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DK260881A - Bis- og mono-kvaternaere ammoniumderivater af 2beta, 16beta-diperidino-5alfa-androstaner fremgangsmaade til fremstilling deraf samt farmaceutiske praeparater indeholdende androstanforbindelserne - Google Patents

Bis- og mono-kvaternaere ammoniumderivater af 2beta, 16beta-diperidino-5alfa-androstaner fremgangsmaade til fremstilling deraf samt farmaceutiske praeparater indeholdende androstanforbindelserne

Info

Publication number
DK260881A
DK260881A DK260881A DK260881A DK260881A DK 260881 A DK260881 A DK 260881A DK 260881 A DK260881 A DK 260881A DK 260881 A DK260881 A DK 260881A DK 260881 A DK260881 A DK 260881A
Authority
DK
Denmark
Prior art keywords
ammonium derivatives
androstanes
preparing
pharmaceutical preparations
diperidino
Prior art date
Application number
DK260881A
Other languages
English (en)
Other versions
DK158741B (da
DK158741C (da
Inventor
J Kelder
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nv filed Critical Akzo Nv
Publication of DK260881A publication Critical patent/DK260881A/da
Publication of DK158741B publication Critical patent/DK158741B/da
Application granted granted Critical
Publication of DK158741C publication Critical patent/DK158741C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK260881A 1979-12-12 1981-06-15 Analogifremgangsmaade til fremstilling af biskvaternaere ammoniumderivater af 2beta,16beta-dipiperidino-5alfa-androstaner DK158741C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB7942883 1979-12-12
GB7942883 1979-12-12
EP8000143 1980-12-09
PCT/EP1980/000143 WO1981001710A1 (en) 1979-12-12 1980-12-09 Mono and bis piperidinium androstanes derivatives

Publications (3)

Publication Number Publication Date
DK260881A true DK260881A (da) 1981-06-25
DK158741B DK158741B (da) 1990-07-09
DK158741C DK158741C (da) 1990-11-26

Family

ID=10509800

Family Applications (1)

Application Number Title Priority Date Filing Date
DK260881A DK158741C (da) 1979-12-12 1981-06-15 Analogifremgangsmaade til fremstilling af biskvaternaere ammoniumderivater af 2beta,16beta-dipiperidino-5alfa-androstaner

Country Status (12)

Country Link
US (1) US4348390A (da)
EP (1) EP0032261B1 (da)
JP (1) JPH026360B2 (da)
AU (1) AU534992B2 (da)
CA (1) CA1153366A (da)
DE (1) DE3065088D1 (da)
DK (1) DK158741C (da)
ES (1) ES8204443A1 (da)
FI (1) FI66394C (da)
HU (1) HU185865B (da)
IE (1) IE50675B1 (da)
WO (1) WO1981001710A1 (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE53463B1 (en) * 1981-06-15 1988-11-23 Akzo Nv Mono-and bisquaternary ammonium derivatives of 2 beta,16 beta-d-amino-5 alpha-androstane derivatives and pharmaceutical preparations containing same
US4726275A (en) * 1983-05-10 1988-02-23 Synthaxe Limited Electronic musical instrument
US5418226A (en) * 1992-04-22 1995-05-23 Akzo N.V. Monoquaternary 2,16-bispiperidinylandrostane derivatives
US5926516A (en) * 1995-05-24 1999-07-20 Siemens Aktiengesellschaft Absorption structure for absorbing neutrons and method for producing an absorption structure
IT1277700B1 (it) * 1995-12-22 1997-11-11 Poli Ind Chimica Spa Processo di preparazione di 2-beta, 16-beta-diamino 3-alfa, 17-beta- diacilossi 5-alfaandrostani, bloccanti neuromuscolari a struttura
US5990124A (en) * 1997-10-24 1999-11-23 Gyermek; Laszlo Neuromuscular relaxants
CN116925171A (zh) * 2023-07-10 2023-10-24 时森海(杭州)医药科技有限公司 含环丙甲基甾体类季铵盐化合物、中间体及其制备方法和应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1138605A (en) * 1965-02-19 1969-01-01 Organon Labor Ltd Improvements in or relating to new 2-ß,16-ß-diamino-androstanes
GB1454749A (en) * 1972-11-29 1976-11-03 Akzo Nv 2beta, 16beta-diamino-androstanes and their preparation
HU172522B (hu) * 1975-08-01 1978-09-28 Richter Gedeon Vegyeszet Sposob poluchenija novykh proizvodnykh 2beta, 16beta-diamino-androstana i ikh chetvertichnykh solej
DE2962627D1 (en) * 1978-09-05 1982-06-09 Akzo Nv Acid addition salts of 16-beta-monoquaternary ammonium derivatives of 2-beta, 16-beta-bis-piperidino-androstanes and pharmaceutical preparations containing same

Also Published As

Publication number Publication date
HU185865B (en) 1985-04-28
WO1981001710A1 (en) 1981-06-25
EP0032261A1 (en) 1981-07-22
IE802566L (en) 1981-06-12
FI66394C (fi) 1984-10-10
JPH026360B2 (da) 1990-02-08
JPS56501761A (da) 1981-12-03
FI811857L (fi) 1981-06-15
AU6640581A (en) 1981-07-06
AU534992B2 (en) 1984-02-23
DK158741B (da) 1990-07-09
DE3065088D1 (en) 1983-11-03
ES497724A0 (es) 1982-05-01
EP0032261B1 (en) 1983-09-28
IE50675B1 (en) 1986-06-11
CA1153366A (en) 1983-09-06
US4348390A (en) 1982-09-07
FI66394B (fi) 1984-06-29
ES8204443A1 (es) 1982-05-01
DK158741C (da) 1990-11-26

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Legal Events

Date Code Title Description
PBP Patent lapsed