DK91083A - Fremgangsmaade til fremstilling af thiazol-derivater - Google Patents

Fremgangsmaade til fremstilling af thiazol-derivater Download PDF

Info

Publication number: DK91083A
Authority: DK; Denmark
Prior art keywords: sub; sup; alkyl; aryl; alkynyl
Prior art date: 1982-03-19

Application number

DK91083A

Other languages

English (en)

Other versions

DK91083D0 (da

Inventor

Richard Paul Pioch

Original Assignee

Lilly Co Eli

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-03-19

Filing date

1983-02-25

Publication date

1983-09-20

1983-02-25 Application filed by Lilly Co Eli filed Critical Lilly Co Eli

1983-02-25 Publication of DK91083D0 publication Critical patent/DK91083D0/da

1983-09-20 Publication of DK91083A publication Critical patent/DK91083A/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/194—Radicals derived from thio- or thiono carboxylic acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/28—Radicals substituted by nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Thiazole And Isothizaole Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Cephalosporin Compounds (AREA)
Treating Waste Gases (AREA)
Earth Drilling (AREA)
Inert Electrodes (AREA)
Fats And Perfumes (AREA)
Diaphragms For Electromechanical Transducers (AREA)
Supply Devices, Intensifiers, Converters, And Telemotors (AREA)

DK91083A 1982-03-19 1983-02-25 Fremgangsmaade til fremstilling af thiazol-derivater DK91083A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/360,034 US4474794A (en)	1982-03-19	1982-03-19	N-Thiazolylmethylthioalkyl-N1 -alkenyl (or alkynyl)guanidines and related compounds

Publications (2)

Publication Number	Publication Date
DK91083D0 DK91083D0 (da)	1983-02-25
DK91083A true DK91083A (da)	1983-09-20

Family

ID=23416322

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK91083A DK91083A (da)	1982-03-19	1983-02-25	Fremgangsmaade til fremstilling af thiazol-derivater

Country Status (22)

Country	Link
US (1)	US4474794A (da)
EP (1)	EP0091220B1 (da)
JP (1)	JPS58170773A (da)
KR (1)	KR840004091A (da)
AT (1)	ATE27156T1 (da)
AU (1)	AU1254583A (da)
CA (1)	CA1190547A (da)
CS (1)	CS236788B2 (da)
DD (1)	DD207376A5 (da)
DE (1)	DE3371514D1 (da)
DK (1)	DK91083A (da)
ES (1)	ES520791A0 (da)
FI (1)	FI830879A7 (da)
GB (1)	GB2116973B (da)
GR (1)	GR77882B (da)
IL (1)	IL68152A0 (da)
NZ (1)	NZ203605A (da)
PH (1)	PH18504A (da)
PL (1)	PL241066A1 (da)
PT (1)	PT76397B (da)
RO (1)	RO85385B (da)
ZA (1)	ZA831882B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0230127A1 (en) *	1985-12-18	1987-07-29	Eli Lilly And Company	Synthesis of nizatidine
EP0285681B1 (de) *	1987-04-06	1993-03-10	HEUMANN PHARMA GMBH & CO	Verfahren zur Herstellung von Nitroethenderivaten
NL9000132A (nl) *	1990-01-19	1991-08-16	Cedona Pharm Bv	Nieuwe thiazoolderivaten.
US20230349922A1 (en)	2020-08-11	2023-11-02	Université De Strasbourg	H2 Blockers Targeting Liver Macrophages for the Prevention and Treatment of Liver Disease and Cancer

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4200578A (en) *	1978-12-18	1980-04-29	Bristol-Myers Company	Thiazole derivatives
US4375547A (en) *	1980-10-02	1983-03-01	Eli Lilly And Company	N-Methyl-N'-2-([(2-dimethylaminomethyl)-4-thiazolyl]methylthio)ethyl 2-nitro-1,1-ethenediamine

1982
- 1982-03-19 US US06/360,034 patent/US4474794A/en not_active Expired - Fee Related
1983
- 1983-02-25 DK DK91083A patent/DK91083A/da not_active Application Discontinuation
- 1983-03-16 GR GR70814A patent/GR77882B/el unknown
- 1983-03-16 DE DE8383301461T patent/DE3371514D1/de not_active Expired
- 1983-03-16 PT PT76397A patent/PT76397B/pt unknown
- 1983-03-16 CA CA000423708A patent/CA1190547A/en not_active Expired
- 1983-03-16 GB GB08307201A patent/GB2116973B/en not_active Expired
- 1983-03-16 RO RO110351A patent/RO85385B/ro unknown
- 1983-03-16 EP EP83301461A patent/EP0091220B1/en not_active Expired
- 1983-03-16 FI FI830879A patent/FI830879A7/fi not_active Application Discontinuation
- 1983-03-16 IL IL68152A patent/IL68152A0/xx unknown
- 1983-03-16 AT AT83301461T patent/ATE27156T1/de not_active IP Right Cessation
- 1983-03-17 DD DD83248911A patent/DD207376A5/de unknown
- 1983-03-17 PH PH28661A patent/PH18504A/en unknown
- 1983-03-17 AU AU12545/83A patent/AU1254583A/en not_active Abandoned
- 1983-03-17 ZA ZA831882A patent/ZA831882B/xx unknown
- 1983-03-17 JP JP58047005A patent/JPS58170773A/ja active Pending
- 1983-03-17 KR KR1019830001082A patent/KR840004091A/ko not_active Abandoned
- 1983-03-17 NZ NZ203605A patent/NZ203605A/en unknown
- 1983-03-17 PL PL24106683A patent/PL241066A1/xx unknown
- 1983-03-18 ES ES520791A patent/ES520791A0/es active Granted
1984
- 1984-03-16 CS CS831821A patent/CS236788B2/cs unknown

Also Published As

Publication number	Publication date
PL241066A1 (en)	1985-01-02
US4474794A (en)	1984-10-02
IL68152A0 (en)	1983-06-15
GR77882B (da)	1984-09-25
FI830879L (fi)	1983-09-20
PH18504A (en)	1985-08-02
ES8405386A1 (es)	1984-06-01
FI830879A7 (fi)	1983-09-20
GB2116973B (en)	1985-08-29
EP0091220A2 (en)	1983-10-12
NZ203605A (en)	1985-10-11
DK91083D0 (da)	1983-02-25
DD207376A5 (de)	1984-02-29
EP0091220A3 (en)	1984-05-23
CA1190547A (en)	1985-07-16
GB8307201D0 (en)	1983-04-20
ES520791A0 (es)	1984-06-01
RO85385A (ro)	1984-11-25
AU1254583A (en)	1983-09-22
PT76397A (en)	1983-04-01
EP0091220B1 (en)	1987-05-13
RO85385B (ro)	1984-11-30
FI830879A0 (fi)	1983-03-16
ZA831882B (en)	1984-11-28
KR840004091A (ko)	1984-10-06
PT76397B (en)	1986-02-04
DE3371514D1 (en)	1987-06-19
GB2116973A (en)	1983-10-05
JPS58170773A (ja)	1983-10-07
CS236788B2 (en)	1985-05-15
ATE27156T1 (de)	1987-05-15

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Legal Events

Date	Code	Title	Description
1985-11-11	AHB	Application shelved due to non-payment