (es)
TW (1) TW200813074A (es)
WO (1) WO2007121924A2 (es)
ZA (1) ZA200808103B (es)

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Also Published As

Publication number Publication date
TW200813074A (en) 2008-03-16
US8193164B2 (en) 2012-06-05
AR060606A1 (es) 2008-07-02
WO2007121924A2 (en) 2007-11-01
NO20084456L (no) 2008-12-09
CR10328A (es) 2008-11-18
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JP2009534341A (ja) 2009-09-24
CN101437829B (zh) 2012-03-21
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AU2007241347A1 (en) 2007-11-01
PE20071228A1 (es) 2008-01-24
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ATE502040T1 (de) 2011-04-15
IL194398A0 (en) 2009-08-03
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HRP20110445T1 (hr) 2011-07-31
MX2008013398A (es) 2008-11-04
US20100190784A1 (en) 2010-07-29
MA30404B1 (fr) 2009-05-04
DE602007013203D1 (de) 2011-04-28
EP2018388A2 (en) 2009-01-28
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ES2363255T3 (es) 2011-07-28
GB0607950D0 (en) 2006-05-31
ZA200808103B (en) 2009-07-29
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CL2007001132A1 (es) 2008-05-23
CY1111568T1 (el) 2015-10-07
KR20080112399A (ko) 2008-12-24
ECSP088837A (es) 2008-11-27
TNSN08409A1 (en) 2010-04-14
SI2018388T1 (sl) 2011-07-29

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