FI20010214L - Asyyliaminoindolijohdannaisia - Google Patents

Asyyliaminoindolijohdannaisia Download PDF

Info

Publication number: FI20010214L
Authority: FI; Finland
Prior art keywords: acylaminoindole; derivatives; acylaminoindole derivatives
Prior art date: 1992-04-10

Application number

FI20010214A

Other languages

English (en)

Swedish (sv)

Inventor

John E Macor

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-04-10

Filing date

2001-02-05

Publication date

2001-02-05

2001-02-05 Application filed by Pfizer filed Critical Pfizer

2001-02-05 Publication of FI20010214L publication Critical patent/FI20010214L/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Obesity (AREA)
Diabetes (AREA)
Hematology (AREA)
Anesthesiology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Child & Adolescent Psychology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Materials For Photolithography (AREA)
Soft Magnetic Materials (AREA)
Supply Devices, Intensifiers, Converters, And Telemotors (AREA)
Pyrrole Compounds (AREA)

FI20010214A 1992-04-10 2001-02-05 Asyyliaminoindolijohdannaisia FI20010214L (fi)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US86638292A	1992-04-10	1992-04-10

Publications (1)

Publication Number	Publication Date
FI20010214L true FI20010214L (fi)	2001-02-05

Family

ID=25347493

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
FI931613A FI111256B (fi)	1992-04-10	1993-04-08	Menetelmä terapeuttisesti käyttökelpoisten asyyliaminoindolijohdannaisten valmistamiseksi
FI20010214A FI20010214L (fi)	1992-04-10	2001-02-05	Asyyliaminoindolijohdannaisia

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
FI931613A FI111256B (fi)	1992-04-10	1993-04-08	Menetelmä terapeuttisesti käyttökelpoisten asyyliaminoindolijohdannaisten valmistamiseksi

Country Status (31)

