DK3097081T3 - Fremgangsmåde til fremstilling af 1-alkyl-3-difluormethyl-5-fluor-1h-pyrazol-4-carbaldehyder og 1-alkyl-3-difluormethyl-5-fluor-1h-pyrazol-4-carboxylater - Google Patents
Fremgangsmåde til fremstilling af 1-alkyl-3-difluormethyl-5-fluor-1h-pyrazol-4-carbaldehyder og 1-alkyl-3-difluormethyl-5-fluor-1h-pyrazol-4-carboxylaterInfo
- Publication number
- DK3097081T3 DK3097081T3 DK15700749.3T DK15700749T DK3097081T3 DK 3097081 T3 DK3097081 T3 DK 3097081T3 DK 15700749 T DK15700749 T DK 15700749T DK 3097081 T3 DK3097081 T3 DK 3097081T3
- Authority
- DK
- Denmark
- Prior art keywords
- difluormethyl
- fluor
- alkyl
- carbaldehyder
- pyrazyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14356001 | 2014-01-24 | ||
| PCT/EP2015/051184 WO2015110493A1 (en) | 2014-01-24 | 2015-01-22 | Method for preparing 1-alkyl-3-difluoromethyl-5-fluor-1h-pyrazole-4-carbaldehydes and 1-alkyl-3-difluoromethyl-5-fluor-1h-pyrazole-4-carboxylates |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK3097081T3 true DK3097081T3 (da) | 2018-01-29 |
Family
ID=50073123
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK15700749.3T DK3097081T3 (da) | 2014-01-24 | 2015-01-22 | Fremgangsmåde til fremstilling af 1-alkyl-3-difluormethyl-5-fluor-1h-pyrazol-4-carbaldehyder og 1-alkyl-3-difluormethyl-5-fluor-1h-pyrazol-4-carboxylater |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US9656966B2 (da) |
| EP (1) | EP3097081B1 (da) |
| JP (1) | JP6462703B2 (da) |
| KR (1) | KR102319577B1 (da) |
| CN (1) | CN105934430B (da) |
| BR (1) | BR112016016397B1 (da) |
| DK (1) | DK3097081T3 (da) |
| ES (1) | ES2657424T3 (da) |
| IL (1) | IL246870B (da) |
| MX (1) | MX361770B (da) |
| TW (1) | TWI628168B (da) |
| WO (1) | WO2015110493A1 (da) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN109694350B (zh) * | 2017-10-20 | 2023-05-09 | 中国科学院上海有机化学研究所 | 一种含氟甲基的化合物及其制备方法 |
| TWI782599B (zh) * | 2020-07-02 | 2022-11-01 | 美商輝瑞股份有限公司 | 胺基嘧啶基衍生物 |
| AR122756A1 (es) * | 2020-07-02 | 2022-10-05 | Pfizer | Preparación de un derivado de pirimidinil-3,8-diazabiciclo[3.2.1]octanilmetanona y sal de este |
| WO2022233129A1 (en) | 2021-05-05 | 2022-11-10 | Fujian Yongjing Technology Co., Ltd | New process for the synthesis of 5-fluoro-3- (difuoromethyl) -5-fluoro-1-methyl-1h-pyrazole-4-carboxylic acid derivatives and the free acid thereof |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5658962A (en) * | 1994-05-20 | 1997-08-19 | Minnesota Mining And Manufacturing Company | Omega-hydrofluoroalkyl ethers, precursor carboxylic acids and derivatives thereof, and their preparation and application |
| US7396850B2 (en) | 2003-01-06 | 2008-07-08 | Eli Lilly And Company | Pyrazole derivative as PPAR modulator |
| PL1781662T3 (pl) | 2004-08-18 | 2011-08-31 | Pfizer | Inhibitory zależnej od RNA polimerazy RNA wirusa zapalenia wątroby typu C, i kompozycje i terapie wykorzystujące je |
| GB0428137D0 (en) * | 2004-12-22 | 2005-01-26 | Syngenta Participations Ag | Novel herbicides |
