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EA200400254A1 - Трициклические имидазопиридины - Google Patents

Трициклические имидазопиридины

Info

Publication number
EA200400254A1
EA200400254A1 EA200400254A EA200400254A EA200400254A1 EA 200400254 A1 EA200400254 A1 EA 200400254A1 EA 200400254 A EA200400254 A EA 200400254A EA 200400254 A EA200400254 A EA 200400254A EA 200400254 A1 EA200400254 A1 EA 200400254A1
Authority
EA
Eurasian Patent Office
Prior art keywords
imidazopiridines
tricyclic
international
compounds
application
Prior art date
Application number
EA200400254A
Other languages
English (en)
Other versions
EA007683B1 (ru
Inventor
Петер Ян Циммерманн
Вольфганг-Александер Зимон
Штефан Постиус
Вольфганг Кромер
Original Assignee
Алтана Фарма Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Алтана Фарма Аг filed Critical Алтана Фарма Аг
Publication of EA200400254A1 publication Critical patent/EA200400254A1/ru
Publication of EA007683B1 publication Critical patent/EA007683B1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14—Ortho-condensed systems
    • C07D491/147—Ortho-condensed systems the condensed system containing one ring with oxygen as ring hetero atom and two rings with nitrogen as ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

В заявке описаны соединения формулы 1, в которой заместители и символы имеют значения, указанные в описании. Эти соединения ингибируют выделение желудочного сока.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200400254A 2001-08-10 2002-07-31 Трициклические имидазопиридины EA007683B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01119321 2001-08-10
PCT/EP2002/008505 WO2003014123A1 (en) 2001-08-10 2002-07-31 Tricyclic imidazopyridines

Publications (2)

Publication Number Publication Date
EA200400254A1 true EA200400254A1 (ru) 2004-08-26
EA007683B1 EA007683B1 (ru) 2006-12-29

Family

ID=8178292

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200400254A EA007683B1 (ru) 2001-08-10 2002-07-31 Трициклические имидазопиридины

Country Status (24)

