EA200600932A1 - Таблетки циталопрама гидробромида - Google Patents
Таблетки циталопрама гидробромидаInfo
- Publication number
- EA200600932A1 EA200600932A1 EA200600932A EA200600932A EA200600932A1 EA 200600932 A1 EA200600932 A1 EA 200600932A1 EA 200600932 A EA200600932 A EA 200600932A EA 200600932 A EA200600932 A EA 200600932A EA 200600932 A1 EA200600932 A1 EA 200600932A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- tablets
- gydrobromide
- citaloprama
- microns
- manufacture
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 abstract 2
- 239000002245 particle Substances 0.000 abstract 2
- WIHMBLDNRMIGDW-UHFFFAOYSA-N 1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-3h-2-benzofuran-5-carbonitrile;hydron;bromide Chemical compound [Br-].O1CC2=CC(C#N)=CC=C2C1(CCC[NH+](C)C)C1=CC=C(F)C=C1 WIHMBLDNRMIGDW-UHFFFAOYSA-N 0.000 abstract 1
- 229920000168 Microcrystalline cellulose Polymers 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 229960000584 citalopram hydrobromide Drugs 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 235000019813 microcrystalline cellulose Nutrition 0.000 abstract 1
- 239000008108 microcrystalline cellulose Substances 0.000 abstract 1
- 229940016286 microcrystalline cellulose Drugs 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Biomedical Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Изобретение относится к таблеткам как с пленочным покрытием, так и без такового, содержащим в качестве активного ингредиента циталопрам гидробромид, имеющий средний размер частиц менее чем 40 мкм, в смеси с микрокристаллической целлюлозой, имеющей средний размер частиц в интервале 90-250 мкм, и другими эксципиентами, применимыми для изготовления таблеток. В изобретении также предложен способ их изготовления.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU0303790A HU227491B1 (en) | 2003-11-25 | 2003-11-25 | Tablet containing citalopram hydrogen bromide |
PCT/HU2004/000110 WO2005051374A1 (en) | 2003-11-25 | 2004-11-24 | Tablets of citalopram hydrobromide |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200600932A1 true EA200600932A1 (ru) | 2006-10-27 |
EA010290B1 EA010290B1 (ru) | 2008-08-29 |
Family
ID=89981808
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200600932A EA010290B1 (ru) | 2003-11-25 | 2004-11-24 | Таблетки циталопрама гидробромида |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP1694321A1 (ru) |
BG (1) | BG109587A (ru) |
CZ (1) | CZ2006376A3 (ru) |
EA (1) | EA010290B1 (ru) |
HU (1) | HU227491B1 (ru) |
PL (1) | PL379864A1 (ru) |
SK (1) | SK50532006A3 (ru) |
UA (1) | UA83094C2 (ru) |
WO (1) | WO2005051374A1 (ru) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI358407B (en) * | 2005-06-22 | 2012-02-21 | Lundbeck & Co As H | Crystalline base of escitalopram and orodispersibl |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6607751B1 (en) * | 1997-10-10 | 2003-08-19 | Intellipharamaceutics Corp. | Controlled release delivery device for pharmaceutical agents incorporating microbial polysaccharide gum |
IES20010693A2 (en) * | 2000-08-10 | 2002-07-10 | Lundbeck & Co As H | Pharmaceutical composition containing citalopram |
AU2001100195B4 (en) * | 2001-01-05 | 2001-12-20 | H Lundbeck As | Pharmaceutical composition containing citalopram. |
-
2003
- 2003-11-25 HU HU0303790A patent/HU227491B1/hu unknown
-
2004
- 2004-11-24 CZ CZ20060376A patent/CZ2006376A3/cs unknown
- 2004-11-24 UA UAA200607053A patent/UA83094C2/ru unknown
- 2004-11-24 EA EA200600932A patent/EA010290B1/ru not_active IP Right Cessation
- 2004-11-24 PL PL379864A patent/PL379864A1/pl not_active Application Discontinuation
- 2004-11-24 EP EP04798748A patent/EP1694321A1/en not_active Withdrawn
- 2004-11-24 WO PCT/HU2004/000110 patent/WO2005051374A1/en active Application Filing
- 2004-11-24 SK SK5053-2006A patent/SK50532006A3/sk not_active Application Discontinuation
-
2006
- 2006-06-23 BG BG109587A patent/BG109587A/bg unknown
Also Published As
Publication number | Publication date |
---|---|
HU227491B1 (en) | 2011-07-28 |
WO2005051374A1 (en) | 2005-06-09 |
SK50532006A3 (sk) | 2006-09-07 |
HU0303790D0 (en) | 2004-03-01 |
HUP0303790A2 (hu) | 2005-08-29 |
UA83094C2 (en) | 2008-06-10 |
CZ2006376A3 (cs) | 2006-10-11 |
EP1694321A1 (en) | 2006-08-30 |
EA010290B1 (ru) | 2008-08-29 |
PL379864A1 (pl) | 2006-11-27 |
BG109587A (bg) | 2006-12-29 |
HUP0303790A3 (en) | 2005-09-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM |
|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): RU |