FI873290A0 - Foerfarande foer syntetisering av penem. - Google Patents
Foerfarande foer syntetisering av penem.Info
- Publication number
- FI873290A0 FI873290A0 FI873290A FI873290A FI873290A0 FI 873290 A0 FI873290 A0 FI 873290A0 FI 873290 A FI873290 A FI 873290A FI 873290 A FI873290 A FI 873290A FI 873290 A0 FI873290 A0 FI 873290A0
- Authority
- FI
- Finland
- Prior art keywords
- syntetisering
- penem
- foerfarande foer
- foerfarande
- foer
- Prior art date
Links
- HHXMXAQDOUCLDN-RXMQYKEDSA-N penem Chemical compound S1C=CN2C(=O)C[C@H]21 HHXMXAQDOUCLDN-RXMQYKEDSA-N 0.000 title 1
- JYLUAHUNORBOAL-UHFFFAOYSA-N 8-oxo-4,5-dithia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid Chemical class OC(=O)C1=CSSC2CC(=O)N12 JYLUAHUNORBOAL-UHFFFAOYSA-N 0.000 abstract 1
- MNFORVFSTILPAW-UHFFFAOYSA-N azetidin-2-one Chemical class O=C1CCN1 MNFORVFSTILPAW-UHFFFAOYSA-N 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 150000002961 penems Chemical class 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Electric Double-Layer Capacitors Or The Like (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Inks, Pencil-Leads, Or Crayons (AREA)
- Paints Or Removers (AREA)
- Control Of El Displays (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Pens And Brushes (AREA)
- Steroid Compounds (AREA)
- Mechanical Pencils And Projecting And Retracting Systems Therefor, And Multi-System Writing Instruments (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US89149386 | 1986-07-29 | ||
| US06/891,493 US4695626A (en) | 1986-07-29 | 1986-07-29 | 1-aza-4,5-dithiabicyclo [4.2.0] oct-2-en-8-one-2 carboxylate esters |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| FI873290A0 true FI873290A0 (fi) | 1987-07-28 |
| FI873290A FI873290A (fi) | 1988-01-30 |
| FI87651B FI87651B (fi) | 1992-10-30 |
| FI87651C FI87651C (fi) | 1993-02-10 |
Family
ID=25398284
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI873290A FI87651C (fi) | 1986-07-29 | 1987-07-28 | Foerfarande foer framstaellning av penemer samt mellanprodukter |
Country Status (18)
| Country | Link |
|---|---|
| US (2) | US4695626A (fi) |
| EP (1) | EP0255307B1 (fi) |
| JP (1) | JPH0737462B2 (fi) |
| KR (1) | KR890004581B1 (fi) |
| AT (1) | ATE70064T1 (fi) |
| AU (1) | AU583465B2 (fi) |
| CA (1) | CA1285275C (fi) |
| DE (1) | DE3774954D1 (fi) |
| DK (1) | DK170169B1 (fi) |
| ES (1) | ES2038665T3 (fi) |
| FI (1) | FI87651C (fi) |
| GR (1) | GR3003660T3 (fi) |
| HU (1) | HU198068B (fi) |
| IE (1) | IE60029B1 (fi) |
| IL (1) | IL83304A (fi) |
| NZ (1) | NZ221201A (fi) |
| PT (1) | PT85407B (fi) |
| ZA (1) | ZA875541B (fi) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU563157B2 (en) * | 1982-12-08 | 1987-07-02 | Farmitalia Carlo Erba S.P.A. | 2-thiacephems and (5r) penems derivatives |
| US4782145A (en) * | 1986-06-02 | 1988-11-01 | Pfizer Inc. | Process for penem derivatives |
| US4751297A (en) * | 1987-03-20 | 1988-06-14 | Pfizer Inc. | Method for preparation of azetidinone-1-oxoacetate by oxidation of the corresponding 2-hydroxyacetate |
| US5191077A (en) * | 1987-05-11 | 1993-03-02 | Pfizer Inc. | Diastereomeric 5R,6S-6-(1R-hydroxyethyl)-2-(cis-1-oxo-3-thiolanylthio)-2-penem-3-carboxylic acids |
| US5013729A (en) * | 1987-05-11 | 1991-05-07 | Pfizer Inc. | Diastereomeric 5R,6S-6-(1R-hydroxyethyl)-2-(cis-1-oxo-3-thiolanylthio)-2-penem-3-carboxylic acids |
| DE19512050A1 (de) * | 1995-03-31 | 1996-10-02 | Gimmy Lindomare Dr | Vorrichtung zum Sichern von Schrauben vor unbefugtem Zugriff |
| WO2005113592A2 (en) * | 2004-05-19 | 2005-12-01 | Maxygen, Inc. | Interferon-alpha polypeptides and conjugates |
| JP2010536385A (ja) | 2007-08-24 | 2010-12-02 | コデクシス， インコーポレイテッド | （ｒ）−３−ヒドロキシチオランの立体選択的生成のための改善されたケトレダクターゼポリペプチド |
