FI954141L - Oksatsolokinolonijohdannaiset, niiden valmistus ja niiden käyttö terapiassa - Google Patents

Oksatsolokinolonijohdannaiset, niiden valmistus ja niiden käyttö terapiassa Download PDF

Info

Publication number: FI954141L
Authority: FI; Finland
Prior art keywords: oxazoloquinolone; therapy; derivatives; preparation; oxazoloquinolone derivatives
Prior art date: 1994-09-05

Application number

FI954141A

Other languages

English (en)

Swedish (sv)

Other versions

FI954141A0 (fi

FI110945B (fi

Inventor

Samir Jegham

Jean Jacques Koenig

Frederic Puech

Philippe Burnier

Lydia Zard

Original Assignee

Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-09-05

Filing date

1995-09-04

Publication date

1996-03-06

1995-09-04 Application filed by Synthelabo filed Critical Synthelabo

1995-09-04 Publication of FI954141A0 publication Critical patent/FI954141A0/fi

1996-03-06 Publication of FI954141L publication Critical patent/FI954141L/fi

2003-04-30 Application granted granted Critical

2003-04-30 Publication of FI110945B publication Critical patent/FI110945B/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Anesthesiology (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Micro-Organisms Or Cultivation Processes Thereof (AREA)
Quinoline Compounds (AREA)

FI954141A 1994-09-05 1995-09-04 Oksatsolokinolinonijohdannaisia, niiden valmistus ja niiden käyttö terapiassa FI110945B (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9410600A FR2724171B1 (fr)	1994-09-05	1994-09-05	Derives de 3,3a,4,5-tetrahydro-1h-oxazolo(3,4-a)quinolein-1-one, leur preparation et leur application en therapeutique
FR9410600		1994-09-05

Publications (3)

Publication Number	Publication Date
FI954141A0 FI954141A0 (fi)	1995-09-04
FI954141L true FI954141L (fi)	1996-03-06
FI110945B FI110945B (fi)	2003-04-30

Family

ID=9466686

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI954141A FI110945B (fi)	1994-09-05	1995-09-04	Oksatsolokinolinonijohdannaisia, niiden valmistus ja niiden käyttö terapiassa

Country Status (28)

Country	Link
US (1)	US5641785A (fi)
EP (1)	EP0699680B1 (fi)
JP (1)	JP4225585B2 (fi)
KR (1)	KR100392523B1 (fi)
CN (1)	CN1055472C (fi)
AT (1)	ATE190311T1 (fi)
AU (1)	AU687591B2 (fi)
CA (1)	CA2157427C (fi)
CZ (1)	CZ286128B6 (fi)
DE (1)	DE69515402T2 (fi)
DK (1)	DK0699680T3 (fi)
ES (1)	ES2145886T3 (fi)
FI (1)	FI110945B (fi)
FR (1)	FR2724171B1 (fi)
GR (1)	GR3033554T3 (fi)
HK (1)	HK1013652A1 (fi)
HU (1)	HU218587B (fi)
IL (1)	IL115276A (fi)
NO (1)	NO306617B1 (fi)
NZ (1)	NZ272920A (fi)
PL (1)	PL184412B1 (fi)
PT (1)	PT699680E (fi)
RU (1)	RU2141482C1 (fi)
SI (1)	SI0699680T1 (fi)
SK (1)	SK281867B6 (fi)
TW (1)	TW356467B (fi)
UA (1)	UA41916C2 (fi)
ZA (1)	ZA957414B (fi)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1078632A1 (en) *	1999-08-16	2001-02-28	Sanofi-Synthelabo	Use of monoamine oxydase inhibitors for the manufacture of drugs intended for the treatment of obesity
WO2005090309A1 (en) *	2004-03-12	2005-09-29	Wyeth	1,2-dihydroquinoline derivatives and method for using the same to treat hiv infection
WO2008112483A2 (en) *	2007-03-09	2008-09-18	Sanofi-Aventis	Substituted dihydro and tetrahydro oxazolopyrimidinones, preparation and use thereof
RU2366430C2 (ru)	2007-05-23	2009-09-10	Виктор Иванович Рощин	Ингибиторы моноаминооксидазы, лекарственное средство и фармацевтическая композиция
AR078171A1 (es)	2009-09-15	2011-10-19	Sanofi Aventis	Dihidrobenzocicloalquiloximetil-oxazolopirimidinonas sustituidas, preparacion y uso de las mismas
CN105949120B (zh) *	2016-05-27	2018-07-24	广东工业大学	一种四齿螯合型单喹啉衍生物及其制备方法和作为神经退行性疾病的金属离子调节剂的应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2624861B1 (fr) *	1987-12-21	1990-06-01	Delalande Sa	Carbamates tricycliques, leur procede de preparation et leur application en therapeutique
ES2013391A6 (es) *	1989-02-08	1990-05-01	Consejo Superior Investigacion	Procedimiento para la preparacion de derivados acetilenicos y alenicos de 2-aminometil -5-metoxiindoles.
JPH04295470A (ja) *	1991-03-22	1992-10-20	Wakamoto Pharmaceut Co Ltd	モノアミンオキシダーゼ−ｂ酵素阻害活性を有する１，２，４−オキサジアゾール誘導体及びその製造法