Country	Link
US (1)	US5498626A (fi)
EP (1)	EP0635015B1 (fi)
JP (1)	JP2544704B2 (fi)
KR (1)	KR0179074B1 (fi)
CN (1)	CN1038506C (fi)
AT (1)	ATE148465T1 (fi)
AU (1)	AU670270B2 (fi)
BR (1)	BR9306221A (fi)
CA (1)	CA2132706C (fi)
CZ (1)	CZ282653B6 (fi)
DE (1)	DE69307875T2 (fi)
DK (1)	DK0635015T3 (fi)
EG (1)	EG20466A (fi)
ES (1)	ES2097496T3 (fi)
FI (2)	FI111256B (fi)
GR (1)	GR3022767T3 (fi)
HR (1)	HRP930753B1 (fi)
HU (1)	HUT64060A (fi)
IL (1)	IL105309A0 (fi)
MX (1)	MX9301996A (fi)
MY (1)	MY115278A (fi)
NO (1)	NO309860B1 (fi)
NZ (1)	NZ251047A (fi)
PL (1)	PL172232B1 (fi)
RU (1)	RU2110516C1 (fi)
SK (1)	SK278182B6 (fi)
TW (1)	TW394769B (fi)
UA (1)	UA34452C2 (fi)
WO (1)	WO1993021180A1 (fi)
YU (1)	YU48916B (fi)
ZA (1)	ZA932536B (fi)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5559246A (en) *	1990-10-15	1996-09-24	Pfizer Inc.	Indole derivatives
US5559129A (en) *	1990-10-15	1996-09-24	Pfizer Inc	Indole derivatives
US5545644A (en) *	1990-10-15	1996-08-13	Pfizer Inc.	Indole derivatives
US5578612A (en) *	1990-10-15	1996-11-26	Pfizer Inc.	Indole derivatives
US5607951A (en) *	1990-10-15	1997-03-04	Pfizer Inc	Indole derivatives
US6380233B1 (en)	1992-04-07	2002-04-30	Pfizer Inc	Indole derivatives as 5-HT1 agonists
CA2133413C (en)	1992-04-07	2001-04-10	John Eugene Macor	Indole derivatives as 5-ht1 antagonists
ES2070772B1 (es) *	1993-08-09	1996-02-16	Pfizer	Derivados de acilaminoindol
CZ59996A3 (en) *	1993-08-31	1996-06-12	Pfizer	5-arylindole derivatives per se and for treating diseases, intermediates for their preparation and pharmaceutical compositions based thereon
GB9402016D0 (en) *	1994-02-02	1994-03-30	Merck Sharp & Dohme	Therapeutic agents
GB9402011D0 (en) *	1994-02-02	1994-03-30	Merck Sharp & Dohme	Therapeutic agents
AU3162695A (en) *	1994-08-03	1996-03-04	Asta Medica Aktiengesellschaft	Indol, indazol, pyridopyrrol and pyridopyrazol derivatives with anti-asthmatic, anti-allergic, anti-inflammatory and immunomodulating effects
GB9417310D0 (en)	1994-08-27	1994-10-19	Pfizer Ltd	Therapeutic agents
GB9420503D0 (en) *	1994-10-11	1994-11-23	Pfizer Ltd	Therapeutic agents
GB9420529D0 (en)	1994-10-12	1994-11-30	Pfizer Ltd	Indoles
WO1999053956A1 (fr) *	1998-04-16	1999-10-28	Yamanouchi Pharmaceutical Co., Ltd.	Remedes contre l'obesite
US5994352A (en) *	1998-11-13	1999-11-30	Pfizer Inc.	5-arylindole derivatives
AU2004206909A1 (en) *	2003-01-22	2004-08-05	Gtx Inc.	Treating androgen deficiency in female (ADIF)-associated conditions with sarms
WO2009071988A1 (en) *	2007-12-07	2009-06-11	Pfizer Inc.	Tosylate salt of trans-n-isobutyl-3-fluoro-3- [3-flu0r0-4- (pyrrolidin-1-yl-methyl) -phenyl] cyclobut anecarboxamide
WO2014078568A1 (en)	2012-11-14	2014-05-22	The Johns Hopkins University	Methods and compositions for treating schizophrenia
CN103408535B (zh) *	2013-08-13	2016-03-02	张家港威胜生物医药有限公司	一种依来曲普坦中间体-5-溴-3-(n-甲基吡咯啉-2-基甲基)-1h-吲哚合成工艺

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA795239B (en) *	1978-10-12	1980-11-26	Glaxo Group Ltd	Heterocyclic compounds
BE889931A (fr) *	1980-08-12	1982-02-11	Glaxo Group Ltd	Derives indoliques, leur preparation et leurs applications en tant que medicaments
GB2083463B (en) *	1980-08-12	1984-05-10	Glaxo Group Ltd	Heterocyclic compounds
GB8600397D0 (en) *	1986-01-08	1986-02-12	Glaxo Group Ltd	Chemical compounds
GB8719167D0 (en) *	1987-08-13	1987-09-23	Glaxo Group Ltd	Chemical compounds
GB8724912D0 (en) *	1987-10-23	1987-11-25	Wellcome Found	Indole derivatives
GB8819024D0 (en) *	1988-08-10	1988-09-14	Glaxo Group Ltd	Chemical compounds
IL96891A0 (en) *	1990-01-17	1992-03-29	Merck Sharp & Dohme	Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them
CA2042295A1 (fr) *	1990-05-15	1991-11-16	Jacques Chauveau	Derives de mediateurs endogenes, leurs sels, procede de preparation, applications, et compositions les renfermant
IL114690A (en) *	1990-06-07	1997-02-18	Wellcome Found	Antimigraine oxazolidinone substituted indole derivatives
JP2575272B2 (ja) *	1990-10-15	1997-01-22	フアイザー・インコーポレイテツド	インドール誘導体
US5208248A (en) *	1991-01-11	1993-05-04	Merck Sharpe & Dohme, Ltd.	Indazole-substituted five-membered heteroaromatic compounds
CZ283018B6 (cs) *	1991-02-01	1997-12-17	Merck Sharp And Dohme Limited	Deriváty imidazolu, triazolu a tetrazolu a farmaceutické přípravky na jejich bázi
ES2143992T3 (es) *	1991-11-25	2000-06-01	Pfizer	Derivados de 5-(hetero- o carbociclilamino)-indol, su preparacion y uso como 5-ht1 agonistas.

