FI944169A - Menetelmä beta-fenyyli-isoseriinin ja sen analogien valmistamiseksi - Google Patents

Menetelmä beta-fenyyli-isoseriinin ja sen analogien valmistamiseksi Download PDF

Info

Publication number: FI944169A
Authority: FI; Finland
Prior art keywords: pct; general formula; phenylisoserine; beta; date sep
Prior art date: 1992-03-10

Application number

FI944169A

Other languages

English (en)

Swedish (sv)

Other versions

FI944169A0 (fi

FI113640B (fi

Inventor

Jean-Dominique Bourzat

Alain Commercon

Original Assignee

Rhone Poulenc Rorer Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-03-10

Filing date

1994-09-09

Publication date

1994-09-09

1994-09-09 Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa

1994-09-09 Publication of FI944169A0 publication Critical patent/FI944169A0/fi

1994-09-09 Publication of FI944169A publication Critical patent/FI944169A/fi

2004-05-31 Application granted granted Critical

2004-05-31 Publication of FI113640B publication Critical patent/FI113640B/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
- C07C227/18—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/22—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from lactams, cyclic ketones or cyclic oximes, e.g. by reactions involving Beckmann rearrangement
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Epoxy Compounds (AREA)
Steroid Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

FI944169A 1992-03-10 1994-09-09 Menetelmä beta-fenyyli-isoseriinin ja sen analogien valmistamiseksi, menetelmässä käytettävän lähtöaineen valmistus ja lähtöaine FI113640B (fi)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
FR9202821A FR2688499B1 (fr)	1992-03-10	1992-03-10	Procede de preparation de la beta-phenylisoserine et de ses analogues.
FR9202821		1992-03-10
FR9300224		1993-03-08
PCT/FR1993/000224 WO1993017997A1 (fr)	1992-03-10	1993-03-08	PROCEDE DE PREPARATION DE LA β-PHENYLISOSERINE ET DE SES ANALOGUES

Publications (3)

Publication Number	Publication Date
FI944169A0 FI944169A0 (fi)	1994-09-09
FI944169A true FI944169A (fi)	1994-09-09
FI113640B FI113640B (fi)	2004-05-31

Family

ID=9427518

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI944169A FI113640B (fi)	1992-03-10	1994-09-09	Menetelmä beta-fenyyli-isoseriinin ja sen analogien valmistamiseksi, menetelmässä käytettävän lähtöaineen valmistus ja lähtöaine

Country Status (25)

