FI781025A - 2'-hydroxi-2-(5-isoxazolylmetyl)-6 7-bentzomorfaner deras syraadditionssalter och dessa innehaollande laekemedel - Google Patents

2'-hydroxi-2-(5-isoxazolylmetyl)-6 7-bentzomorfaner deras syraadditionssalter och dessa innehaollande laekemedel

Info

Publication number: FI781025A
Authority: FI; Finland
Prior art keywords: bentzomorfaner; hydroxi; isoxazolylmethyl; ceiling model; dessa innehaollande
Prior art date: 1977-04-15

Application number

FI781025A

Other languages

English (en)

Other versions

FI63399C (fi

FI63399B (fi

Inventor

Herbert Merz

Klaus Stockhaus

Original Assignee

Boehringer Sohn Ingelheim

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-04-15

Filing date

1978-04-04

Publication date

1978-10-16

1978-04-04 Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim

1978-10-16 Publication of FI781025A publication Critical patent/FI781025A/fi

1983-02-28 Application granted granted Critical

1983-02-28 Publication of FI63399B publication Critical patent/FI63399B/fi

1983-06-10 Publication of FI63399C publication Critical patent/FI63399C/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Organic Chemistry (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Dermatology (AREA)
Molecular Biology (AREA)
Biophysics (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Pain & Pain Management (AREA)
General Chemical & Material Sciences (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Plural Heterocyclic Compounds (AREA)

FI781025A 1977-04-15 1978-04-04 Foerfarande foer framstaellning av farmakologiskt vaerdefulla 2'-hydroxi-2-(5-isoxazolylmetyl)-6,7-bensomorfaner och derassyraadditionssalter FI63399C (fi)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19772716687 DE2716687A1 (de)	1977-04-15	1977-04-15	2'-hydroxy-2-(5-isoxazolylmethyl)-6,7benzomorphane, deren saeureadditionssalze und diese enthaltende arzneimittel
DE2716687		1977-04-15

Publications (3)

Publication Number	Publication Date
FI781025A true FI781025A (fi)	1978-10-16
FI63399B FI63399B (fi)	1983-02-28
FI63399C FI63399C (fi)	1983-06-10

Family

ID=6006359

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI781025A FI63399C (fi)	1977-04-15	1978-04-04	Foerfarande foer framstaellning av farmakologiskt vaerdefulla 2'-hydroxi-2-(5-isoxazolylmetyl)-6,7-bensomorfaner och derassyraadditionssalter

Country Status (25)

Country	Link
US (1)	US4133888A (fi)
JP (1)	JPS53130671A (fi)
AT (3)	AT358192B (fi)
AU (1)	AU514938B2 (fi)
BE (1)	BE866013A (fi)
CA (1)	CA1079726A (fi)
CH (1)	CH638519A5 (fi)
DE (1)	DE2716687A1 (fi)
DK (1)	DK144678C (fi)
ES (3)	ES468798A1 (fi)
FI (1)	FI63399C (fi)
FR (1)	FR2387228A1 (fi)
GB (1)	GB1575156A (fi)
GR (1)	GR64819B (fi)
IE (1)	IE46722B1 (fi)
IL (1)	IL54509A (fi)
IT (1)	IT1102595B (fi)
LU (1)	LU79430A1 (fi)
NL (1)	NL7803977A (fi)
NO (1)	NO148418C (fi)
NZ (1)	NZ186971A (fi)
PH (1)	PH13854A (fi)
PT (1)	PT67907B (fi)
SE (1)	SE430160B (fi)
ZA (1)	ZA782149B (fi)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1575009A (en) *	1976-06-21	1980-09-17	Acf Chemiefarma Nv	6,7-benzomorphan derivatives
NL7907800A (nl)	1979-10-23	1981-04-27	Acf Chemiefarma Nv	Nieuwe 6,7-benzomorfanderivaten en zuuradditiezouten daarvan, farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werkwijze voor het bereiden van deze verbindingen en de farmaceutische preparaten.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3499906A (en) *	1966-05-20	1970-03-10	Merck & Co Inc	5,9-diethyl-2'-hydroxy-2-substituted-6,7-benzomorphans
CS166801B2 (fi) *	1971-02-08	1976-03-29	Boehringer Sohn Ingelheim
US3853889A (en) *	1973-07-18	1974-12-10	Bristol Myers Co	3,14-substituted-8-oxamorphinans
DE2411382C3 (de) *	1974-03-09	1979-09-06	C.H. Boehringer Sohn, 6507 Ingelheim	2-Tetrahydrofurfuryl-6,7-benzomorphane, Verfahren zur Herstellung und deren Verwendung
DE2437610A1 (de) *	1974-08-05	1976-02-26	Boehringer Sohn Ingelheim	Neue 5,9-beta-disubstituierte 2-tetrahydrofurfuryl-6,7-benzomorphane, deren saeureadditionssalze, ihre verwendung als arzneimittel und verfahren zu deren herstellung