1993
- 1993-03-04 US US08/295,792 patent/US5498626A/en not_active Expired - Fee Related
- 1993-03-04 DK DK93907096.7T patent/DK0635015T3/da active
- 1993-03-04 UA UA94105907A patent/UA34452C2/uk unknown
- 1993-03-04 JP JP5518302A patent/JP2544704B2/ja not_active Expired - Fee Related
- 1993-03-04 WO PCT/US1993/001807 patent/WO1993021180A1/en active IP Right Grant
- 1993-03-04 EP EP93907096A patent/EP0635015B1/en not_active Expired - Lifetime
- 1993-03-04 BR BR9306221A patent/BR9306221A/pt not_active Application Discontinuation
- 1993-03-04 AU AU37821/93A patent/AU670270B2/en not_active Ceased
- 1993-03-04 CZ CZ942477A patent/CZ282653B6/cs not_active IP Right Cessation
- 1993-03-04 NZ NZ251047A patent/NZ251047A/en unknown
- 1993-03-04 KR KR1019940703551A patent/KR0179074B1/ko not_active Expired - Fee Related
- 1993-03-04 CA CA002132706A patent/CA2132706C/en not_active Expired - Fee Related
- 1993-03-04 SK SK1207-94A patent/SK278182B6/sk unknown
- 1993-03-04 PL PL93305558A patent/PL172232B1/pl not_active IP Right Cessation
- 1993-03-04 AT AT93907096T patent/ATE148465T1/de not_active IP Right Cessation
- 1993-03-04 ES ES93907096T patent/ES2097496T3/es not_active Expired - Lifetime
- 1993-03-04 DE DE69307875T patent/DE69307875T2/de not_active Expired - Fee Related
- 1993-03-04 RU RU94045902/04A patent/RU2110516C1/ru not_active IP Right Cessation
- 1993-03-09 TW TW082101732A patent/TW394769B/zh active
- 1993-04-02 HR HR930753A patent/HRP930753B1/xx not_active IP Right Cessation
- 1993-04-05 IL IL105309A patent/IL105309A0/xx not_active IP Right Cessation
- 1993-04-06 MX MX9301996A patent/MX9301996A/es unknown
- 1993-04-07 EG EG21493A patent/EG20466A/xx active
- 1993-04-08 MY MYPI93000646A patent/MY115278A/en unknown
- 1993-04-08 ZA ZA932536A patent/ZA932536B/xx unknown
- 1993-04-08 FI FI931613A patent/FI111256B/fi not_active IP Right Cessation
- 1993-04-09 YU YU25593A patent/YU48916B/sh unknown
- 1993-04-09 CN CN93104439A patent/CN1038506C/zh not_active Expired - Fee Related
- 1993-04-09 HU HU9301048A patent/HUT64060A/hu unknown
1994
- 1994-10-07 NO NO943803A patent/NO309860B1/no not_active IP Right Cessation
1997
- 1997-03-07 GR GR970400451T patent/GR3022767T3/el unknown
2001
- 2001-02-05 FI FI20010214A patent/FI20010214L/fi unknown