Country	Link
US (2)	US5608102A (fi)
EP (1)	EP0630365B1 (fi)
JP (1)	JP3278768B2 (fi)
KR (1)	KR100272650B1 (fi)
AT (1)	ATE159512T1 (fi)
AU (1)	AU667886B2 (fi)
CA (1)	CA2130333C (fi)
CZ (1)	CZ283613B6 (fi)
DE (1)	DE69314779T2 (fi)
DK (1)	DK0630365T3 (fi)
ES (1)	ES2109509T3 (fi)
FI (1)	FI113640B (fi)
FR (1)	FR2688499B1 (fi)
GE (1)	GEP19981430B (fi)
GR (1)	GR3025117T3 (fi)
HU (1)	HU213621B (fi)
MX (1)	MX9301268A (fi)
NO (1)	NO304515B1 (fi)
NZ (1)	NZ249899A (fi)
PL (1)	PL171551B1 (fi)
RU (1)	RU2103258C1 (fi)
SK (1)	SK281297B6 (fi)
TW (1)	TW252971B (fi)
WO (1)	WO1993017997A1 (fi)
ZA (1)	ZA931677B (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE69507702T2 (de) *	1994-07-26	1999-08-26	Indena S.P.A.	Semisynthetisch taxal derivate mit antitumor wirkung
US6765015B2 (en) *	1995-12-13	2004-07-20	Xechem International, Inc.	Halogenated paclitaxel derivatives
US6111144A (en)	1997-08-21	2000-08-29	Florida State University	Method for the synthesis of a taxane intermediate
AU1701699A (en) *	1997-11-19	1999-06-07	Xechem International, Inc.	Halogenated paclitaxel derivatives
ITMI991483A1 (it) *	1999-07-06	2001-01-06	Indena Spa	Derivati tassanici e procedimenti per la loro preparazione
EP1229934B1 (en)	1999-10-01	2014-03-05	Immunogen, Inc.	Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents
JP2002080435A (ja) *	2000-06-26	2002-03-19	Kanegafuchi Chem Ind Co Ltd	３−アミノ−２−ヒドロキシプロピオン酸誘導体の製造法
JP4142444B2 (ja)	2001-03-07	2008-09-03	第一三共株式会社	２−アゼチジノン誘導体の製造方法
PL1961735T3 (pl) *	2007-02-22	2010-04-30	Indena Spa	Sposób wytwarzania octanu metylowego estru (2r,3s)-3-fenyloizoseryny
EP2080764B1 (en)	2008-01-18	2012-08-22	INDENA S.p.A.	Solid forms of ortataxel
CN102408356A (zh) *	2011-09-28	2012-04-11	北京东方协和医药生物技术有限公司	一种多西他赛手性侧链中间体的制备方法
ES2896882T3 (es) *	2014-02-03	2022-02-28	Quadriga Biosciences Inc	Beta-aminoácidos beta sustituidos y análogos como agentes quimioterapéuticos
CN111100026A (zh) *	2019-12-30	2020-05-05	重庆市碚圣医药科技股份有限公司	一种紫杉醇恶唑环侧链中间体的制备方法
CN112574134A (zh) *	2020-12-30	2021-03-30	重庆市碚圣医药科技股份有限公司	一种多西紫杉醇侧链的合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2629819B1 (fr) *	1988-04-06	1990-11-16	Rhone Poulenc Sante	Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii
IT1231751B (it) *	1989-04-12	1991-12-21	Sigma Tau Ind Farmaceuti	Procedimento per la produzione di r(+) amminocarnitina e s(-) amminocarnitina
US5175315A (en) *	1989-05-31	1992-12-29	Florida State University	Method for preparation of taxol using β-lactam
US5304670A (en) *	1989-08-23	1994-04-19	Centre National De La Recherche Scientifique	Process for the enantioselective preparation of phenylisoserine derivatives
FR2658510B1 (fr) *	1990-02-21	1992-04-30	Rhone Poulenc Sante	Nouveau derive de la beta-phenylisoserine, sa preparation et son emploi.
US5294737A (en) *	1992-02-27	1994-03-15	The Research Foundation State University Of New York	Process for the production of chiral hydroxy-β-lactams and hydroxyamino acids derived therefrom

1992
- 1992-03-10 FR FR9202821A patent/FR2688499B1/fr not_active Expired - Fee Related
1993
- 1993-03-08 DK DK93918746.4T patent/DK0630365T3/da active
- 1993-03-08 CZ CZ942185A patent/CZ283613B6/cs not_active IP Right Cessation
- 1993-03-08 JP JP51539493A patent/JP3278768B2/ja not_active Expired - Lifetime
- 1993-03-08 ES ES93918746T patent/ES2109509T3/es not_active Expired - Lifetime
- 1993-03-08 KR KR1019940703156A patent/KR100272650B1/ko not_active IP Right Cessation
- 1993-03-08 MX MX9301268A patent/MX9301268A/es unknown
- 1993-03-08 WO PCT/FR1993/000224 patent/WO1993017997A1/fr active IP Right Grant
- 1993-03-08 US US08/295,677 patent/US5608102A/en not_active Expired - Lifetime
- 1993-03-08 HU HU9402590A patent/HU213621B/hu unknown
- 1993-03-08 GE GEAP19932472A patent/GEP19981430B/en unknown
- 1993-03-08 PL PL93305059A patent/PL171551B1/pl unknown
- 1993-03-08 RU RU94045799A patent/RU2103258C1/ru active
- 1993-03-08 NZ NZ249899A patent/NZ249899A/en not_active IP Right Cessation
- 1993-03-08 DE DE69314779T patent/DE69314779T2/de not_active Expired - Lifetime
- 1993-03-08 AT AT93918746T patent/ATE159512T1/de active
- 1993-03-08 EP EP93918746A patent/EP0630365B1/fr not_active Expired - Lifetime
- 1993-03-08 AU AU37557/93A patent/AU667886B2/en not_active Expired
- 1993-03-08 CA CA002130333A patent/CA2130333C/fr not_active Expired - Lifetime
- 1993-03-08 SK SK1085-94A patent/SK281297B6/sk not_active IP Right Cessation
- 1993-03-09 ZA ZA931677A patent/ZA931677B/xx unknown
- 1993-03-10 TW TW082101775A patent/TW252971B/zh not_active IP Right Cessation
1994
- 1994-09-05 NO NO943280A patent/NO304515B1/no not_active IP Right Cessation
- 1994-09-09 FI FI944169A patent/FI113640B/fi not_active IP Right Cessation
1996
- 1996-08-23 US US08/697,420 patent/US5763628A/en not_active Expired - Lifetime
1997
- 1997-10-23 GR GR970401615T patent/GR3025117T3/el unknown