Country Link
US (1) US7223771B2 (ru)
EP (1) EP1419163B9 (ru)
JP (1) JP2005504761A (ru)
KR (1) KR20040023739A (ru)
CN (1) CN1329395C (ru)
AT (1) ATE297931T1 (ru)
BR (1) BR0211826A (ru)
CA (1) CA2452803A1 (ru)
DE (1) DE60204701T2 (ru)
DK (1) DK1419163T5 (ru)
EA (1) EA007683B1 (ru)
ES (1) ES2243788T3 (ru)
HR (1) HRP20040229A2 (ru)
HU (1) HUP0500330A3 (ru)
IL (1) IL159554A0 (ru)
MX (1) MXPA04001277A (ru)
NO (1) NO20040604L (ru)
NZ (1) NZ531520A (ru)
PL (1) PL368195A1 (ru)
PT (1) PT1419163E (ru)
SI (1) SI1419163T1 (ru)
TW (1) TWD111798S1 (ru)
WO (1) WO2003014123A1 (ru)
ZA (1) ZA200400918B (ru)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA05010310A (es) 2003-04-04 2005-11-17 Altana Pharma Ag Bencimidazoles ciclicos.
AR044129A1 (es) 2003-05-06 2005-08-24 Altana Pharma Ag Compuestos intermedios de imidazopiridina. proceso de preparacion.
AU2004243444A1 (en) * 2003-05-27 2004-12-09 Altana Pharma Ag Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility
EP1697358A1 (en) * 2003-12-19 2006-09-06 Altana Pharma AG Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
AR046941A1 (es) * 2003-12-19 2006-01-04 Altana Pharma Ag Imidazopiridinas triciclicas y su uso como inhibidores de secrecion de acido gastrico
AR047605A1 (es) * 2004-02-17 2006-01-25 Altana Pharma Ag Imidazopiridinas triciclicas e intermediarios en la sintesis de las mismas,sus procesos de preparacion,composiciones farmaceuticas que los contienen y usos.
EP1735318A2 (en) * 2004-03-17 2006-12-27 Altana Pharma AG 7h-8,9-dihydro-pyrano(2,3-c)imidazo(1,2a)pyridine derivatives and their use as gastric acid secretion inhibitors
WO2005090346A2 (en) * 2004-03-22 2005-09-29 Altana Pharma Ag 7, 8, 9, 10- tetrahydro-imidazo [2,1-a] isoquinoline derivatives and their use as gastric acid secretion inhibitors
AR048869A1 (es) * 2004-04-26 2006-06-07 Altana Pharma Ag Bencimidazoles triciclicos
DE602005002751T2 (de) * 2004-06-09 2008-07-17 Nycomed Gmbh Substituierte tricyclische benzimidazole
AR051041A1 (es) * 2004-10-04 2006-12-13 Altana Pharma Ag Bencimidazoles triciclicos condensados
AR054772A1 (es) * 2005-06-16 2007-07-18 Altana Pharma Ag Espiro- imidazopiridinas como inhibidores de la secrecion de acido gastrico
EP2004643A1 (en) * 2006-03-31 2008-12-24 Novartis AG Organic compounds
WO2008071766A2 (en) * 2006-12-14 2008-06-19 Nycomed Gmbh Spiro-indene substituted imidazonaphythyridine and pyranoimidazopyridine derivatives as inhibitors of gastric acid secretion
KR200452179Y1 (ko) * 2009-05-20 2011-02-10 주식회사 신성일렉스 항공 장애물 표시 장치
WO2011004882A1 (ja) 2009-07-09 2011-01-13 ラクオリア創薬株式会社 消化管運動異常が関与する疾患を治療するためのアシッドポンプ拮抗剤
GB201321730D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4468400A (en) * 1982-12-20 1984-08-28 Schering Corporation Antiulcer tricyclic imidazo [1,2-a]pyridines
SE9401197D0 (sv) * 1994-04-11 1994-04-11 Astra Ab Active compounds
EP0971922B1 (en) 1997-03-24 2004-04-28 ALTANA Pharma AG Tetrahydropyrido compounds
IL131407A0 (en) * 1997-03-24 2001-01-28 Byk Gulden Lomberg Chem Fab Tetrahydropyrido compounds medicaments containing the same and the use thereof
JP2001526703A (ja) * 1997-05-28 2001-12-18 ビイク グルデン ロンベルク ヒエーミツシエ フアブリーク ゲゼルシヤフト ミツト ベシユレンクテル ハフツング 縮合ジヒドロピラン
CN1221553C (zh) * 2000-03-29 2005-10-05 奥坦纳医药公司 三环咪唑并吡啶类化合物及药物组合物

Also Published As

Publication number Publication date
CA2452803A1 (en) 2003-02-20
EP1419163B9 (en) 2005-11-09
EP1419163B1 (en) 2005-06-15
HK1066213A1 (en) 2005-03-18
US7223771B2 (en) 2007-05-29
IL159554A0 (en) 2004-06-01
NZ531520A (en) 2005-10-28
EA007683B1 (ru) 2006-12-29
CN1541219A (zh) 2004-10-27
MXPA04001277A (es) 2004-05-27
HUP0500330A2 (hu) 2005-07-28
ZA200400918B (en) 2005-04-20
DK1419163T3 (da) 2005-10-17
PL368195A1 (en) 2005-03-21
SI1419163T1 (sl) 2005-12-31
WO2003014123A1 (en) 2003-02-20
TWD111798S1 (zh) 2006-07-11
JP2005504761A (ja) 2005-02-17
PT1419163E (pt) 2005-10-31
DE60204701T2 (de) 2006-08-03
HRP20040229A2 (en) 2005-02-28
US20050049272A1 (en) 2005-03-03
KR20040023739A (ko) 2004-03-18
DE60204701D1 (de) 2005-07-21
NO20040604L (no) 2004-02-10
HUP0500330A3 (en) 2009-12-28
ES2243788T3 (es) 2005-12-01
DK1419163T5 (da) 2005-12-19
BR0211826A (pt) 2005-06-28
CN1329395C (zh) 2007-08-01
ATE297931T1 (de) 2005-07-15
EP1419163A1 (en) 2004-05-19

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): BY RU