Also Published As

Publication number	Publication date
HRP930753A2 (en)	1994-10-31
WO1993021180A1 (en)	1993-10-28
NZ251047A (en)	1996-09-25
FI931613A0 (fi)	1993-04-08
HRP930753B1 (en)	2000-10-31
BR9306221A (pt)	1998-06-30
MX9301996A (es)	1994-03-31
KR0179074B1 (ko)	1999-03-20
GR3022767T3 (en)	1997-06-30
NO943803L (no)	1994-10-07
NO943803D0 (no)	1994-10-07
RU94045902A (ru)	1996-08-27
PL172232B1 (pl)	1997-08-29
SK120794A3 (en)	1995-05-10
DK0635015T3 (da)	1997-03-17
EP0635015A1 (en)	1995-01-25
FI931613L (fi)	1993-10-11
TW394769B (en)	2000-06-21
HU9301048D0 (en)	1993-06-28
JP2544704B2 (ja)	1996-10-16
IL105309A0 (en)	1993-08-18
YU25593A (sh)	1996-10-09
CN1080288A (zh)	1994-01-05
ATE148465T1 (de)	1997-02-15
JPH07501831A (ja)	1995-02-23
YU48916B (sh)	2002-11-15
NO309860B1 (no)	2001-04-09
FI111256B (fi)	2003-06-30
EP0635015B1 (en)	1997-01-29
EG20466A (en)	1999-05-31
CZ247794A3 (en)	1995-07-12
AU670270B2 (en)	1996-07-11
UA34452C2 (uk)	2001-03-15
ES2097496T3 (es)	1997-04-01
RU2110516C1 (ru)	1998-05-10
KR950700903A (ko)	1995-02-20
SK278182B6 (en)	1996-03-06
CZ282653B6 (cs)	1997-08-13
ZA932536B (en)	1994-10-08
CA2132706C (en)	1998-08-04
DE69307875T2 (de)	1997-05-22
MY115278A (en)	2003-05-31
DE69307875D1 (de)	1997-03-13
US5498626A (en)	1996-03-12
HUT64060A (en)	1993-11-29
AU3782193A (en)	1993-11-18
CN1038506C (zh)	1998-05-27
CA2132706A1 (en)	1993-10-28

Publication	Publication Date	Title
FI930208L (fi)	1993-07-21	Kinazolinderivat
FI980341L (fi)	1998-02-13	2-oksi-indolijohdannaisia
ATA75293A (de)	1997-11-15	Indolderivate
DE69208877D1 (de)	1996-04-11	Chinuclidinderivate
FI924159L (fi)	1993-03-19	Benzanilidderivat
NO922182D0 (no)	1992-06-02	Krystallinske oksatiolan-derivater
FI935902L (fi)	1994-02-10	Ofodrad foerslutningsanordning
DE69330497D1 (de)	2001-08-30	Chinazolin-derivate
FI925763A0 (fi)	1992-12-18	Fungicida 2-imidazolin-5-on- och 2-imidazolin-5-tionderivat
FI923726L (fi)	1993-02-24	Sulfaterade glykosaminoglykanoidderivat
FI20010214L (fi)	2001-02-05	Asyyliaminoindolijohdannaisia
FI945674L (fi)	1995-06-03	Substituoidut 2beta-morfoliini-androstaanijohdannaiset
DE59308714D1 (de)	1998-07-30	Cyclobutan-benzol-derivate
FI20002460L (fi)	2000-11-09	4-difenyylimetyylipiperidiinijohdannaisia
FI943885L (fi)	1995-02-25	Penaami-johdannaiset
AT399443B (de)	1995-05-26	Sportschuh
FI944044L (fi)	1995-03-03	Fenyylialkanoliamiinijohdannaiset
FI935243L (fi)	1994-01-11	Pyridonkarboxylsyraderivat
ATA236892A (de)	1996-12-15	Rotornut
NO952288D0 (no)	1995-06-09	Benzazepinon-derivater
DE69313890D1 (de)	1997-10-23	5-Aminoflavon-Derivate
FI930367L (fi)	1993-08-01	Puridinderivat
FI924145L (fi)	1993-03-18	3-cykloalkylprop-2-enamidderivat
DE59407726D1 (de)	1999-03-11	3-Aryl-4-hydroxy-3-dihydrofuranon-Derivate
FI942070L (fi)	1994-05-05	Nitroksialkyyliamidijohdannaiset