1977
- 1977-04-15 DE DE19772716687 patent/DE2716687A1/de not_active Ceased
1978
- 1978-04-04 FI FI781025A patent/FI63399C/fi not_active IP Right Cessation
- 1978-04-06 AT AT241978A patent/AT358192B/de not_active IP Right Cessation
- 1978-04-06 GR GR55915A patent/GR64819B/el unknown
- 1978-04-12 CH CH394078A patent/CH638519A5/de not_active IP Right Cessation
- 1978-04-12 US US05/895,631 patent/US4133888A/en not_active Expired - Lifetime
- 1978-04-13 IT IT48887/78A patent/IT1102595B/it active
- 1978-04-13 LU LU79430A patent/LU79430A1/de unknown
- 1978-04-14 JP JP4409178A patent/JPS53130671A/ja active Pending
- 1978-04-14 IE IE742/78A patent/IE46722B1/en unknown
- 1978-04-14 FR FR7811110A patent/FR2387228A1/fr active Granted
- 1978-04-14 PT PT67907A patent/PT67907B/pt unknown
- 1978-04-14 BE BE186818A patent/BE866013A/xx not_active IP Right Cessation
- 1978-04-14 ZA ZA00782149A patent/ZA782149B/xx unknown
- 1978-04-14 IL IL54509A patent/IL54509A/xx unknown
- 1978-04-14 ES ES468798A patent/ES468798A1/es not_active Expired
- 1978-04-14 DK DK163578A patent/DK144678C/da not_active IP Right Cessation
- 1978-04-14 NZ NZ186971A patent/NZ186971A/xx unknown
- 1978-04-14 GB GB14796/78A patent/GB1575156A/en not_active Expired
- 1978-04-14 SE SE7804260A patent/SE430160B/sv not_active IP Right Cessation
- 1978-04-14 NO NO781310A patent/NO148418C/no unknown
- 1978-04-14 AU AU35098/78A patent/AU514938B2/en not_active Expired
- 1978-04-14 PH PH21010A patent/PH13854A/en unknown
- 1978-04-14 NL NL7803977A patent/NL7803977A/xx not_active Application Discontinuation
- 1978-04-14 CA CA301,198A patent/CA1079726A/en not_active Expired
- 1978-08-07 ES ES472407A patent/ES472407A1/es not_active Expired
- 1978-08-07 ES ES472408A patent/ES472408A1/es not_active Expired
1979
- 1979-08-14 AT AT552079A patent/AT360667B/de not_active IP Right Cessation
- 1979-08-14 AT AT551979A patent/AT360666B/de not_active IP Right Cessation

