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FI940733A - Polymeerisitoutuneet paklitakselijohdannaiset - Google Patents

Polymeerisitoutuneet paklitakselijohdannaiset Download PDF

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Publication number
FI940733A
FI940733A FI940733A FI940733A FI940733A FI 940733 A FI940733 A FI 940733A FI 940733 A FI940733 A FI 940733A FI 940733 A FI940733 A FI 940733A FI 940733 A FI940733 A FI 940733A
Authority
FI
Finland
Prior art keywords
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gly
leu
ala
beta
Prior art date
Application number
FI940733A
Other languages
English (en)
Swedish (sv)
Other versions
FI940733A0 (fi
Inventor
Nicola Mongelli
Francesco Angelucci
Enrico Pesenti
Antonino Suarato
Giovanni Biasoli
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of FI940733A0 publication Critical patent/FI940733A0/fi
Publication of FI940733A publication Critical patent/FI940733A/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/58—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. poly[meth]acrylate, polyacrylamide, polystyrene, polyvinylpyrrolidone, polyvinylalcohol or polystyrene sulfonic acid resin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Epoxy Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Analysing Materials By The Use Of Radiation (AREA)
FI940733A 1992-06-19 1994-02-16 Polymeerisitoutuneet paklitakselijohdannaiset FI940733A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929213077A GB9213077D0 (en) 1992-06-19 1992-06-19 Polymerbound taxol derivatives
PCT/EP1993/001433 WO1994000156A1 (en) 1992-06-19 1993-06-07 Polymer-bound paclitaxel derivatives

Publications (2)

Publication Number Publication Date
FI940733A0 FI940733A0 (fi) 1994-02-16
FI940733A true FI940733A (fi) 1994-02-16

Family

ID=10717411

Family Applications (1)

Application Number Title Priority Date Filing Date
FI940733A FI940733A (fi) 1992-06-19 1994-02-16 Polymeerisitoutuneet paklitakselijohdannaiset

Country Status (25)

Country Link
US (4) US5362831A (fi)
EP (1) EP0600062B1 (fi)
JP (1) JP3693340B2 (fi)
KR (1) KR100281606B1 (fi)
CN (1) CN1041281C (fi)
AT (1) ATE205725T1 (fi)
AU (2) AU659750B2 (fi)
CA (1) CA2112482A1 (fi)
CZ (1) CZ62094A3 (fi)
DE (1) DE69330776T2 (fi)
ES (1) ES2164663T3 (fi)
FI (1) FI940733A (fi)
GB (1) GB9213077D0 (fi)
HU (2) HUT67914A (fi)
IL (1) IL106023A (fi)
MX (1) MX9303598A (fi)
MY (1) MY109213A (fi)
NZ (1) NZ253116A (fi)
PL (1) PL173898B1 (fi)
RU (1) RU2130462C1 (fi)
SG (1) SG49248A1 (fi)
TW (1) TW266201B (fi)
UA (1) UA39926C2 (fi)
WO (1) WO1994000156A1 (fi)
ZA (1) ZA934388B (fi)

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* Cited by examiner, † Cited by third party
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HU9400800D0 (en) 1994-06-28
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KR100281606B1 (ko) 2001-02-15
CN1041281C (zh) 1998-12-23
AU1628295A (en) 1995-06-22
NZ253116A (en) 1996-05-28
MX9303598A (es) 1994-01-31
US5719265A (en) 1998-02-17
ATE205725T1 (de) 2001-10-15
US5569720A (en) 1996-10-29
EP0600062A1 (en) 1994-06-08
DE69330776T2 (de) 2002-07-04
SG49248A1 (en) 1998-05-18
HUT67914A (en) 1995-05-29
PL302437A1 (en) 1994-07-25
WO1994000156A1 (en) 1994-01-06
MY109213A (en) 1996-12-31
HU211291A9 (en) 1995-11-28
ZA934388B (en) 1994-08-29
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GB9213077D0 (en) 1992-08-05
US5362831A (en) 1994-11-08
CZ62094A3 (en) 1994-07-13
TW266201B (fi) 1995-12-21
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EP0600062B1 (en) 2001-09-19
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CN1079971A (zh) 1993-12-29
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UA39926C2 (uk) 2001-07-16
CA2112482A1 (en) 1994-01-06
RU2130462C1 (ru) 1999-05-20
AU659750B2 (en) 1995-05-25
IL106023A (en) 1998-03-10
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AU671247B2 (en) 1996-08-15

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