| EP3523309B1 (en) * | 2016-10-10 | 2024-04-17 | The Johns Hopkins University | Antibacterial agents against d,d- and l,d-transpeptidases |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH541577A (de) * | 1970-11-03 | 1973-09-15 | Ciba Geigy Ag | Verfahren zur Herstellung thiaheterocyclischer Verbindungen |
| EP0176064A1 (en) * | 1980-11-06 | 1986-04-02 | Hoechst Uk Limited | Intermediates for the production of 7-oxo-4-thia-1-aza[3,2,0]heptane and 7-oxo-4-thia-1-aza[3,2,0]hept-2-ene derivatives |
| JPS57176988A (en) * | 1981-04-09 | 1982-10-30 | Sankyo Co Ltd | Penam-3-carboxylic acid derivative and its preparation |
| GB2131432B (en) * | 1982-12-08 | 1986-10-15 | Erba Farmitalia | Preparation of (5r)-penem derivatives |
| AU563157B2 (en) * | 1982-12-08 | 1987-07-02 | Farmitalia Carlo Erba S.P.A. | 2-thiacephems and (5r) penems derivatives |
| EP0115308A3 (en) * | 1983-01-25 | 1984-10-10 | Merck & Co. Inc. | 2-unsaturated alkylthio-pen-2-em-3-carboxylic acids and process for preparing substituted 2-thioxopenams and 2-substituted thiopenems |
| DE3464610D1 (de) * | 1983-06-21 | 1987-08-13 | Pfizer | 2-alkylthiopenem derivatives |
| EP0132101A1 (en) * | 1983-07-14 | 1985-01-23 | Pfizer Inc. | 2-Heterocycloalkylthiopenem derivatives |
-
1986
- 1986-07-29 US US06/891,493 patent/US4695626A/en not_active Expired - Fee Related
-
1987
- 1987-06-16 US US07/062,798 patent/US4782146A/en not_active Expired - Lifetime
- 1987-07-23 IL IL83304A patent/IL83304A/xx not_active IP Right Cessation
- 1987-07-24 EP EP87306586A patent/EP0255307B1/en not_active Expired - Lifetime
- 1987-07-24 AT AT87306586T patent/ATE70064T1/de not_active IP Right Cessation
- 1987-07-24 ES ES198787306586T patent/ES2038665T3/es not_active Expired - Lifetime
- 1987-07-24 DE DE8787306586T patent/DE3774954D1/de not_active Expired - Lifetime
- 1987-07-27 PT PT85407A patent/PT85407B/pt unknown
- 1987-07-27 CA CA000543040A patent/CA1285275C/en not_active Expired - Lifetime
- 1987-07-27 NZ NZ221201A patent/NZ221201A/xx unknown
- 1987-07-28 ZA ZA875541A patent/ZA875541B/xx unknown
- 1987-07-28 JP JP62186763A patent/JPH0737462B2/ja not_active Expired - Lifetime
- 1987-07-28 HU HU873463A patent/HU198068B/hu not_active IP Right Cessation
- 1987-07-28 AU AU76187/87A patent/AU583465B2/en not_active Ceased
- 1987-07-28 FI FI873290A patent/FI87651C/fi not_active IP Right Cessation
- 1987-07-28 DK DK392287A patent/DK170169B1/da not_active IP Right Cessation
- 1987-07-28 IE IE204687A patent/IE60029B1/en not_active IP Right Cessation
- 1987-07-28 KR KR1019870008186A patent/KR890004581B1/ko not_active IP Right Cessation
-
1992
- 1992-01-27 GR GR920400089T patent/GR3003660T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA875541B (en) | 1989-03-29 |
| US4695626A (en) | 1987-09-22 |
| NZ221201A (en) | 1990-06-26 |
| IE872046L (en) | 1988-01-29 |
| EP0255307A1 (en) | 1988-02-03 |
| US4782146A (en) | 1988-11-01 |
| IL83304A0 (en) | 1987-12-31 |
| DK170169B1 (da) | 1995-06-06 |
| AU583465B2 (en) | 1989-04-27 |
| CA1285275C (en) | 1991-06-25 |
| DE3774954D1 (de) | 1992-01-16 |
| AU7618787A (en) | 1988-02-04 |
| KR880001668A (ko) | 1988-04-26 |
| HU198068B (en) | 1989-07-28 |
| IE60029B1 (en) | 1994-05-18 |
| HUT45067A (en) | 1988-05-30 |
| IL83304A (en) | 1992-06-21 |
| KR890004581B1 (ko) | 1989-11-16 |
| DK392287A (da) | 1988-01-30 |
| GR3003660T3 (fi) | 1993-03-16 |
| ES2038665T3 (es) | 1993-08-01 |
| PT85407B (pt) | 1990-04-30 |
| JPH0737462B2 (ja) | 1995-04-26 |
| FI873290A (fi) | 1988-01-30 |
| PT85407A (en) | 1987-08-01 |
| JPS6341481A (ja) | 1988-02-22 |
| DK392287D0 (da) | 1987-07-28 |
| FI87651C (fi) | 1993-02-10 |
| ATE70064T1 (de) | 1991-12-15 |
| EP0255307B1 (en) | 1991-12-04 |
| FI87651B (fi) | 1992-10-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application lapsed | ||
| MM | Patent lapsed | ||
| MM | Patent lapsed |
Owner name: PFIZER INC. |