[go: up one dir, main page]

ES8704964A1 - Un procedimiento para preparar derivados esteres del antibiotico l 17046. - Google Patents

Un procedimiento para preparar derivados esteres del antibiotico l 17046.

Info

Publication number
ES8704964A1
ES8704964A1 ES548789A ES548789A ES8704964A1 ES 8704964 A1 ES8704964 A1 ES 8704964A1 ES 548789 A ES548789 A ES 548789A ES 548789 A ES548789 A ES 548789A ES 8704964 A1 ES8704964 A1 ES 8704964A1
Authority
ES
Spain
Prior art keywords
antibiotic
ester derivatives
directed
antimicrobial activity
positive bacteria
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES548789A
Other languages
English (en)
Other versions
ES548789A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gruppo Lepetit SpA
Original Assignee
Gruppo Lepetit SpA
Lepetit SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruppo Lepetit SpA, Lepetit SpA filed Critical Gruppo Lepetit SpA
Publication of ES548789A0 publication Critical patent/ES548789A0/es
Publication of ES8704964A1 publication Critical patent/ES8704964A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H3/00—Compounds containing only hydrogen atoms and saccharide radicals having only carbon, hydrogen, and oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/19—Antibiotic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Biotechnology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Catalysts (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS ESTERES DEL ANTIBIOTICO L 17046, DE FORMULA GENERAL (I), Y SUS SALES DE ADICION DE ACIDO FARMACEUTICAMENTE ACEPTABLES. CONSISTE EN HACER REACCIONAR UN DERIVADO ANTIBIOTICO L 17046 N-PROTEGIDO, DE FORMULA GENERAL (II), EN LA QUE A Y M REPRESENTAN CADA UNO DE ELLOS UN ATOMO DE HIDROGENO; B ES UN GRUPO N-ACETIL-B-D-GLUCOSAMINILO; Y R1 REPRESENTA UN GRUPO PROTECTOR DE NITROGENO, CON UN COMPUESTO DE FORMULA GENERAL (III), EN LA QUE R REPRESENTA ALQUILO O HIDROALQUILO; Y X REPRESENTA UN ATOMO DE CLORO, BROMO O YODO, EN UN DISOLVENTE APROTICO POLAR ORGANICO INERTE. DE APLICACION EN FARMACIA.
ES548789A 1984-11-13 1985-11-12 Un procedimiento para preparar derivados esteres del antibiotico l 17046. Expired ES8704964A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB848428619A GB8428619D0 (en) 1984-11-13 1984-11-13 Derivatives of antibiotic l 17046

Publications (2)

Publication Number Publication Date
ES548789A0 ES548789A0 (es) 1987-04-16
ES8704964A1 true ES8704964A1 (es) 1987-04-16

Family

ID=10569641

Family Applications (1)

Application Number Title Priority Date Filing Date
ES548789A Expired ES8704964A1 (es) 1984-11-13 1985-11-12 Un procedimiento para preparar derivados esteres del antibiotico l 17046.

Country Status (13)

Country Link
US (1) US4661470A (es)
EP (1) EP0182157B1 (es)
JP (1) JPS61122300A (es)
KR (1) KR860004076A (es)
AT (1) ATE78261T1 (es)
CA (1) CA1250098A (es)
DE (1) DE3586344T2 (es)
DK (1) DK508885A (es)
ES (1) ES8704964A1 (es)
GB (1) GB8428619D0 (es)
HU (1) HU196228B (es)
IL (1) IL76996A0 (es)
ZA (1) ZA858449B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT86457B (pt) * 1986-12-30 1990-11-20 Smithkline Beecham Corp Processo para a preparacao de glicopeptidos glicosilados e de composicoes que os contem
US4882313A (en) * 1987-07-31 1989-11-21 Smithkline Beckman Corporation Carboxamide derivatives of glycopeptides
GB8808658D0 (en) * 1988-04-13 1988-05-18 Lepetit Spa Aglycons of a/16686 antibiotics
US5606036A (en) * 1991-03-27 1997-02-25 Gruppo Lepetit Spa Antibiotic A 40926 ester derivatives
SG87877A1 (en) * 1998-12-23 2002-04-16 Advanced Medicine Inc Glycopeptide derivatives and pharmaceutical compositions containing the same
HU230190B1 (hu) * 1998-12-23 2015-09-28 Theravance, Inc Glikopeptidszármazékok és ezeket tartalmazó gyógyászati kompozíciók
US20060074014A1 (en) * 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
EP1565201B1 (en) 2002-11-18 2018-10-31 Vicuron Pharmaceuticals, Inc. Methods of administering dalbavancin for treatment of bacterial infections
US7119061B2 (en) * 2002-11-18 2006-10-10 Vicuron Pharmaceuticals, Inc. Dalbavancin compositions for treatment of bacterial infections