| DE102005009457A1 (de) * | 2005-03-02 | 2006-09-07 | Bayer Cropscience Ag | Verfahren zum Herstellen von Alkylaniliden |
| EP1721899A1 (en) * | 2005-05-13 | 2006-11-15 | Bayer CropScience S.A. | Process for the preparation of a carboxamide derivative |
| WO2008006540A1 (en) * | 2006-07-12 | 2008-01-17 | Syngenta Participations Ag | Triazolopyridine derivatives as herbicides |
| GB0813436D0 (en) * | 2008-07-22 | 2008-08-27 | Syngenta Participations Ag | Insecticidal compounds |
| AR076839A1 (es) * | 2009-05-15 | 2011-07-13 | Bayer Cropscience Ag | Derivados fungicidas de pirazol carboxamidas |
| EP2325173A1 (de) | 2009-11-19 | 2011-05-25 | Bayer CropScience AG | Verfahren zum Herstellen von 5-Fluor-1-alkyl-3-fluoralkyl-1H-pyrazol-4-carbonsäurechloriden |
| BR112012027170B1 (pt) | 2010-04-23 | 2018-02-14 | Bayer Intellectual Property Gmbh | Processo para a preparação de cloretos e fluoretos de 5-fluoro-1-alquil-3-fluoroalquil-1h- pirazol-4-carbonila, bem como compostos intermediários dos mesmos |
| JP5889299B2 (ja) * | 2010-07-23 | 2016-03-22 | ソルヴェイ（ソシエテ アノニム） | １−置換−３−フルオロアルキル−ピラゾール−４−カルボン酸のエステルの調製方法 |
| JP5854049B2 (ja) * | 2011-01-28 | 2016-02-09 | 日本電気株式会社 | 通信システム、制御情報中継装置、制御装置、制御情報の送信方法およびプログラム |
| US9145369B2 (en) | 2012-05-14 | 2015-09-29 | Bayer Cropscience Ag | Process for preparing 1-alkyl-3-fluoroalkyl-1H-pyrazole-4-carboxylic acid chlorides |
-
2015
- 2015-01-22 KR KR1020167023073A patent/KR102319577B1/ko active Active
- 2015-01-22 JP JP2016547519A patent/JP6462703B2/ja not_active Expired - Fee Related
- 2015-01-22 CN CN201580005766.1A patent/CN105934430B/zh not_active Expired - Fee Related
- 2015-01-22 EP EP15700749.3A patent/EP3097081B1/en active Active
- 2015-01-22 MX MX2016009325A patent/MX361770B/es active IP Right Grant
- 2015-01-22 BR BR112016016397-4A patent/BR112016016397B1/pt not_active IP Right Cessation
- 2015-01-22 ES ES15700749.3T patent/ES2657424T3/es active Active
- 2015-01-22 WO PCT/EP2015/051184 patent/WO2015110493A1/en active Application Filing
- 2015-01-22 US US15/113,377 patent/US9656966B2/en active Active
- 2015-01-22 DK DK15700749.3T patent/DK3097081T3/da active
- 2015-01-23 TW TW104102409A patent/TWI628168B/zh active
-
2016
- 2016-07-21 IL IL246870A patent/IL246870B/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| TWI628168B (zh) | 2018-07-01 |
| KR102319577B1 (ko) | 2021-10-29 |
| MX2016009325A (es) | 2016-10-13 |
| JP6462703B2 (ja) | 2019-01-30 |
| KR20160111506A (ko) | 2016-09-26 |
| EP3097081A1 (en) | 2016-11-30 |
| CN105934430A (zh) | 2016-09-07 |
| US20170008852A1 (en) | 2017-01-12 |
| ES2657424T3 (es) | 2018-03-05 |
| MX361770B (es) | 2018-12-17 |
| IL246870B (en) | 2018-03-29 |
| TW201615625A (zh) | 2016-05-01 |
| BR112016016397B1 (pt) | 2021-06-29 |
| JP2017506219A (ja) | 2017-03-02 |
| CN105934430B (zh) | 2018-03-16 |
| US9656966B2 (en) | 2017-05-23 |
| WO2015110493A1 (en) | 2015-07-30 |
| EP3097081B1 (en) | 2018-01-10 |
| BR112016016397A2 (pt) | 2018-12-26 |
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