1994
- 1994-09-05 FR FR9410600A patent/FR2724171B1/fr not_active Expired - Lifetime
1995
- 1995-09-01 DE DE69515402T patent/DE69515402T2/de not_active Expired - Lifetime
- 1995-09-01 CA CA2157427A patent/CA2157427C/en not_active Expired - Lifetime
- 1995-09-01 DK DK95401989T patent/DK0699680T3/da active
- 1995-09-01 EP EP95401989A patent/EP0699680B1/fr not_active Expired - Lifetime
- 1995-09-01 AT AT95401989T patent/ATE190311T1/de active
- 1995-09-01 US US08/523,508 patent/US5641785A/en not_active Expired - Lifetime
- 1995-09-01 ES ES95401989T patent/ES2145886T3/es not_active Expired - Lifetime
- 1995-09-01 SI SI9530413T patent/SI0699680T1/xx unknown
- 1995-09-01 PT PT95401989T patent/PT699680E/pt unknown
- 1995-09-02 TW TW084109192A patent/TW356467B/zh not_active IP Right Cessation
- 1995-09-04 CN CN95117143A patent/CN1055472C/zh not_active Expired - Lifetime
- 1995-09-04 KR KR1019950028714A patent/KR100392523B1/ko not_active Expired - Lifetime
- 1995-09-04 CZ CZ19952262A patent/CZ286128B6/cs not_active IP Right Cessation
- 1995-09-04 SK SK1089-95A patent/SK281867B6/sk not_active IP Right Cessation
- 1995-09-04 RU RU95114741A patent/RU2141482C1/ru active
- 1995-09-04 ZA ZA957414A patent/ZA957414B/xx unknown
- 1995-09-04 UA UA95094019A patent/UA41916C2/uk unknown
- 1995-09-04 FI FI954141A patent/FI110945B/fi not_active IP Right Cessation
- 1995-09-04 NZ NZ272920A patent/NZ272920A/en not_active IP Right Cessation
- 1995-09-04 PL PL95310273A patent/PL184412B1/pl unknown
- 1995-09-04 AU AU30415/95A patent/AU687591B2/en not_active Expired
- 1995-09-04 HU HU9502578A patent/HU218587B/hu unknown
- 1995-09-04 JP JP22646295A patent/JP4225585B2/ja not_active Expired - Lifetime
- 1995-09-04 NO NO953458A patent/NO306617B1/no not_active IP Right Cessation
- 1995-09-12 IL IL11527695A patent/IL115276A/en not_active IP Right Cessation
1998
- 1998-12-23 HK HK98114972A patent/HK1013652A1/xx not_active IP Right Cessation
2000
- 2000-05-31 GR GR20000401246T patent/GR3033554T3/el unknown

Also Published As

Publication number	Publication date
JP4225585B2 (ja)	2009-02-18
CN1055472C (zh)	2000-08-16
US5641785A (en)	1997-06-24
AU3041595A (en)	1996-03-21
DK0699680T3 (da)	2000-08-21
PT699680E (pt)	2000-08-31
NO953458D0 (no)	1995-09-04
PL184412B1 (pl)	2002-10-31
ATE190311T1 (de)	2000-03-15
SK281867B6 (sk)	2001-08-06
EP0699680B1 (fr)	2000-03-08
TW356467B (en)	1999-04-21
RU2141482C1 (ru)	1999-11-20
UA41916C2 (uk)	2001-10-15
HU9502578D0 (en)	1995-11-28
ZA957414B (en)	1996-04-15
ES2145886T3 (es)	2000-07-16
NO306617B1 (no)	1999-11-29
NO953458L (no)	1996-03-06
AU687591B2 (en)	1998-02-26
FR2724171A1 (fr)	1996-03-08
CN1128763A (zh)	1996-08-14
DE69515402D1 (de)	2000-04-13
CA2157427C (en)	2010-06-01
CZ286128B6 (cs)	2000-01-12
IL115276A0 (en)	1996-01-19
FI954141A0 (fi)	1995-09-04
IL115276A (en)	1998-12-06
KR100392523B1 (ko)	2003-11-12
CA2157427A1 (en)	1996-03-06
HU218587B (hu)	2000-10-28
JPH0899881A (ja)	1996-04-16
NZ272920A (en)	1998-03-25
KR960010648A (ko)	1996-04-20
DE69515402T2 (de)	2000-10-19
SI0699680T1 (en)	2000-10-31
SK108995A3 (en)	1996-06-05
GR3033554T3 (en)	2000-09-29
CZ226295A3 (en)	1996-03-13
PL310273A1 (en)	1996-03-18
HK1013652A1 (en)	1999-09-03
EP0699680A1 (fr)	1996-03-06
FI110945B (fi)	2003-04-30
FR2724171B1 (fr)	1997-01-03
HUT73435A (en)	1996-07-29

