[go: up one dir, main page]

ES475533A1 - Un metodo para la preparacion de formas racemicas y optica- mente activas de 2-(4-difenilil)-n-(dimetilamino-alquil)pro-pionamida - Google Patents

Un metodo para la preparacion de formas racemicas y optica- mente activas de 2-(4-difenilil)-n-(dimetilamino-alquil)pro-pionamida

Info

Publication number
ES475533A1
ES475533A1 ES475533A ES475533A ES475533A1 ES 475533 A1 ES475533 A1 ES 475533A1 ES 475533 A ES475533 A ES 475533A ES 475533 A ES475533 A ES 475533A ES 475533 A1 ES475533 A1 ES 475533A1
Authority
ES
Spain
Prior art keywords
novel
manufacture
amide derivative
novel compounds
parenteral
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES475533A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
A Menarini SAS
Original Assignee
A Menarini SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by A Menarini SAS filed Critical A Menarini SAS
Publication of ES475533A1 publication Critical patent/ES475533A1/es
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES475533A 1977-11-30 1978-11-29 Un metodo para la preparacion de formas racemicas y optica- mente activas de 2-(4-difenilil)-n-(dimetilamino-alquil)pro-pionamida Expired ES475533A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT964377A IT1090782B (it) 1977-11-30 1977-11-30 2 4 bifenilil 2 dietilamino alchil propionamide suoi sali e procedimenti di fabbricazione relativi

Publications (1)

Publication Number Publication Date
ES475533A1 true ES475533A1 (es) 1980-01-16

Family

ID=11132874

Family Applications (1)

Application Number Title Priority Date Filing Date
ES475533A Expired ES475533A1 (es) 1977-11-30 1978-11-29 Un metodo para la preparacion de formas racemicas y optica- mente activas de 2-(4-difenilil)-n-(dimetilamino-alquil)pro-pionamida

Country Status (9)

Country Link
JP (1) JPS5490157A (ja)
BE (1) BE872403A (ja)
CA (1) CA1118446A (ja)
CH (1) CH637370A5 (ja)
DE (1) DE2851416A1 (ja)
ES (1) ES475533A1 (ja)
FR (1) FR2410641A1 (ja)
IT (1) IT1090782B (ja)
NL (1) NL7811698A (ja)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20012025A1 (it) * 2001-09-28 2003-03-28 Dompe Spa Sali di ammonio quaternari di omega-amminoalchilammidi di acidi r 2-aril-propionici e composizioni farmaceutiche che li contengono
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
PL2049482T3 (pl) * 2006-08-08 2016-04-29 Techfields Biochem Co Ltd Dodatnio naładowane rozpuszczalne w wodzie proleki kwasów arylo- i heteroarylooctowych o bardzo dużej szybkości przenikania przez skórę
JP5424880B2 (ja) * 2006-08-15 2014-02-26 テックフィールズ バイオケム カンパニー リミテッド 非常に速い皮膚透過率を有するアリール−及びヘテロアリールプロピオン酸の正荷電水溶性プロドラッグ
AU2013206218B2 (en) * 2006-08-15 2016-06-30 Techfields Biochem Co. Ltd Positively charged water-soluble prodrugs of aryl- and heteroarylpropionic acids with very fast skin penetration rate
RU2509076C2 (ru) 2007-06-04 2014-03-10 Текфилдз Инк Пролекарства нестероидных противовоспалительных средств (nsaia) c очень высокой скоростью проникновения через кожу и мембраны и новые медицинские применения указанных пролекарств
RU2765463C2 (ru) 2008-12-04 2022-01-31 Чунси ЮЙ Композиции интенсивного проникновения и их применение
JP5940036B2 (ja) * 2013-10-08 2016-06-29 テックフィールズ バイオケム カンパニー リミテッド 非常に速い皮膚透過率を有するアリール−及びヘテロアリールプロピオン酸の正荷電水溶性プロドラッグ
JP6290947B2 (ja) * 2016-02-05 2018-03-07 テックフィールズ バイオケム カンパニー リミテッド 非常に速い皮膚透過率を有するアリール−及びヘテロアリールプロピオン酸の正荷電水溶性プロドラッグ