Also Published As

Publication number	Publication date
ES468798A1 (es)	1978-12-01
FI63399C (fi)	1983-06-10
CH638519A5 (de)	1983-09-30
NZ186971A (en)	1980-10-24
IT1102595B (it)	1985-10-07
BE866013A (fr)	1978-10-16
ATA551979A (de)	1980-06-15
AU3509878A (en)	1979-10-18
CA1079726A (en)	1980-06-17
IE780742L (en)	1978-10-15
LU79430A1 (de)	1979-05-25
AT360666B (de)	1981-01-26
SE430160B (sv)	1983-10-24
ES472408A1 (es)	1979-04-01
DK144678B (da)	1982-05-10
PH13854A (en)	1980-10-22
ZA782149B (en)	1979-12-27
IT7848887A0 (it)	1978-04-13
DE2716687A1 (de)	1978-10-19
AU514938B2 (en)	1981-03-05
JPS53130671A (en)	1978-11-14
FR2387228A1 (fr)	1978-11-10
IL54509A0 (en)	1978-07-31
IE46722B1 (en)	1983-09-07
ES472407A1 (es)	1979-04-01
PT67907A (fr)	1978-05-01
SE7804260L (sv)	1978-10-16
NO781310L (no)	1978-10-17
AT358192B (de)	1980-08-25
GR64819B (en)	1980-06-03
ATA552079A (de)	1980-06-15
AT360667B (de)	1981-01-26
ATA241978A (de)	1980-01-15
PT67907B (fr)	1980-06-16
DK163578A (da)	1978-10-16
FR2387228B1 (fi)	1981-05-29
DK144678C (da)	1982-10-11
NO148418B (no)	1983-06-27
NO148418C (no)	1983-10-05
GB1575156A (en)	1980-09-17
NL7803977A (nl)	1978-10-17
IL54509A (en)	1982-04-30
FI63399B (fi)	1983-02-28
US4133888A (en)	1979-01-09

Publication	Publication Date	Title
FI780365A (fi)	1978-08-11	Anordning foer dosering av laekemedel
FI54627B (fi)	1978-09-29	Foerrfarande och anordning i torkpartiet i en papersmaskin
FI783329A (fi)	1979-05-09	Foerbaettringar i och angaoende ytbehandlingar
FI65935B (fi)	1984-04-30	Temperaturbestaendig slipkropp och foerfarande foer framstaellning daerav
IT1112641B (it)	1986-01-20	Respiratore
FI780225A (fi)	1978-07-25	Toalettstolsinsats och saett tillverka densamma
FI780565A (fi)	1978-08-23	Foerfarande foer framstaellning av d 1-5-metyltetrahydrofolsyra och salter daerav
FI821762A0 (fi)	1982-05-19	Dekorativa bestickgrepp och foerfarande foer deras framstaellning
FI780240A (fi)	1978-08-19	Blandningsventilanordning foer kallt och varmt vatten
IT1100022B (it)	1985-09-28	Apparecchio d'innaffiatura
FI781218A (fi)	1978-10-28	Totalbestaemning av hormoner och laekemedel
FI783991A (fi)	1979-06-28	Foerfarande foer behandling av hypertension och laekemedel foer detta
DK481878A (da)	1979-05-01	Loefteindretning
IT1174253B (it)	1987-07-01	Respiratore
FI782173A (fi)	1979-01-07	Benzylpyrimidiner foerfarande foer framstaellning av dem och laekemedel innehaollande dessa
FI780693A (fi)	1978-09-06	Bensylpyrimidiner foerfarande foer deras framstaellning och desamma innehaollande laekemedel
FI780355A (fi)	1978-08-05	Halvsyntetiska 4"-amino-oleando-mycinderivat
SE7800659L (sv)	1978-09-29	Profilfres
FI781025A (fi)	1978-10-16	2'-hydroxi-2-(5-isoxazolylmetyl)-6 7-bentzomorfaner deras syraadditionssalter och dessa innehaollande laekemedel
FI780354A (fi)	1978-08-05	Halvsyntetiska 4"-erytromysin-a-derivat
FI780427A (fi)	1978-08-15	Heterocyklopyrimidiner foereningar och terapeutiskt foerfarande
FI780420A (fi)	1978-08-15	Everninomicinderivat och deras framstaellning
FI780394A (fi)	1978-08-25	Skidkaenga och en foer denna avsedd skidbindning
FI780313A (fi)	1978-08-10	Mellanprodukter och framstaellningsfoerfaranden
FI780336A (fi)	1978-08-26	Triazolo-thieno-diazepin-1-oner foerfarande foer deras framstaellning och laekemedel

Legal Events

Date	Code	Title	Description
2004-08-31	MM	Patent lapsed	Owner name: C.H. BOEHRINGER SOHN