Publication	Publication Date	Title
FI955235L (fi)	1996-05-03	Oksatsolidiinionijohdannaiset, niiden valmistus ja käyttö
FI944600A0 (fi)	1994-10-03	Imidatsol-4-yylipiperidiinijohdannaisia, niiden valmistus ja niiden käyttö terapiassa
FI964311L (fi)	1996-10-25	Bifunktionaalinen proteiini, valmistus ja käyttö
EE9700039A (et)	1997-08-15	Teraapias kasutatavad spiro-asabitsüklilised ühendid ja nende valmistamise protsess
FI953479A0 (fi)	1995-07-18	1-aryylipyrimidiinijohdannaiset ja niiden farmaseuttinen käyttö
EE9800459A (et)	1999-06-15	Spiro-piperidiini derivaadid ja nende kasutamine terapeutiliste toimeainetena
EE9600172A (et)	1997-06-16	Puriin-6-ooni derivaadid, nende valmistamismeetod, kasutamine ravimite valmistamiseks ja ravimid
EE200000037A (et)	2000-10-16	Atsüülpiperasinüülpürimidiinide derivaadid, nende valmistamine ja kasutamine ravimitena
FI955140L (fi)	1995-10-27	Uusia kinoksaliinidionijohdannaisia, niiden valmistus ja käyttö lääkkeissä
FI950458L (fi)	1995-08-04	N-(3-aminopropyyli)-N-fenyyli-5,6,7,8-tetrahydronaftalen-2-karboksamidijohdannaiset, niiden valmistus ja terapeuttinen käyttö
IL99612A0 (en)	1992-08-18	2-aminopyrimidine-4-carboxamide derivatives,their preparation and their use in therapy
EE9700288A (et)	1998-04-15	Asatsükloalkaani derivaadid, nende valmistamine ja kasutamine ravis
EE9900218A (et)	1999-12-15	1,4-diasabitsüklo[2.2.2]okt-2-üülmetüülbensoaadi derivaadid, nende valmistamine ja kasutamine raviks
EE04317B1 (et)	2004-06-15	4-okso-3,5-dihüdro-4H-püridasino[4.5-b]indool-1-etaanamiidi derivaadid, nende valmistamine ja kasutamine raviks
EE9800333A (et)	1999-04-15	Uued furaandiarüülmetülideeni derivaadid, nende valmistamise meetod ja kasutamine teraapias
FI940186A0 (fi)	1994-01-14	9H-imidatso/1,2-a/bentsimidatsoli-3-asetamidijohdannaisia, niiden valmistus ja niiden käyttö terapiassa
EE200000207A (et)	2001-04-16	8-asabitsüklo[3.2.1]oktaan-3-metaanamiini derivaadid, nende valmistamine ja terapeutiline kasutamine
EE9900135A (et)	1999-12-15	N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks
IL101617A0 (en)	1992-12-30	2-aminopyrimidine-4-carboxamide derivatives,their preparation and their application in therapy
FI954141L (fi)	1996-03-06	Oksatsolokinolonijohdannaiset, niiden valmistus ja niiden käyttö terapiassa
FI941963L (fi)	1994-10-29	Pyridiinijohdannaiset, niiden valmistus ja käyttö
FI956251A0 (fi)	1995-12-22	1-okso-2-(fenyylisulfonyyliamino)pentyylipiperidiinijohdannaiset, niiden valmistus ja terapeuttinen käyttö
FI955386L (fi)	1995-11-08	4-p-fluoribentsoyyli-1-piperidinyyli-propoksi-kromen-4-onijohdannaiset, niiden valmistus ja käyttö psykoosin ja skitsofrenian hoidossa
FI971317A (fi)	1997-03-27	Uusia heterosyklisiä, substituoituja imidatsolokinoksalinoneja, niiden valmistus ja käyttö
EE200000018A (et)	2000-08-15	6-pürrolidiin-2-üülpüridiinid, nende valmistamine ja terapeutiline kasutamine

Legal Events

Date	Code	Title	Description
2005-01-19	PC	Transfer of assignment of patent	Owner name: SANOFI-AVENTIS
2015-10-23	MA	Patent expired