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1584547A (ja) * 1968-06-05 1969-12-26
FR1593024A (ja) * 1968-09-18 1970-05-25
FR2119846A1 (en) * 1970-12-28 1972-08-11 Choay Sa N,n-diethylaminoethylamide of para isobutyl phenylacetic - acid - antiinflammatory and analgesic
US4145435A (en) * 1976-11-12 1979-03-20 The Upjohn Company 2-aminocycloaliphatic amide compounds

Also Published As

Publication number Publication date
FR2410641A1 (fr) 1979-06-29
BE872403A (fr) 1979-03-16
NL7811698A (nl) 1979-06-01
IT1090782B (it) 1985-06-26
DE2851416C2 (ja) 1989-02-23
JPS5490157A (en) 1979-07-17
CH637370A5 (en) 1983-07-29
DE2851416A1 (de) 1979-05-31
CA1118446A (en) 1982-02-16
FR2410641B1 (ja) 1983-04-15
JPS631286B2 (ja) 1988-01-12

Similar Documents

Publication Publication Date Title
ES485188A1 (es) Procedimiento para preparar 1-piperazina-carboxamidas y car-botiamidas
SE7614258L (sv) Forfarande for framstellning av kinazoloderivat
DE3686248D1 (de) Piperidinderivat, seine verwendung und diese enthaltende pharmazeutische zusammensetzung.
IL57648A (en) 2-substituted-5,9-dimethyl-2'-hydroxy-6,7-benzomorphanes,their preparation and pharmaceutical compositions containing them
FR2361901A1 (fr) Derives de substitution de nucleotides et medicament contenant ces substances
NO940523L (no) Nye pyrazin-derivater
ES8401961A1 (es) Procedimiento para la preparacion de nuevas n-(4-indolil-piperidino-alcohil-bencimidazolonas sustituidas.
ES475533A1 (es) Un metodo para la preparacion de formas racemicas y optica- mente activas de 2-(4-difenilil)-n-(dimetilamino-alquil)pro-pionamida
ATE59632T1 (de) Dihydrodibenzocycloheptylidenethylamin-derivate
GB1086192A (en) Phenylcyclopropane derivatives
SE8102220L (sv) Anvendning av substituerade derivat av 4-fenyl-4-oxo-2-butensyra sasom lekemedel
ES466851A1 (es) Procedimiento para la preparacion de 2-bromo-6-fluor-n-2- imidazolidinilidenbenzamina.
ES427079A1 (es) Un metodo de preparacion de fenotiazidas sustituidas por fluor en la posicion 7.
ES8502116A1 (es) Un compuesto de pirazolpiridina.
ES450897A1 (es) Procedimiento para la preparacion de n-(r-tetrahidrofurfu- ril)-noroximorfona y n-(s-tetrahidrofurfuril)-noroximorfona.
ES8203882A1 (es) Un procedimiento para la preparacion de 1-(8-quinole- il)-2-pirrolidinona y sus sales de adicion de acido
GB1169945A (en) Pharmaceutical Compositions containing Diphenylalkyl-amine Derivatives
ES466192A1 (es) Procedimiento para la obtencion de derivados de la isoqui- noleina.
ES466493A1 (es) Procedimiento de fabricacion de acidos a-aril-a -oxo-isovalericos.
IL71068A0 (en) N-arylpiperazine derivative,its preparation and pharmaceutical compositions containing it
FI862636A0 (fi) Farmaceutiska kompositoner med neuroleptisk effekt och foerfarande foer deras framstaellning.
AU530930B2 (en) Pharmaceutical compositions and method of treating heart disease
ES8305759A1 (es) "un procedimiento para la preparacion de 1-(1,3-bendodioxol-5-il)-2-pirrolidinona".
IL61769A0 (en) 2-phenylamino-imidazolines-(2),their preparation and pharmaceutical compositions containing them
ES8106147A1 (es) Procedimiento para preparar un 1,2,4-triazol-3-tiol

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19991102