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FI971227L - Pyramidinylpyrazolderivat - Google Patents

Pyramidinylpyrazolderivat Download PDF

Info

Publication number
FI971227L
FI971227L FI971227A FI971227A FI971227L FI 971227 L FI971227 L FI 971227L FI 971227 A FI971227 A FI 971227A FI 971227 A FI971227 A FI 971227A FI 971227 L FI971227 L FI 971227L
Authority
FI
Finland
Prior art keywords
pyramidinylpyrazole
derivatives
pyramidinylpyrazole derivatives
Prior art date
Application number
FI971227A
Other languages
English (en)
Finnish (fi)
Other versions
FI971227A0 (sv
Inventor
Akio Ejima
Masamichi Sugimori
Ikuo Mitsui
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of FI971227A0 publication Critical patent/FI971227A0/sv
Publication of FI971227L publication Critical patent/FI971227L/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
FI971227A 1994-09-26 1997-03-24 Pyramidinylpyrazolderivat FI971227L (sv)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP22942294 1994-09-26
JP13501095 1995-06-01
PCT/JP1995/001934 WO1996010024A1 (en) 1994-09-26 1995-09-25 Pyrimidinylpyrazole derivative

Publications (2)

Publication Number Publication Date
FI971227A0 FI971227A0 (sv) 1997-03-24
FI971227L true FI971227L (sv) 1997-05-23

Family

ID=26468965

Family Applications (1)

Application Number Title Priority Date Filing Date
FI971227A FI971227L (sv) 1994-09-26 1997-03-24 Pyramidinylpyrazolderivat

Country Status (14)

Country Link
US (1) US5852019A (sv)
EP (1) EP0784055B1 (sv)
KR (1) KR100388568B1 (sv)
CN (1) CN1071754C (sv)
AT (1) ATE232528T1 (sv)
CA (1) CA2201110A1 (sv)
DE (2) DE69529619D1 (sv)
DK (1) DK0784055T3 (sv)
ES (1) ES2192584T3 (sv)
FI (1) FI971227L (sv)
HK (1) HK1001396A1 (sv)
NO (1) NO313196B1 (sv)
TW (1) TW312694B (sv)
WO (1) WO1996010024A1 (sv)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU724394B2 (en) * 1997-01-27 2000-09-21 Daiichi Pharmaceutical Co., Ltd. Pyrazole derivatives
US6169086B1 (en) 1997-01-27 2001-01-02 Daiichi Pharmaceutical Co., Ltd. Pyrazole derivatives
AU4800299A (en) * 1998-07-24 2000-02-14 Daiichi Pharmaceutical Co., Ltd. Pyrazole derivatives and salts thereof
JP4709388B2 (ja) * 1999-01-25 2011-06-22 全薬工業株式会社 複素環式化合物及びそれを有効成分とする抗腫瘍剤
JP3836436B2 (ja) * 2001-04-27 2006-10-25 全薬工業株式会社 複素環式化合物及びそれを有効成分とする抗腫瘍剤
WO2003011837A1 (en) * 2001-08-01 2003-02-13 Merck & Co., Inc. Tyrosine kinase inhibitors
FR2850379B1 (fr) * 2003-01-28 2006-11-17 Aventis Pharma Sa Produits n-aryl-heteroaromatiques, compositions les contenant et utilisation
JP2006516656A (ja) * 2003-01-28 2006-07-06 アヴェンティス ファーマ エス.エー. N−アリールヘテロ芳香族物質、それを含む組成物およびその用途
US20050130989A1 (en) * 2003-01-28 2005-06-16 Aventis Pharma S. A. N-arylheteroaromatic products compositions containing them and use thereof
WO2005028467A1 (en) * 2003-09-15 2005-03-31 Anadys Pharmaceuticals, Inc. Antibacterial 3,5-diaminopiperidine-substitute aromatic and heteroaromatic compounds
DK1741714T3 (da) 2004-03-31 2013-04-15 Zenyaku Kogyo Kk Heterocyklisk forbindelse og middel mod ondartet turmor, der indeholder denne som aktiv ingrediens
JP5089377B2 (ja) * 2005-03-11 2012-12-05 全薬工業株式会社 複素環式化合物を有効成分とする免疫抑制剤及び抗腫瘍剤
US20070244110A1 (en) * 2006-04-14 2007-10-18 Zenyaku Kogyo Kabushiki Kaisha Treatment of prostate cancer, melanoma or hepatic cancer
MX2009003821A (es) 2006-10-10 2009-05-25 Amgen Inc Compuestos de n-aril pirazol para usarse contra la diabetes.
EP3285581B1 (en) * 2015-03-26 2021-08-11 Merck Sharp & Dohme Corp. Pyrazolyl pyrimidinone compounds as pde2 inhibitors
CA3038280A1 (en) 2015-09-30 2017-04-06 Max-Planck-Gesellschaft Zur Forderung Der Wissenschaften E.V. - Generalverwaltung Heteroaryl derivatives as sepiapterin reductase inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3778433A (en) * 1969-04-18 1973-12-11 Sumitomo Chemical Co Process for producing benzodiazepine derivatives
JPS4842072A (sv) * 1971-09-29 1973-06-19
JPS61129129A (ja) * 1984-11-28 1986-06-17 Kureha Chem Ind Co Ltd 抗腫瘍剤
US5102893A (en) * 1986-07-07 1992-04-07 Warner-Lambert Company Trans-6-(2-(n-heteroaryl-3,5-disubstituted)pyrazol-4-yl)-ethyl- or ethenyl)tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis

Also Published As

Publication number Publication date
CA2201110A1 (en) 1996-04-04
CN1166833A (zh) 1997-12-03
DE69529619D1 (en) 2003-03-20
NO971384D0 (no) 1997-03-24
HK1001396A1 (en) 1998-06-19
TW312694B (sv) 1997-08-11
KR970706275A (ko) 1997-11-03
FI971227A0 (sv) 1997-03-24
EP0784055A4 (en) 1998-01-07
EP0784055A1 (en) 1997-07-16
CN1071754C (zh) 2001-09-26
NO313196B1 (no) 2002-08-26
WO1996010024A1 (en) 1996-04-04
ATE232528T1 (de) 2003-02-15
US5852019A (en) 1998-12-22
DE69529619T2 (de) 2003-12-18
DK0784055T3 (da) 2003-06-02
KR100388568B1 (ko) 2003-10-04
EP0784055B1 (en) 2003-02-12
ES2192584T3 (es) 2003-10-16
NO971384L (no) 1997-05-23
DE69529619T4 (de) 2005-01-27

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