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FI945957A - N-substituoidut 3-atsabisyklo/3.2.0/heptaanijohdannaiset neurolepteinä jne. - Google Patents

N-substituoidut 3-atsabisyklo/3.2.0/heptaanijohdannaiset neurolepteinä jne. Download PDF

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Publication number
FI945957A
FI945957A FI945957A FI945957A FI945957A FI 945957 A FI945957 A FI 945957A FI 945957 A FI945957 A FI 945957A FI 945957 A FI945957 A FI 945957A FI 945957 A FI945957 A FI 945957A
Authority
FI
Finland
Prior art keywords
pct
neuroleptics
azabicyclo
substituted
sec
Prior art date
Application number
FI945957A
Other languages
English (en)
Swedish (sv)
Other versions
FI108726B (fi
FI945957A0 (fi
Inventor
Gerd Steiner
Liliane Unger
Berthold Behl
Hans-Juergen Teschendorf
Rainer Munschauer
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of FI945957A publication Critical patent/FI945957A/fi
Publication of FI945957A0 publication Critical patent/FI945957A0/fi
Application granted granted Critical
Publication of FI108726B publication Critical patent/FI108726B/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI945957A 1992-06-19 1994-12-19 Menetelmä kaavan (I) mukaisten N-substituoitujen 3-atsabisyklo[3.2.0]heptaanijohdannaisten valmistamiseksi FI108726B (fi)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
DE4219974 1992-06-19
DE4219974 1992-06-19
DE4243287 1992-12-21
DE4243287A DE4243287A1 (de) 1992-06-19 1992-12-21 N-Substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
PCT/EP1993/001438 WO1994000458A1 (de) 1992-06-19 1993-06-08 N-substituierte 3-azabicyclo[3.2.0]heptanderivate als neuroleptika usw.
EP9301438 1993-06-08
CN93114691A CN1039996C (zh) 1992-06-19 1993-12-11 N-取代氮杂双环庚烷衍生物及其用途
CN93114691 1993-12-11

Publications (3)

Publication Number Publication Date
FI945957A true FI945957A (fi) 1994-12-19
FI945957A0 FI945957A0 (fi) 1994-12-19
FI108726B FI108726B (fi) 2002-03-15

Family

ID=36940125

Family Applications (1)

Application Number Title Priority Date Filing Date
FI945957A FI108726B (fi) 1992-06-19 1994-12-19 Menetelmä kaavan (I) mukaisten N-substituoitujen 3-atsabisyklo[3.2.0]heptaanijohdannaisten valmistamiseksi

Country Status (24)