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ199196A (en) * 1980-12-18 1985-01-31 Lilly Co Eli Antibiotic a-4696 factor g and growth-promoting compositions;actinoplanes missouriensis atcc 31681
FI73697C (fi) * 1982-06-08 1987-11-09 Lepetit Spa Foerfarande foer framstaellning av individuella faktorer 1, 2, 3, 4 och 5 av teikomysin a2.
GB8307847D0 (en) * 1983-03-22 1983-04-27 Lepetit Spa Antibiotics l 17054 and l 17046
GB8415092D0 (en) * 1984-06-13 1984-07-18 Lepetit Spa Ester derivatives

Also Published As

Publication number Publication date
DK508885D0 (da) 1985-11-05
EP0182157A3 (en) 1987-12-09
DK508885A (da) 1986-05-14
ES548789A0 (es) 1987-04-16
ZA858449B (en) 1986-08-27
US4661470A (en) 1987-04-28
DE3586344D1 (de) 1992-08-20
EP0182157B1 (en) 1992-07-15
EP0182157A2 (en) 1986-05-28
GB8428619D0 (en) 1984-12-19
KR860004076A (ko) 1986-06-16
IL76996A0 (en) 1986-04-29
JPS61122300A (ja) 1986-06-10
CA1250098A (en) 1989-02-14
ATE78261T1 (de) 1992-08-15
HU196228B (en) 1988-10-28
HUT41053A (en) 1987-03-30
DE3586344T2 (de) 1993-03-11

Similar Documents

Publication Publication Date Title
YU45524B (en) Process for preparing derivatives of s(-)-pyridobenzoxazine
ES470437A1 (es) Un procedimiento para la preparacion de nuevos esteres an- tibacterianos
JO1704B1 (en) New potent compounds
EP0177940A3 (en) Hydrazine derivatives and their use
ES8704964A1 (es) Un procedimiento para preparar derivados esteres del antibiotico l 17046.
GR3024925T3 (en) Antifungal agent, its preparation and microorganism therefor
SE8502135D0 (sv) 4'-deschlororebeccamycin and process for its preparation
ES8606360A1 (es) Un derivado de cefalosporina.
ES8609366A1 (es) Un procedimiento para preparar un derivado de ester de des- glucoteicoplanina
CA2053359A1 (en) Heteroaroyl derivatives of monocyclic beta-lactam antibiotics
GB2199746B (en) Stabilization of antibiotic compositions with salts.
DE3885394D1 (de) Teicoplaninähnliche Derivate.
AU2857492A (en) Improved fish production
AU558707B2 (en) Water soluble rifamycin derivatives
GR75173B (es)
CA1270247C (en) 3-ACYLAMINO-2-OXO-1-AZETIDINESULFONIC ACIDS
IN172911B (es)
ES8107309A1 (es) Un procedimiento de produccion de derivados de 7 -metoxice- falosporina
CA1271750C (en) 3-ACYLAMINO-2-OXO-1-AZETIDINESULFONIC ACIDS
ZA841850B (en) 2'-desoxyoxanosine,a process for the preparation thereof and its use as a medicament
SU1226790A1 (ru) Реагент для предотвращения роста сульфатвосстанавливающих бактерий
SU1231878A1 (ru) Антибиотик 985 и, обладающий антибактериальной активностью, и штамм streptomyces chromopurpureus subsp. chiketamanus subsp. nov. 985 - продуцент антибиотика 985 и
SU1262908A1 (ru) Гидрохлорид 1-(2'-этоксиэтил)-4-фенил-4-пропионилоксипиперидина, обладающий анальгетической активностью
SU1455633A1 (ru) О,о-диизопропил-о-[1, 1-диметил-2-пропилтио-2-(о-о-диизопропилфосфорил)- имино]-этилфосфат, обладающий бактерицидной активностью
SU1448442A1 (ru) Препарат для лечения и профилактики вольфартиоза сельскохозяйственных животных

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970401