Also Published As

Publication number	Publication date
KR100272650B1 (ko)	2000-11-15
HUT68540A (en)	1995-06-28
WO1993017997A1 (fr)	1993-09-16
RU94045799A (ru)	1996-07-20
NZ249899A (en)	1996-01-26
SK108594A3 (en)	1995-02-08
DE69314779D1 (de)	1997-11-27
CZ283613B6 (cs)	1998-05-13
GEP19981430B (en)	1998-10-30
FI944169A0 (fi)	1994-09-09
JPH07504425A (ja)	1995-05-18
AU667886B2 (en)	1996-04-18
CA2130333C (fr)	2002-11-26
EP0630365A1 (fr)	1994-12-28
FI113640B (fi)	2004-05-31
NO943280D0 (no)	1994-09-05
AU3755793A (en)	1993-10-05
TW252971B (fi)	1995-08-01
DK0630365T3 (da)	1998-03-02
KR950700234A (ko)	1995-01-16
HU213621B (en)	1997-08-28
GR3025117T3 (en)	1998-01-30
EP0630365B1 (fr)	1997-10-22
SK281297B6 (sk)	2001-02-12
CZ218594A3 (en)	1995-11-15
FR2688499B1 (fr)	1994-05-06
ATE159512T1 (de)	1997-11-15
HU9402590D0 (en)	1994-11-28
NO304515B1 (no)	1999-01-04
CA2130333A1 (fr)	1993-09-16
MX9301268A (es)	1993-09-01
PL171551B1 (pl)	1997-05-30
ES2109509T3 (es)	1998-01-16
RU2103258C1 (ru)	1998-01-27
NO943280L (no)	1994-09-05
ZA931677B (en)	1993-10-06
US5608102A (en)	1997-03-04
DE69314779T2 (de)	1998-02-26
US5763628A (en)	1998-06-09
JP3278768B2 (ja)	2002-04-30
FR2688499A1 (fr)	1993-09-17

Publication	Publication Date	Title
FI944169A (fi)	1994-09-09	Menetelmä beta-fenyyli-isoseriinin ja sen analogien valmistamiseksi
EP0339237A3 (en)	1991-01-09	Phenol substituted gem-diphosphonate derivatives, process for their preparation and pharmaceutical compositions containing them
PL293795A1 (en)	1993-03-08	Method of obtaining cyclic urea derivatives
ES2010114A6 (es)	1989-10-16	Procedimiento de preparacion de derivados de los acidos 1,4-dihidro-4-oxoquinolein-3-carboxilicos.
FI954898A0 (fi)	1995-10-13	Vesiliukoiset kamptotesiinijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö kasvaintenvastaisina aineina
AU699480B2 (en)	1998-12-03	2,2-Dichloroalkane carboxylic acids, processes for their production and pharmaceutical agents containing these
FI870589A0 (fi)	1987-02-12	Ny farmaceutisk sammansaettning och foerfarande foer framstaellning av den.
ATE165827T1 (de)	1998-05-15	Herstellung von n-acetylneuraminsäure-derivaten
ZA952771B (en)	1996-10-04	Novel compound
ATE246515T1 (de)	2003-08-15	Verfahren zur herstellung von oralen dosierungsformulierungen enthaltend diclofenac
AU5644296A (en)	1996-11-21	Novel heterocyclic chemistry
BR9610175A (pt)	1998-08-11	Composto processo de preparação do composto composição farmacêutica e utilização do composto
HUT53103A (en)	1990-09-28	Process for the preparation of new 20,21-dinor-eburnamenine derivatives, new intermediates thereof, as well as pharmaceutical compositions containing said compounds as active ingredients
BR9306870A (pt)	1998-12-08	Derivados farmacologicamente ativos de (aminometila terciária) - benzenometanol
PT1214315E (pt)	2003-09-30	Esteres derivados do acido 1,4-di-hidropiridina-5-carboxilico e metodo para a sua preparacao
ZA937317B (en)	1994-04-22	Process for the stereoselective preparation of a beta-phenylisoserine derivative and its use for the preparation of taxane derivatives
IT1247508B (it)	1994-12-17	Composizioni farmaceutiche contenenti l'estere 4-(2 metilamminoetil)- 1,2- fenilenicodell`acido 2-metilpropanoico per il trattamento della neurootticopatia glaucomatosa

Legal Events

Date	Code	Title	Description
2013-04-10	MA	Patent expired