Country Link
US (1) US5475105A (fi)
EP (1) EP0647231B1 (fi)
JP (1) JP3171258B2 (fi)
CN (2) CN1042133C (fi)
AT (1) ATE157366T1 (fi)
AU (1) AU671130B2 (fi)
BG (1) BG62350B2 (fi)
CA (1) CA2138289C (fi)
CZ (1) CZ288787B6 (fi)
DE (2) DE4243287A1 (fi)
DK (1) DK0647231T3 (fi)
ES (1) ES2107035T3 (fi)
FI (1) FI108726B (fi)
GR (1) GR3025095T3 (fi)
HU (1) HU218911B (fi)
IL (1) IL105989A (fi)
NO (1) NO305176B1 (fi)
NZ (1) NZ253121A (fi)
PH (1) PH30466A (fi)
RU (1) RU2135503C1 (fi)
SG (1) SG44782A1 (fi)
TW (1) TW408126B (fi)
WO (1) WO1994000458A1 (fi)
ZA (1) ZA934374B (fi)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4427648A1 (de) * 1994-08-04 1996-02-08 Basf Ag N-Stubstituierte 3-Azabicyclo[3,2,0,]heptan-Derivate, ihre Herstellung und Verwendung
DE4338396A1 (de) * 1993-11-10 1995-05-11 Basf Ag N-Substituierte Azabicycloalkan-Derivate, ihre Herstellung und Verwendung
DE4341403A1 (de) * 1993-12-04 1995-06-08 Basf Ag N-substituierte 3-Azabicycloalkan-Derivate, ihre Herstellung und Verwendung
DE4341402A1 (de) * 1993-12-04 1995-06-08 Basf Ag N-substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
DE4427647A1 (de) * 1994-08-04 1996-02-08 Basf Ag N-substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
US5929080A (en) * 1997-05-06 1999-07-27 American Cyanamid Company Method of treating polycystic kidney disease
US6323209B1 (en) 1997-11-06 2001-11-27 American Cyanamid Company Method of treating or inhibiting colonic polyps
DE19836406A1 (de) 1998-08-12 2000-02-17 Basf Ag N-Substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
US6458821B1 (en) * 1998-08-12 2002-10-01 Abbott Laboratories N-substituted azabicycloheptane derivatives, production and use thereof
DE19836404A1 (de) * 1998-08-12 2000-02-17 Basf Ag N-Substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung
DE19848521A1 (de) * 1998-10-21 2000-04-27 Basf Ag Verfahren zur Herstellung von (+)-exo-6-Phenyl-3-azabicyclo-[3.2.0]heptanen
DE19960074A1 (de) * 1999-12-13 2001-06-21 Basf Ag Neues Salz von Belaperidone und dessen Modifikationen
WO2002014295A1 (en) * 2000-08-16 2002-02-21 Elena Alexandrovna Izakson Thiazine derivatives having antibacterial and antiviral action
MX2007004358A (es) * 2004-10-14 2007-07-17 Abbott Gmbh & Co Kg Compuestos de azabicicloheptilo adecuados para tratar trastornos que responden a la modulacion del receptor de dopamina d3.
EP1874801A4 (en) * 2005-03-07 2009-03-25 Univ North Carolina MEANS OF INHIBITING RECA ACTIVITIES FOR THE CONTROL OF ANTIBIOTIC-SITES BACTERIAL PATHOGENESE
ES2610508T3 (es) 2006-11-22 2017-04-27 Clinical Research Associates, Llc Métodos para tratar el síndrome de Down, el síndrome del cromosoma X frágil y el autismo
RU2478099C2 (ru) * 2007-07-27 2013-03-27 Актелион Фармасьютиклз Лтд Производные 2-аза-бицикло[3.3.0]октана
AU2015308350B2 (en) 2014-08-29 2020-03-05 Tes Pharma S.R.L. Inhibitors of alpha-amino-beta-carboxymuconic acid semialdehyde decarboxylase
CN112010851A (zh) * 2020-06-30 2020-12-01 浙江美诺华药物化学有限公司 一种莫西沙星盐酸盐的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3155668A (en) * 1960-04-11 1964-11-03 Sterling Drug Inc 1-[3-, 2-, and 1-indolyl)-lower-alkyl]-tertiary amines and intermediates therefor
US3328390A (en) * 1962-02-27 1967-06-27 Tri Kem Corp Certain azabicycloalkane compounds
US4443451A (en) * 1981-07-15 1984-04-17 Janssen Pharmaceutica N.V. Bicyclic pyrimidin-5-one derivatives
US4540318A (en) * 1982-07-29 1985-09-10 Robert Bosch, Gmbh Rotary electrical tool with speed control, especially drill
DE3228303A1 (de) * 1982-07-29 1984-02-02 Robert Bosch Gmbh, 7000 Stuttgart Elektrische motorregelung
US4605655A (en) * 1984-03-06 1986-08-12 Bristol-Myers Company Antipsychotic 1-fluorophenylbutyl-4-(2-pyrimidinyl)piperazine derivatives
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles

Also Published As

Publication number Publication date
CZ323794A3 (en) 1995-05-17
CA2138289C (en) 2004-03-02
HUT71351A (en) 1995-11-28
PH30466A (en) 1997-05-28
ZA934374B (en) 1994-12-19
RU95105435A (ru) 1996-11-20
DK0647231T3 (da) 1997-09-29
DE4243287A1 (de) 1993-12-23
AU4323893A (en) 1994-01-24
IL105989A0 (en) 1993-10-20
CN1042133C (zh) 1999-02-17
NZ253121A (en) 1995-12-21
IL105989A (en) 1997-02-18
GR3025095T3 (en) 1998-01-30
CZ288787B6 (cs) 2001-09-12
EP0647231A1 (de) 1995-04-12
SG44782A1 (en) 1997-12-19
EP0647231B1 (de) 1997-08-27
DE59307217D1 (de) 1997-10-02
FI108726B (fi) 2002-03-15
NO944892L (no) 1995-02-13
HU218911B (hu) 2000-12-28
NO305176B1 (no) 1999-04-12
NO944892D0 (no) 1994-12-16
ES2107035T3 (es) 1997-11-16
ATE157366T1 (de) 1997-09-15
CN1039996C (zh) 1998-09-30
CA2138289A1 (en) 1994-01-06
CN1087341A (zh) 1994-06-01
CN1105358A (zh) 1995-07-19
FI945957A0 (fi) 1994-12-19
AU671130B2 (en) 1996-08-15
WO1994000458A1 (de) 1994-01-06
BG62350B2 (bg) 1999-08-31
TW408126B (en) 2000-10-11
RU2135503C1 (ru) 1999-08-27
JP3171258B2 (ja) 2001-05-28
JPH07507771A (ja) 1995-08-31
US5475105A (en) 1995-12-12

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