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DK3546456T3 - Krystal af pyrido[3, 4-d]pyrimidinderivat eller solvat deraf - Google Patents

Krystal af pyrido[3, 4-d]pyrimidinderivat eller solvat deraf Download PDF

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Publication number
DK3546456T3
DK3546456T3 DK17873876.1T DK17873876T DK3546456T3 DK 3546456 T3 DK3546456 T3 DK 3546456T3 DK 17873876 T DK17873876 T DK 17873876T DK 3546456 T3 DK3546456 T3 DK 3546456T3
Authority
DK
Denmark
Prior art keywords
pyrido
solvate
crystal
pyrimidine derivative
pyrimidine
Prior art date
Application number
DK17873876.1T
Other languages
English (en)
Inventor
Hidetoshi Miyamoto
Tsuyoshi Mizuno
Gen Unoki
Yuki Miyazawa
Naoki Yajima
Original Assignee
Teijin Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teijin Pharma Ltd filed Critical Teijin Pharma Ltd
Application granted granted Critical
Publication of DK3546456T3 publication Critical patent/DK3546456T3/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Vascular Medicine (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Walking Sticks, Umbrellas, And Fans (AREA)
DK17873876.1T 2016-11-28 2017-11-27 Krystal af pyrido[3, 4-d]pyrimidinderivat eller solvat deraf DK3546456T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2016229973 2016-11-28
PCT/JP2017/042437 WO2018097295A1 (ja) 2016-11-28 2017-11-27 ピリド[3,4-d]ピリミジン誘導体又はその溶媒和物の結晶

Publications (1)

Publication Number Publication Date
DK3546456T3 true DK3546456T3 (da) 2022-03-07

Family

ID=62196036

Family Applications (1)

Application Number Title Priority Date Filing Date
DK17873876.1T DK3546456T3 (da) 2016-11-28 2017-11-27 Krystal af pyrido[3, 4-d]pyrimidinderivat eller solvat deraf

Country Status (30)

Country Link
US (1) US11261182B2 (da)
EP (1) EP3546456B1 (da)
JP (2) JP6745905B2 (da)
KR (1) KR102352637B1 (da)
CN (1) CN109996800B (da)
AU (1) AU2017364805B2 (da)
CA (1) CA3041854C (da)
CL (3) CL2019001420A1 (da)
CO (1) CO2019005513A2 (da)
CY (1) CY1125045T1 (da)
DK (1) DK3546456T3 (da)
EC (1) ECSP19037197A (da)
ES (1) ES2905437T3 (da)
HR (1) HRP20220065T1 (da)
HU (1) HUE057706T2 (da)
IL (1) IL266313B2 (da)
LT (1) LT3546456T (da)
MA (1) MA45887B1 (da)
MX (1) MX382362B (da)
MY (1) MY199852A (da)
PE (2) PE20191133A1 (da)
PH (1) PH12019500905A1 (da)
PL (1) PL3546456T3 (da)
PT (1) PT3546456T (da)
RS (1) RS63004B1 (da)
SI (1) SI3546456T1 (da)
TW (1) TWI755452B (da)
UA (1) UA124273C2 (da)
WO (1) WO2018097295A1 (da)
ZA (1) ZA201902828B (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023109959A1 (zh) * 2021-12-16 2023-06-22 药捷安康(南京)科技股份有限公司 Cdk9抑制剂及其用途
WO2025070601A1 (ja) * 2023-09-27 2025-04-03 帝人ファーマ株式会社 関節リウマチ治療薬

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL220952B1 (pl) 2002-01-22 2016-01-29 Warner Lambert Co 2-(Pirydyn-2-yloamino)pirydo[2,3-d]pirymidyn-7-ony
BRPI0406809A (pt) * 2003-01-17 2005-12-27 Warner Lambert Co Heterociclos substituìdos de 2-aminopiridina como inibidores da proliferação celular
ATE412650T1 (de) * 2003-07-11 2008-11-15 Warner Lambert Co Isethionat salz eines selektiven cdk4 inhibitors
PE20110419A1 (es) 2008-08-22 2011-07-13 Novartis Ag Compuestos de pirrolo-pirimidina como inhibidores de cdk
GB201216017D0 (en) 2012-09-07 2012-10-24 Cancer Rec Tech Ltd Inhibitor compounds
NZ718190A (en) * 2013-08-23 2017-10-27 Neupharma Inc Substituted quinazolines for inhibiting kinase activity
GB201403536D0 (en) * 2014-02-28 2014-04-16 Cancer Rec Tech Ltd Inhibitor compounds
TR201819419T4 (tr) * 2014-05-29 2019-01-21 Taiho Pharmaceutical Co Ltd Yeni tetrahidropiridopirimidin bileşiği veya tuzu.
CA2961610A1 (en) 2014-09-17 2016-03-24 Quanticel Pharmaceuticals, Inc. Histone demethylase inhibitors
PT3305785T (pt) * 2015-05-29 2021-10-13 Teijin Pharma Ltd Derivado de pirido[3,4-d]pirimidina e seu sal farmaceuticamente aceitável

Also Published As

Publication number Publication date
IL266313B1 (en) 2023-08-01
HRP20220065T1 (hr) 2022-04-15
AU2017364805A2 (en) 2019-10-24
EP3546456A4 (en) 2020-04-29
CY1125045T1 (el) 2023-03-24
MA45887A1 (fr) 2020-11-30
JPWO2018097295A1 (ja) 2019-06-24
LT3546456T (lt) 2022-03-10
EP3546456B1 (en) 2022-01-12
BR112019009448A2 (pt) 2019-07-30
KR20190067247A (ko) 2019-06-14
SI3546456T1 (sl) 2022-04-29
MY199852A (en) 2023-11-25
PE20250397A1 (es) 2025-02-11
WO2018097295A1 (ja) 2018-05-31
ECSP19037197A (es) 2019-06-30
MX382362B (es) 2025-03-13
PL3546456T3 (pl) 2022-05-02
UA124273C2 (uk) 2021-08-18
JP7149980B2 (ja) 2022-10-07
CN109996800A (zh) 2019-07-09
CA3041854A1 (en) 2018-05-31
PE20191133A1 (es) 2019-09-02
ZA201902828B (en) 2022-05-25
AU2017364805B2 (en) 2021-12-16
HUE057706T2 (hu) 2022-05-28
JP6745905B2 (ja) 2020-08-26
IL266313A (en) 2019-06-30
IL266313B2 (en) 2023-12-01
PH12019500905A1 (en) 2019-08-19
NZ752990A (en) 2025-08-29
CL2019001420A1 (es) 2019-08-30
CL2021001448A1 (es) 2022-01-14
EP3546456A1 (en) 2019-10-02
CN109996800B (zh) 2021-11-19
ES2905437T3 (es) 2022-04-08
CL2021001447A1 (es) 2022-01-14
KR102352637B1 (ko) 2022-01-17
RU2019116389A3 (da) 2021-04-16
CO2019005513A2 (es) 2019-07-31
TW201833105A (zh) 2018-09-16
MA45887B1 (fr) 2021-04-30
RU2019116389A (ru) 2020-11-30
RS63004B1 (sr) 2022-03-31
AU2017364805A1 (en) 2019-05-09
PT3546456T (pt) 2022-02-28
US20210276997A1 (en) 2021-09-09
MX2019005717A (es) 2019-08-12
JP2020121989A (ja) 2020-08-13
TWI755452B (zh) 2022-02-21
US11261182B2 (en) 2022-03-01
CA3041854C (en) 2025-05-13

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