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EA201001556A1 - Соединения, включающие противовоспалительный фармакофор, и способы их применения - Google Patents

Соединения, включающие противовоспалительный фармакофор, и способы их применения

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Publication number
EA201001556A1
EA201001556A1 EA201001556A EA201001556A EA201001556A1 EA 201001556 A1 EA201001556 A1 EA 201001556A1 EA 201001556 A EA201001556 A EA 201001556A EA 201001556 A EA201001556 A EA 201001556A EA 201001556 A1 EA201001556 A1 EA 201001556A1
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EA
Eurasian Patent Office
Prior art keywords
methods
inflammatory
application
pharmacofor
compounds including
Prior art date
Application number
EA201001556A
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English (en)
Other versions
EA020467B1 (ru
Inventor
Эрик Андерсон
Гэри Л. Бэултэн
Дебэрэ А. Фергусон
Зин Джайэнг
Роберт мл. Крэл
Патрик М. Обрайэн
Мелеэн Висник
Original Assignee
Ритэ Фамэсутикл, Инк.
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Publication of EA201001556A1 publication Critical patent/EA201001556A1/ru
Publication of EA020467B1 publication Critical patent/EA020467B1/ru

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    • C07C255/46—Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of non-condensed rings
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
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  • Diabetes (AREA)
  • Cardiology (AREA)
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  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Epidemiology (AREA)
  • Toxicology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Oncology (AREA)
  • Endocrinology (AREA)

Abstract

Изобретение направлено на создание новых соединений, содержащих следующий противовоспалительный фармакофоргде X, Rи Rтакие, как определено в данной заявке. Предлагается также фармацевтическая композиция, комплекты и изделия, содержащие такие соединения, способы и промежуточные вещества, применяемые при приготовлении соединений, а также способы применения соединений и композиций.
EA201001556A 2008-04-18 2009-04-20 Соединения, обладающие противовоспалительной активностью, и фармацевтическая композиция на их основе EA020467B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4636308P 2008-04-18 2008-04-18
PCT/US2009/041177 WO2009146218A2 (en) 2008-04-18 2009-04-20 Compounds including an anti-inflammatory pharmacore and methods of use

Publications (2)

Publication Number Publication Date
EA201001556A1 true EA201001556A1 (ru) 2011-06-30
EA020467B1 EA020467B1 (ru) 2014-11-28

Family

ID=40934110

Family Applications (1)

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EA201001556A EA020467B1 (ru) 2008-04-18 2009-04-20 Соединения, обладающие противовоспалительной активностью, и фармацевтическая композиция на их основе

Country Status (16)

Country Link
US (4) US8258329B2 (ru)
EP (1) EP2279196B1 (ru)
JP (1) JP5564490B2 (ru)
KR (1) KR101665042B1 (ru)
CN (2) CN102066397B (ru)
AU (1) AU2009251437B2 (ru)
BR (1) BRPI0911105B1 (ru)
CA (1) CA2721665C (ru)
CO (1) CO6311105A2 (ru)
EA (1) EA020467B1 (ru)
IL (1) IL208760A0 (ru)
MX (2) MX339476B (ru)
NZ (1) NZ588708A (ru)
SG (1) SG190564A1 (ru)
TW (1) TW201006474A (ru)
WO (1) WO2009146218A2 (ru)

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WO2009146218A8 (en) 2010-02-25
CA2721665C (en) 2017-01-24
MX2010011435A (es) 2011-01-25
US20100048887A1 (en) 2010-02-25
CN102066397B (zh) 2013-09-11

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